Target Details
| UniProt AC | P11362 |
|---|---|
| Gene Symbol | FGFR1 |
| Protein Name | Fibroblast growth factor receptor 1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07679 (I-set) PF00047 (ig) PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 3,320
- Clinical molecules 348
- Avg pChEMBL 7.53
KEGG Pathways (18)
- Adherens junction
- Breast cancer
- Cadherin signaling
- Calcium signaling pathway
- Central carbon metabolism in cancer
- IgSF CAM signaling
- MAPK signaling pathway
- Melanoma
- PI3K-Akt signaling pathway
- Parathyroid hormone synthesis, secretion and action
- Pathways in cancer
- Prostate cancer
- Proteoglycans in cancer
- Rap1 signaling pathway
- Ras signaling pathway
- Regulation of actin cytoskeleton
- Signaling pathways regulating pluripotency of stem cells
- Thermogenesis
Associated Diseases (8)
Active Molecules (3,320)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WHXUXVVTKNDEIG
|
10.0 | IC50 | 2 | — | |
LHWABYLWRJNIIY
|
9.9 | IC50 | 7 | — | |
UXYDXGKJWBUZOQ
|
9.8 | IC50 | 4 | — | |
WWGLOQFMJUZFTJ
|
9.7 | IC50 | 8 | — | |
YTUFDWZVYPHDSZ
|
9.7 | IC50 | 2 | — | |
FDYYKFWGYGBXLY
|
9.7 | IC50 | 4 | — | |
NSZYKHCVXAXWHM
|
9.7 | IC50 | 2 | — | |
YYMGAHUGGLEVAR
|
9.7 | IC50 | 4 | — | |
XUZLJISSHBHXIF
|
9.7 | IC50 | 2 | — | |
YTHRBLRSHNEQKN
|
9.6 | IC50 | 2 | — | |
PRXXXHCKGRNFLJ
|
9.6 | IC50 | 8 | — | |
ZXPCBIFWQMMSJO
|
9.6 | IC50 | 2 | — | |
KVXZTXINLAKEHW
|
9.6 | IC50 | 2 | — | |
ZJHASKJKRUOFBR
|
9.6 | IC50 | 2 | — | |
QMVLDDIBAIRUIH
|
9.6 | IC50 | 2 | — | |
USRVMHONXWVKPD
|
9.6 | IC50 | 4 | — | |
AKXGEYBQTHJGSZ
|
9.5 | IC50 | 2 | — | |
CTUHAAWNNBQIDY
|
9.5 | IC50 | 4 | — | |
NHFDRBXTEDBWCZ
|
9.5 | Kd | 12 | Yes | |
WJWCBGVYWUSETH
|
9.5 | IC50 | 2 | — | |
XVQAACIPBICWNT
|
9.5 | IC50 | 2 | — | |
YSMBBAKJHNAZTO
|
9.5 | IC50 | 2 | — | |
HFFXKEYAEKHCQX
|
9.5 | IC50 | 3 | — | |
ZCVBFVHTDQMQLA
|
9.5 | IC50 | 2 | — | |
FRMYRJLJMOMOEN
|
9.5 | IC50 | 2 | — | |
RKEGHFXOJUHWGF
|
9.5 | IC50 | 2 | — | |
FXDKQASVFHPYLG
|
9.5 | IC50 | 2 | — | |
FMGRQWRWTCYNKA
|
9.4 | IC50 | 5 | — | |
FZQIDLWMPZESRJ
|
9.4 | IC50 | 2 | — | |
GJWYRFYNBUUNMD
|
9.4 | IC50 | 2 | — | |
PURTYFIQUYZYMN
|
9.4 | IC50 | 2 | — | |
SFYGBVJAWPTPMZ
|
9.4 | IC50 | 2 | — | |
SSJSBIYCNYSJNH
|
9.4 | IC50 | 2 | — | |
XQENQGTVHFJEKT
|
9.4 | IC50 | 2 | — | |
FARNSAZMRIPYES
|
9.4 | IC50 | 2 | — | |
HCDMJFOHIXMBOV
|
9.4 | IC50 | 4 | — | |
JNTRATZGRSGDTJ
|
9.4 | IC50 | 2 | — | |
LPQUYUMWALKVKH
|
9.4 | IC50 | 2 | — | |
RMPLDNDYWZJAKD
|
9.4 | IC50 | 2 | — | |
AWNATJMQNZMYAX
|
9.4 | IC50 | 5 | — | |
VWRIGODGUPSDSL
|
9.4 | IC50 | 2 | — | |
CGXQXIOHFLFFRH
|
9.4 | IC50 | 4 | — | |
YWDKSGWRKAMORO
|
9.3 | IC50 | 5 | — | |
VDZZYOJYLLNBTD
|
9.3 | IC50 | 4 | — | |
MPYUMMWCLQVMLG
|
9.3 | IC50 | 11 | — | |
OWFCRBSDJKZKBD
|
9.3 | IC50 | 5 | — | |
PVLAKZNIDMGUHQ
|
9.3 | IC50 | 2 | — | |
QNXOYMFBIACDSL
|
9.3 | IC50 | 5 | — | |
XSFHSBDHUMMKQC
|
9.3 | IC50 | 4 | — | |
XTLRUHNSWCKNBK
|
9.3 | IC50 | 5 | — |