Target Details
| UniProt AC | P11309 |
|---|---|
| Gene Symbol | PIM1 |
| Protein Name | Serine/threonine-protein kinase pim-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,647
- Clinical molecules 25
- Avg pChEMBL 8.21
KEGG Pathways (5)
Active Molecules (2,647)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JOPRUVPDUTVSLP
|
9.7 | Ki | 3 | — | |
MFWAZGZFSFQQCU
|
9.7 | Ki | 3 | — | |
RNTZOUPFYLQDEB
|
9.7 | Ki | 3 | — | |
BUJRKYOHJDUKTN
|
9.6 | Ki | 3 | — | |
DQTHXAXXKAPXNF
|
9.6 | IC50 | 3 | — | |
PTORCEYGCGXHDH
|
9.6 | IC50 | 3 | — | |
QBCXALHYIBOFGV
|
9.6 | IC50 | 3 | — | |
WUOXBBAOJFCZKX
|
9.6 | IC50 | 3 | — | |
XERUWQHYFFRDQN
|
9.6 | IC50 | 3 | — | |
ZRNYLUKSHWKQCV
|
9.6 | IC50 | 3 | — | |
COOCHYZLHYBZPZ
|
9.6 | Ki | 3 | — | |
QVLHMFIFIGHQBW
|
9.6 | Ki | 3 | — | |
RMGUESBYRVXIQU
|
9.6 | IC50 | 2 | — | |
VMXPVSNGJHSTAJ
|
9.6 | IC50 | 2 | — | |
XKEPASMYHMOCPP
|
9.6 | IC50 | 3 | — | |
HNGYLMVBNQDLKS
|
9.6 | IC50 | 2 | — | |
IWGQMHPNGOJNRQ
|
9.6 | IC50 | 2 | — | |
LMYCHBCZOYRSRO
|
9.6 | Ki | 3 | — | |
AZVAKSGTTHXSPK
|
9.6 | IC50 | 2 | — | |
HVHOUFFQELRRFO
|
9.6 | IC50 | 2 | — | |
LKZPAYSWYUKKEK
|
9.6 | Ki | 3 | — | |
MDXOTNRTTAMQJG
|
9.6 | IC50 | 2 | — | |
NDXAAESWIVMHKZ
|
9.6 | IC50 | 2 | — | |
WKPYUMZOLALQOY
|
9.6 | Ki | 3 | — | |
XJYVGYJMUZECDN
|
9.6 | Ki | 3 | — | |
DYXVMMFGWUCEJQ
|
9.6 | Ki | 3 | — | |
CHCYABPIGAAURP
|
9.6 | Ki | 3 | — | |
CHFXZLZGCMQMBM
|
9.6 | IC50 | 3 | — | |
DWLQBQZTZFLKIC
|
9.6 | IC50 | 3 | — | |
FGLBTUNMAVXKMV
|
9.6 | IC50 | 3 | — | |
IDAHTGCAQFARTJ
|
9.6 | Ki | 3 | — | |
NHGHGBJFWZDMBT
|
9.6 | Ki | 3 | — | |
SGCVXQAEURWEAZ
|
9.6 | IC50 | 2 | — | |
AWGKTRLRSXPVMA
|
9.5 | IC50 | 2 | — | |
UEDHQXFKWCZABY
|
9.5 | Ki | 3 | — | |
UMICCZFMUZBZJG
|
9.5 | IC50 | 2 | — | |
PFVAOPOASVOPOG
|
9.5 | Ki | 3 | — | |
SWVVEDSPZBMVBS
|
9.5 | IC50 | 2 | — | |
CMCGBWKSQYENCR
|
9.5 | IC50 | 2 | — | |
DDQXBYGNFGPJRL
|
9.5 | IC50 | 3 | — | |
FGEAUESYLAVMMS
|
9.5 | IC50 | 2 | — | |
HTQXVRONIVCCQX
|
9.5 | IC50 | 3 | — | |
JYNVODGAIHNSGN
|
9.5 | IC50 | 2 | — | |
KBIGBJJRXNTKSO
|
9.5 | IC50 | 2 | — | |
MLBSKYGOXRDFII
|
9.5 | IC50 | 2 | — | |
NAJNBAVODHIQHE
|
9.5 | IC50 | 2 | — | |
QYMQRLSRAFFKQN
|
9.5 | IC50 | 2 | — | |
RBYSKZSYRQTJLG
|
9.5 | IC50 | 2 | — | |
TUMIEGHWQWSXPG
|
9.5 | IC50 | 3 | — | |
UZKVHHUKSZZZFF
|
9.5 | IC50 | 2 | — |