Target Details
| UniProt AC | P11309 |
|---|---|
| Gene Symbol | PIM1 |
| Protein Name | Serine/threonine-protein kinase pim-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,647
- Clinical molecules 25
- Avg pChEMBL 8.21
KEGG Pathways (5)
Active Molecules (2,647)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MEKFXUFACKZUCV
|
6.1 | IC50 | 9 | — | |
PGPHHJBZEGSUNE
|
6.1 | IC50 | 21 | — | |
PGPHHJBZEGSUNE
|
6.1 | IC50 | 17 | — | |
HCBIATVCCJRSKR
|
6.0 | IC50 | 5 | — | |
ODHWZXUUXOFUQZ
|
6.0 | IC50 | 3 | — | |
SGIZECXZFLAGBW
|
6.0 | IC50 | 2 | — | |
GVMDVMPNOAVKJR
|
6.0 | Ki | 26 | Yes | |
NNPANFBXAYOEKG
|
6.0 | IC50 | 2 | — | |
KGPGFQWBCSZGEL
|
6.0 | Kd | 59 | Yes | |
KZNIFHPLKGYRTM
|
6.0 | IC50 | 21 | Yes | |
WCRZDULJXSERSJ
|
6.0 | IC50 | 2 | — | |
ARJGUVIAPHIKLE
|
6.0 | IC50 | 2 | — | |
JANQPHRPUAYQTA
|
6.0 | IC50 | 5 | — | |
VRXBTIZULFDBAA
|
6.0 | IC50 | 2 | — | |
YEPMKNVGDPFWNG
|
6.0 | IC50 | 2 | — | |
HXXLFEGOFNHPAQ
|
6.0 | IC50 | 2 | — | |
AKWVKIGCMCHYJT
|
6.0 | Ki | 8 | — | |
BWKXBXIDANAPTC
|
6.0 | IC50 | 2 | — | |
DYHKEGKDOOZETF
|
6.0 | IC50 | 9 | — | |
DZIPQNPWTUXXSJ
|
6.0 | Ki | 18 | — | |
FUMCKNCUEAQHCV
|
6.0 | Ki | 103 | — | |
IMXNSLXJEYDPGL
|
6.0 | IC50 | 2 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
JHYHWHUTTXJICB
|
6.0 | Ki | 18 | — | |
JRLSUZIPUYDUKX
|
6.0 | Ki | 22 | — | |
KCAOZWGHCAZVLE
|
6.0 | IC50 | 2 | — | |
KHVVJKLNKLQLJZ
|
6.0 | IC50 | 288 | — | |
KWRXWPRFIUJQBP
|
6.0 | Ki | 25 | — | |
LPILBMJJRGTKOQ
|
6.0 | Ki | 27 | — | |
MAHFVAHPQSLLJF
|
6.0 | IC50 | 288 | — | |
MHWHPWMWKYXCRJ
|
6.0 | Ki | 32 | — | |
OLVBAUVSICCWEJ
|
6.0 | Ki | 39 | — | |
OUJZYQBEFNDJQN
|
6.0 | Ki | 71 | — | |
PKQJCYXKRNGUKQ
|
6.0 | IC50 | 6 | — | |
RGOPHVZLEMGMBZ
|
6.0 | Ki | 20 | — | |
RIBBPSYZBQQTQC
|
6.0 | Ki | 15 | — | |
RKDYDLMULRETNX
|
6.0 | Ki | 8 | — | |
UIRCQOKSJDLYBB
|
6.0 | Ki | 50 | — | |
ULVWJFBHQIXEPE
|
6.0 | Ki | 10 | — | |
URNZTLZSAVLTIZ
|
6.0 | Ki | 26 | — | |
UUYUVYXSHUTRGO
|
6.0 | Ki | 4 | — | |
VSPFURGQAYMVAN
|
6.0 | Ki | 17 | — | |
WZISGNDZZPSYRP
|
6.0 | Ki | 20 | — | |
XBDWKVLCDCUNHH
|
6.0 | Ki | 18 | — | |
XSRHBCYNCKAFKS
|
6.0 | Ki | 45 | — | |
YGKFZWJWKPZPQM
|
6.0 | Ki | 13 | — | |
YQKSNDNARJQAHP
|
6.0 | Ki | 12 | — |