Target Details
| UniProt AC | P11309 |
|---|---|
| Gene Symbol | PIM1 |
| Protein Name | Serine/threonine-protein kinase pim-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,647
- Clinical molecules 25
- Avg pChEMBL 8.21
KEGG Pathways (5)
Active Molecules (2,647)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KLGUOFQVXLDGTK
|
10.0 | IC50 | 2 | — | |
LPHDIQKURFDTPO
|
10.0 | IC50 | 2 | — | |
OSSMVZDTZQMDKR
|
10.0 | IC50 | 3 | — | |
OXMLPWDSSOSNEW
|
10.0 | IC50 | 3 | — | |
OZMKGYXZDRVOCC
|
10.0 | IC50 | 3 | — | |
PCKUZAUQQUCSJT
|
10.0 | IC50 | 2 | — | |
UOMPPOVQMYNXST
|
10.0 | IC50 | 3 | — | |
VHSCLASKZPNLMQ
|
10.0 | IC50 | 3 | — | |
XNTIENONSOGMRS
|
10.0 | IC50 | 2 | — | |
YWQCLSBVOVPANW
|
10.0 | IC50 | 2 | — | |
QBMHBUSZNODSPS
|
10.0 | Ki | 3 | — | |
RYNYBECHFAHSNA
|
10.0 | Ki | 3 | — | |
AWEQRQAMCRCOJY
|
10.0 | Ki | 3 | — | |
WLBVZYXAXNRNOX
|
10.0 | Ki | 3 | — | |
WTEOQEQLDVVRQM
|
10.0 | IC50 | 2 | — | |
XFQXLZJUIKQXOU
|
10.0 | Ki | 3 | — | |
UMSZCQJFRUIBCG
|
9.9 | Ki | 3 | — | |
GPGQKMLTKINISD
|
9.9 | IC50 | 3 | — | |
MZEDYGZPEWMQOQ
|
9.9 | Ki | 3 | — | |
LNMWCDOUCVMIEV
|
9.9 | Ki | 3 | — | |
PBVKOULOPAMXJJ
|
9.9 | Ki | 3 | — | |
AMLBGFLCAMEAEJ
|
9.9 | Ki | 3 | — | |
CBTMNZYWVBDQRS
|
9.9 | IC50 | 3 | — | |
GZNLJOZSXCJLOV
|
9.9 | Ki | 3 | — | |
HWMOBKCNNBAOSF
|
9.9 | Ki | 3 | — | |
ORPVEVRJSBYOAF
|
9.9 | IC50 | 2 | — | |
QXRGGZYZVNNLQV
|
9.9 | IC50 | 3 | — | |
ZMLWOFMZTHIIIJ
|
9.9 | IC50 | 2 | — | |
CYOQMLSODZDBGH
|
9.9 | Ki | 3 | — | |
QUQHXWRFOPDKOE
|
9.9 | Ki | 3 | — | |
CVOUMUUAQGOVCQ
|
9.9 | Ki | 3 | — | |
AYNCNNOVAOFEMG
|
9.9 | IC50 | 3 | — | |
HRAGREQODMBNFS
|
9.9 | Ki | 3 | — | |
OLIOBBIZJBFLQG
|
9.9 | IC50 | 3 | — | |
QYFGCYLEXSUIII
|
9.9 | IC50 | 3 | — | |
WLKLBBSKBUEHCT
|
9.9 | IC50 | 2 | — | |
FFBXBFZMXQAJBH
|
9.9 | Ki | 3 | — | |
LBSWUVMKCABART
|
9.9 | Ki | 3 | — | |
NVIMRDPIWGJULC
|
9.9 | Ki | 3 | — | |
MRSQWVHHJSPXOI
|
9.8 | IC50 | 3 | — | |
QKQSCRNMPDQOQG
|
9.8 | Ki | 3 | — | |
QOBRNBJEEWVJLW
|
9.8 | IC50 | 3 | — | |
RXIVHKXXRWBNDH
|
9.8 | IC50 | 3 | — | |
XIXPZKIRXUHXDD
|
9.8 | IC50 | 2 | — | |
NDXJCTYWGYPGPM
|
9.8 | Ki | 3 | — | |
KEENMEQOTGVAOA
|
9.8 | Ki | 3 | — | |
KTRUDSZOTYPXRK
|
9.8 | Ki | 3 | — | |
SFYXMVJWOAJPOJ
|
9.8 | Ki | 3 | — | |
TWMFYPYXRNFCRE
|
9.8 | Ki | 3 | — | |
OTCBQVWPAUVEEA
|
9.8 | Ki | 3 | — |