Target Details
| UniProt AC | P11362 |
|---|---|
| Gene Symbol | FGFR1 |
| Protein Name | Fibroblast growth factor receptor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF00047 (ig) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 3,320
- Clinical molecules 348
- Avg pChEMBL 7.53
KEGG Pathways (18)
- Adherens junction
- Breast cancer
- Cadherin signaling
- Calcium signaling pathway
- Central carbon metabolism in cancer
- IgSF CAM signaling
- MAPK signaling pathway
- Melanoma
- PI3K-Akt signaling pathway
- Parathyroid hormone synthesis, secretion and action
- Pathways in cancer
- Prostate cancer
- Proteoglycans in cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
- Signaling pathways regulating pluripotency of stem cells
- Thermogenesis
Associated Diseases (8)
Active Molecules (3,320)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HRSOTZFHFDXFAE
|
9.2 | IC50 | 5 | — | |
RVYNZDFXTZHHFU
|
9.2 | IC50 | 2 | — | |
SECZNHBHHKOBMC
|
9.2 | IC50 | 2 | — | |
QPQVFVWZSRRLKL
|
9.2 | IC50 | 2 | — | |
CERLJSLIKVDHSK
|
9.2 | IC50 | 2 | — | |
HMJWDRNCIBKVLK
|
9.2 | IC50 | 2 | — | |
IBHARKZDQBGJAJ
|
9.2 | IC50 | 2 | — | |
LBKNXKHZVKUMAV
|
9.2 | IC50 | 2 | — | |
PUIXMSRTTHLNKI
|
9.2 | IC50 | 12 | — | |
UJKFLFOBPZHDJN
|
9.2 | IC50 | 3 | — | |
VDTUZTRVIPIQEC
|
9.2 | Kd | 3 | — | |
ZMYXCQOKPQVAIY
|
9.2 | IC50 | 2 | — | |
ZQTUTQJCMVRZQW
|
9.2 | IC50 | 2 | — | |
GTZRCWSMTBJVNU
|
9.2 | IC50 | 3 | — | |
SPXNVPJERGMJSD
|
9.2 | IC50 | 3 | — | |
XFZJRMKUNDQXMW
|
9.2 | IC50 | 5 | — | |
AKNCKKKGJAAVEH
|
9.2 | IC50 | 2 | — | |
BRGNIALEUFSUFN
|
9.2 | IC50 | 3 | — | |
CUUBVEXZVSAYPH
|
9.2 | IC50 | 2 | — | |
DIVGFMHEBBBJGH
|
9.2 | IC50 | 2 | — | |
DLLAXFDTFVKUAV
|
9.2 | IC50 | 2 | — | |
GWOHWBYOVFLZGM
|
9.2 | IC50 | 2 | — | |
WAZQJIQKCRAOBX
|
9.2 | IC50 | 2 | — | |
YISJWEXLNFHRNW
|
9.2 | IC50 | 4 | — | |
MRSOJHDLCLHTOL
|
9.1 | IC50 | 5 | — | |
NMFMLTFZEUDACF
|
9.1 | IC50 | 4 | — | |
QHCGPJPIPKDWAT
|
9.1 | IC50 | 8 | — | |
ACXLCIADWYPDHD
|
9.1 | IC50 | 2 | — | |
BYEGVFRRTLAAQA
|
9.1 | IC50 | 2 | — | |
DOWBTQHWXGZIER
|
9.1 | IC50 | 2 | — | |
GMNMMGZZBZYAMO
|
9.1 | IC50 | 2 | — | |
HUVVCRLMPWOMJX
|
9.1 | IC50 | 4 | — | |
JKWPSZWWCDRXFP
|
9.1 | IC50 | 2 | — | |
LJJPNXWNMVOUCI
|
9.1 | IC50 | 2 | — | |
MXSDIGYURCYKOV
|
9.1 | IC50 | 5 | — | |
PKCCJOWYVJUGKD
|
9.1 | IC50 | 3 | — | |
QWGUTUKCPRERRM
|
9.1 | IC50 | 2 | — | |
WYSRIBSZOQNKSS
|
9.1 | IC50 | 2 | — | |
KTMMZCLUGNPLAT
|
9.1 | IC50 | 3 | — | |
SIDXAOMKSAWATD
|
9.1 | IC50 | 2 | — | |
ODRNQGSZGLHVGG
|
9.1 | IC50 | 5 | — | |
QPILVXXWABVBBV
|
9.1 | IC50 | 5 | — | |
ZGQVGBIOCZBGDY
|
9.1 | IC50 | 2 | — | |
BAWZESLJEVSFRN
|
9.1 | IC50 | 6 | — | |
CGFYKMPVFSVIHD
|
9.1 | IC50 | 2 | — | |
CVTLXZHZCMNAPK
|
9.1 | Kd | 3 | — | |
FVECKDIACHPELI
|
9.1 | IC50 | 2 | — | |
GEMHNNGOAKEHGC
|
9.1 | IC50 | 2 | — | |
GRJFVVYLSWWNRI
|
9.1 | IC50 | 2 | — | |
KBUPLPBZRGPNCS
|
9.1 | IC50 | 2 | — |