Target Details
| UniProt AC | P11309 |
|---|---|
| Gene Symbol | PIM1 |
| Protein Name | Serine/threonine-protein kinase pim-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,647
- Clinical molecules 25
- Avg pChEMBL 8.21
KEGG Pathways (5)
Active Molecules (2,647)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OYEPHAQZHMCGRV
|
9.8 | IC50 | 3 | — | |
QBMHBUSZNODSPS
|
9.8 | Ki | 3 | — | |
UBOPIWHFWYMNOM
|
9.8 | IC50 | 2 | — | |
UOJNFBQURVKKJP
|
9.8 | IC50 | 2 | — | |
WHGGAJVOOZRMSO
|
9.8 | Ki | 3 | — | |
ATMQYZNWXYJUNO
|
9.8 | Ki | 3 | — | |
QWBBMEBGXUMEIM
|
9.8 | Ki | 3 | — | |
RPRPMROISJUPTE
|
9.8 | Ki | 3 | — | |
GAIGYASYQJMNNF
|
9.8 | IC50 | 3 | — | |
JPOSDFHBASHSQE
|
9.8 | IC50 | 3 | — | |
LGHKQPUVKJCZNF
|
9.8 | IC50 | 3 | — | |
WVGRLEUUFBQQLW
|
9.8 | IC50 | 3 | — | |
QDSYVSQEYVFTTI
|
9.8 | Ki | 3 | — | |
QJYRTBVKAJEXQS
|
9.8 | IC50 | 2 | — | |
SSVDHMHVZBAMPA
|
9.8 | Ki | 3 | — | |
AWFOXFITUCSTPY
|
9.7 | Ki | 3 | — | |
BGXXCYLUQOQXBF
|
9.7 | IC50 | 2 | — | |
GPGQKMLTKINISD
|
9.7 | IC50 | 2 | — | |
HVZQLRXKWHBUAJ
|
9.7 | IC50 | 3 | — | |
QVQNZMJSTKPJKL
|
9.7 | IC50 | 2 | — | |
VBLIOVPAIOHWTR
|
9.7 | Ki | 3 | — | |
XUPURJISFWXKAO
|
9.7 | IC50 | 2 | — | |
LBUJNZMSBAMNNW
|
9.7 | IC50 | 2 | — | |
NDQPAYWKSVOGPA
|
9.7 | IC50 | 2 | — | |
IGZIVKKJEQRJRW
|
9.7 | IC50 | 3 | — | |
PPKOMRSAECKGDB
|
9.7 | IC50 | 2 | — | |
URJWEBIIRXSJGD
|
9.7 | IC50 | 2 | — | |
LBUJNZMSBAMNNW
|
9.7 | IC50 | 2 | — | |
DGNBLVOENHCAGS
|
9.7 | IC50 | 3 | — | |
GOHDRFMFMTWCFA
|
9.7 | Ki | 3 | — | |
HPFPEYFODXCUDT
|
9.7 | IC50 | 2 | — | |
JUAIGMUUJDBFBA
|
9.7 | IC50 | 2 | — | |
KLGUOFQVXLDGTK
|
9.7 | IC50 | 2 | — | |
KWQWZDJFPORDSD
|
9.7 | IC50 | 2 | — | |
LPHDIQKURFDTPO
|
9.7 | IC50 | 2 | — | |
LUTLMEWAYGPCHC
|
9.7 | IC50 | 2 | — | |
LXUFTOZVBIOJCM
|
9.7 | IC50 | 2 | — | |
NLDMLONURZMDCO
|
9.7 | IC50 | 2 | — | |
QHOGQRUUXZIZIW
|
9.7 | Ki | 3 | — | |
SICGXIYTLNIGLG
|
9.7 | IC50 | 2 | — | |
VZTFDJHUSZRUMV
|
9.7 | IC50 | 2 | — | |
WFTRLROTBYTPTM
|
9.7 | IC50 | 2 | — | |
ZUJJFZSSMJANFF
|
9.7 | IC50 | 2 | — | |
IGYTYDLTGAZLER
|
9.7 | IC50 | 3 | — | |
NICUEZQIMBHMRX
|
9.7 | IC50 | 2 | — | |
SDHRADPEFDLIKD
|
9.7 | IC50 | 3 | — | |
HFJWCXGBCKLGBC
|
9.7 | Ki | 3 | — | |
LOJFDCLZRGKRBD
|
9.7 | Ki | 3 | — | |
FPUFRVZXLSMBNG
|
9.7 | IC50 | 3 | — | |
DPCSEKLXKDUSOY
|
9.7 | Ki | 3 | — |