Target Details
| UniProt AC | P11362 |
|---|---|
| Gene Symbol | FGFR1 |
| Protein Name | Fibroblast growth factor receptor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF00047 (ig) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 3,320
- Clinical molecules 348
- Avg pChEMBL 7.53
KEGG Pathways (18)
- Adherens junction
- Breast cancer
- Cadherin signaling
- Calcium signaling pathway
- Central carbon metabolism in cancer
- IgSF CAM signaling
- MAPK signaling pathway
- Melanoma
- PI3K-Akt signaling pathway
- Parathyroid hormone synthesis, secretion and action
- Pathways in cancer
- Prostate cancer
- Proteoglycans in cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
- Signaling pathways regulating pluripotency of stem cells
- Thermogenesis
Associated Diseases (8)
Active Molecules (3,320)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
ZAPUSNWRFJVSGX
|
8.4 | IC50 | 5 | — | |
BAUFTYOWRVUSNA
|
8.4 | IC50 | 2 | — | |
GJZVBYXLNIFOGB
|
8.4 | IC50 | 2 | — | |
KFKYFVCBOAGDTP
|
8.4 | IC50 | 3 | — | |
LBNJJAOYBCVITR
|
8.4 | IC50 | 2 | — | |
MKWMZFFPSBNEIH
|
8.4 | IC50 | 2 | — | |
SFYNOFFYMQHBAL
|
8.4 | IC50 | 4 | — | |
SXANNSUWWUIUKO
|
8.4 | IC50 | 2 | — | |
SXYFYNVZTYNDKV
|
8.4 | IC50 | 5 | — | |
UKAGLCCFNDEZAF
|
8.4 | IC50 | 2 | — | |
ZAWBYXATEBIOBQ
|
8.4 | IC50 | 5 | — | |
CJVVXRNKGDZSSX
|
8.3 | IC50 | 3 | — | |
KVOZGEJRFWGHFZ
|
8.3 | IC50 | 4 | — | |
NGLRSTVZLVHSJO
|
8.3 | IC50 | 5 | — | |
QIPJHJWIOASAOJ
|
8.3 | IC50 | 2 | — | |
SBMIDSNPTHVUMU
|
8.3 | IC50 | 2 | — | |
VJRPDSCCZRPRJC
|
8.3 | IC50 | 4 | — | |
BHTIIMSZAXKDLF
|
8.3 | IC50 | 2 | — | |
IGXJTXDPMDXZJZ
|
8.3 | IC50 | 3 | — | |
MCCRDQXDXGETPQ
|
8.3 | IC50 | 5 | — | |
MZLXXVIDRYUZIM
|
8.3 | IC50 | 5 | — | |
NYIBFGMWXRONJG
|
8.3 | IC50 | 2 | — | |
POKUGRIXYDIRKM
|
8.3 | IC50 | 3 | — | |
FFMFQCPBWNBRTM
|
8.3 | IC50 | 2 | — | |
HJJBUHHTOHQWIR
|
8.3 | IC50 | 4 | — | |
OLAHOMJCDNXHFI
|
8.3 | IC50 | 5 | — | |
FHYRHQXTHUGBJV
|
8.3 | IC50 | 4 | — | |
GHNNOOKRRJQEEH
|
8.3 | IC50 | 5 | — | |
KSQSKRYGIKNQHZ
|
8.3 | IC50 | 2 | — | |
PMWJNWXMNAKMHW
|
8.3 | IC50 | 5 | — | |
LGWVEHCWSZKUPK
|
8.3 | IC50 | 4 | — | |
VYMBMEPSKRYKBW
|
8.3 | Ki | 2 | — | |
YRIBONQFXXVSAU
|
8.3 | IC50 | 5 | — | |
AHSYHYFTUKZLCI
|
8.3 | IC50 | 5 | — | |
DXQBCGUEDOHNHP
|
8.3 | IC50 | 12 | — | |
LBHGMHQDOQYTKT
|
8.3 | IC50 | 5 | — | |
MZDGOELKRMAQFI
|
8.3 | IC50 | 2 | — | |
OGJAKSRIKBDGTD
|
8.3 | IC50 | 2 | — | |
OLAHOMJCDNXHFI
|
8.3 | IC50 | 5 | — | |
PAGYYFBXLGVGOO
|
8.3 | IC50 | 3 | — | |
PRVGMAOUBRLMGU
|
8.3 | IC50 | 4 | — | |
TVFMZRKDNNYDFP
|
8.3 | IC50 | 3 | — | |
TVUWQDLBEOZVOU
|
8.3 | Ki | 41 | — | |
TWEPCUUZZJESFX
|
8.3 | IC50 | 3 | — | |
WOGGKLMGFJJKGY
|
8.3 | IC50 | 5 | — | |
WXAXVITWIABKBN
|
8.3 | IC50 | 5 | — | |
IEZSYOTXLDGZAI
|
8.3 | Kd | 3 | — | |
NYNQETWJMMSWJX
|
8.3 | IC50 | 3 | — | |
QULAUQOGDDJGPW
|
8.3 | IC50 | 5 | — | |
RBNKCLPELCJMAS
|
8.3 | IC50 | 2 | — |