Target Details
| UniProt AC | P11362 |
|---|---|
| Gene Symbol | FGFR1 |
| Protein Name | Fibroblast growth factor receptor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF00047 (ig) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 3,320
- Clinical molecules 348
- Avg pChEMBL 7.53
KEGG Pathways (18)
- Adherens junction
- Breast cancer
- Cadherin signaling
- Calcium signaling pathway
- Central carbon metabolism in cancer
- IgSF CAM signaling
- MAPK signaling pathway
- Melanoma
- PI3K-Akt signaling pathway
- Parathyroid hormone synthesis, secretion and action
- Pathways in cancer
- Prostate cancer
- Proteoglycans in cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
- Signaling pathways regulating pluripotency of stem cells
- Thermogenesis
Associated Diseases (8)
Active Molecules (3,320)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KVNSXBAQSWMTDX
|
8.4 | IC50 | 2 | — | |
NCHRMJWKKXNHAK
|
8.4 | IC50 | 3 | — | |
NYJMVCWYBMPHTD
|
8.4 | IC50 | 4 | — | |
UJGBKUMKLLDSQI
|
8.4 | IC50 | 5 | — | |
VGVUCVKLHHCRRJ
|
8.4 | IC50 | 5 | — | |
XGETWASHPOMFBX
|
8.4 | IC50 | 3 | — | |
XMLPCBKZIXENAI
|
8.4 | IC50 | 4 | — | |
YXVDEILMUVTDMK
|
8.4 | IC50 | 3 | — | |
YZRLWPBYTMKRQR
|
8.4 | IC50 | 11 | — | |
AHEDUFSEDRFCTH
|
8.4 | IC50 | 4 | — | |
BSKSTNRPIFLDMV
|
8.4 | IC50 | 2 | — | |
GNLBGLKGCLZAOZ
|
8.4 | IC50 | 2 | — | |
HCDBDJBZIKAUDL
|
8.4 | IC50 | 2 | — | |
LKMLECIRYJPQOC
|
8.4 | IC50 | 5 | — | |
QALGNRWHDJCSGL
|
8.4 | IC50 | 2 | — | |
QXCPWDLEEJRGER
|
8.4 | IC50 | 2 | — | |
RYRVRXVRRSZALT
|
8.4 | IC50 | 5 | — | |
SGDJFAPTKOZVKU
|
8.4 | IC50 | 2 | — | |
SPQDHLUXHUIWBR
|
8.4 | IC50 | 2 | — | |
TUFWCZFZSQLLMZ
|
8.4 | IC50 | 4 | — | |
WTEYUYQDYILCNS
|
8.4 | IC50 | 5 | — | |
YEUQGBIVRQMUQR
|
8.4 | IC50 | 2 | — | |
YLXCHDHMROIYKA
|
8.4 | Kd | 3 | — | |
BRKGRQVBHFZISR
|
8.4 | pIC50 | 7 | Yes | |
BZFULTDZKYXUOC
|
8.4 | IC50 | 5 | — | |
DDSTUHINLNZIIZ
|
8.4 | pIC50 | 2 | Yes | |
IANNGBSXAWBFAQ
|
8.4 | IC50 | 2 | — | |
PTNPCFXETPRXSF
|
8.4 | IC50 | 3 | — | |
QWKBMCGLZANBBQ
|
8.4 | IC50 | 2 | — | |
UYTRUCYRZKTLND
|
8.4 | pIC50 | 2 | Yes | |
XVGFNPAYRAJLCR
|
8.4 | IC50 | 2 | — | |
ZBNZXTGUTAYRHI
|
8.4 | pIC50 | 102 | Yes | |
IOJGQJINDPXDDW
|
8.4 | IC50 | 5 | — | |
QQZSRHQZWOITQR
|
8.4 | IC50 | 4 | — | |
RVPLSKAFRYMLOL
|
8.4 | IC50 | 2 | — | |
YFCQTEWBNUGUFK
|
8.4 | IC50 | 2 | — | |
YMXQQOATOHFDLF
|
8.4 | IC50 | 5 | — | |
AVEPOXATJSYYGP
|
8.4 | IC50 | 5 | — | |
HPCVPAAIFAFKQL
|
8.4 | IC50 | 5 | — | |
KBATXXSVGCJBDV
|
8.4 | IC50 | 2 | — | |
KFGHIGPSLAQEPJ
|
8.4 | IC50 | 2 | — | |
KIKNWMSSCYMPJH
|
8.4 | IC50 | 2 | — | |
MBGRVTQYUJDPEX
|
8.4 | IC50 | 2 | — | |
MWMHYAXGYUGPBU
|
8.4 | IC50 | 5 | — | |
PPFQKJGJQXSDJS
|
8.4 | IC50 | 5 | — | |
RUUWTDVRBGAQCD
|
8.4 | IC50 | 3 | — | |
TZKBVRDEOITLRB
|
8.4 | IC50 | 7 | — | |
XPJRQSVFOCSTQP
|
8.4 | IC50 | 3 | — | |
AJQGJOSWZUAVFV
|
8.4 | IC50 | 3 | — | |
HRADXFDASOBMPX
|
8.4 | IC50 | 5 | — |