Target Details
| UniProt AC | P11309 |
|---|---|
| Gene Symbol | PIM1 |
| Protein Name | Serine/threonine-protein kinase pim-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,647
- Clinical molecules 25
- Avg pChEMBL 8.21
KEGG Pathways (5)
Active Molecules (2,647)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WYLHMLXNDVQUDF
|
9.5 | IC50 | 2 | — | |
WZGQPKOXPDHTTO
|
9.5 | IC50 | 2 | — | |
YAJGELPVDBECTQ
|
9.5 | IC50 | 2 | — | |
OUQSBZMPAZAVIV
|
9.5 | Ki | 3 | — | |
PLLDESOQBJZGSQ
|
9.5 | IC50 | 3 | — | |
QUOGNIKIMQZJJU
|
9.5 | IC50 | 3 | — | |
WLBVZYXAXNRNOX
|
9.5 | Ki | 3 | — | |
LQILNMFAVKTKBG
|
9.5 | IC50 | 2 | — | |
IQBPADAUYOSODU
|
9.5 | IC50 | 2 | — | |
PPKOMRSAECKGDB
|
9.5 | IC50 | 2 | — | |
JVWOWDAKPHFJQW
|
9.5 | Ki | 3 | — | |
NMBLJOILHIVHIT
|
9.5 | IC50 | 2 | — | |
VJXUXTWQBIILQL
|
9.5 | Ki | 3 | — | |
WRMDZFXPBIHCOL
|
9.5 | IC50 | 2 | — | |
XELTWQUXHGQCGM
|
9.5 | IC50 | 3 | — | |
ZTBXPWKLMHSULU
|
9.5 | IC50 | 2 | — | |
CPVVGAAUXSVJPE
|
9.4 | Ki | 3 | — | |
SCIFRMHWIBCWPT
|
9.4 | IC50 | 3 | — | |
ZQNLSYAFNSXFET
|
9.4 | IC50 | 2 | — | |
MZEDYGZPEWMQOQ
|
9.4 | Ki | 3 | — | |
CNQCLTYXKCWIMW
|
9.4 | IC50 | 3 | — | |
QJTHIJNIWCBEOX
|
9.4 | IC50 | 3 | — | |
JUDXZPPDZZPKEK
|
9.4 | IC50 | 3 | — | |
MYYHUGRZNUGCBD
|
9.4 | Ki | 3 | — | |
ONYPOVGNOIYPIW
|
9.4 | Ki | 3 | — | |
UKAGZEMTXTYYHX
|
9.4 | Ki | 3 | — | |
ASZCABSVZBJTKA
|
9.4 | IC50 | 3 | — | |
ATAYWLYXDVOCIF
|
9.4 | IC50 | 2 | — | |
BYFQNMWZRKKFRI
|
9.4 | IC50 | 3 | — | |
DPERSSXJBGKIEL
|
9.4 | Ki | 3 | — | |
FCGLYPSBPNFQRF
|
9.4 | IC50 | 3 | — | |
HODYSLLYOCDDRP
|
9.4 | IC50 | 2 | — | |
KRDXOKMAYHDEQM
|
9.4 | IC50 | 2 | — | |
MAODNWJWGVULBD
|
9.4 | IC50 | 3 | — | |
MCUJKPPARUPFJM
|
9.4 | IC50 | 3 | — | |
MCUJKPPARUPFJM
|
9.4 | IC50 | 11 | — | |
MLAWVMHISKOVHW
|
9.4 | IC50 | 3 | — | |
UFXCEAJTAFSFJV
|
9.4 | IC50 | 3 | — | |
UPIKPYVJDQBIIJ
|
9.4 | IC50 | 3 | — | |
UXRRXGUVXSSVLD
|
9.4 | IC50 | 2 | — | |
VDBZBBXSPQNDOH
|
9.4 | Ki | 3 | — | |
VSNMUUOHBUNKOQ
|
9.4 | IC50 | 2 | — | |
WTOWWRBBMUWWAX
|
9.4 | IC50 | 3 | — | |
YVAQXIXCFJWYDN
|
9.4 | IC50 | 2 | — | |
BMRHAWSJNXXRJI
|
9.4 | IC50 | 2 | — | |
QEULBJUCNBXCDE
|
9.4 | Ki | 3 | — | |
ZHIKDHHAKGWUBZ
|
9.4 | Ki | 3 | — | |
HIWTYESDVJEVCS
|
9.4 | Ki | 3 | — | |
LNMWCDOUCVMIEV
|
9.4 | Ki | 3 | — | |
VYVLVTDHSCQXGE
|
9.4 | Ki | 3 | — |