Target Details
| UniProt AC | P11309 |
|---|---|
| Gene Symbol | PIM1 |
| Protein Name | Serine/threonine-protein kinase pim-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,647
- Clinical molecules 25
- Avg pChEMBL 8.21
KEGG Pathways (5)
Active Molecules (2,647)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
IDXOFDAWMQNDDL
|
6.2 | IC50 | 3 | — | |
IXFGPIBQUFVMNS
|
6.2 | IC50 | 2 | — | |
NEBJGJOGYMUDIV
|
6.2 | IC50 | 3 | — | |
RKDWPINBHFDPDR
|
6.2 | IC50 | 3 | — | |
TYUZGXHLSQZYAQ
|
6.2 | IC50 | 3 | — | |
QLWFPXXGZGCHFQ
|
6.1 | IC50 | 5 | — | |
CTOSZAUWENPXGH
|
6.1 | IC50 | 2 | — | |
RJGLNSNPZNKTGL
|
6.1 | IC50 | 2 | — | |
UAGUOISHFNNZGY
|
6.1 | IC50 | 2 | — | |
YLEPCOMPXJKHRR
|
6.1 | IC50 | 2 | — | |
MXZKCOUOYWSEKW
|
6.1 | IC50 | 2 | — | |
BIIVYFLTOXDAOV
|
6.1 | Ki | 31 | — | |
CKVWQORGCCEYHS
|
6.1 | Ki | 50 | — | |
CXZZKTFGTNQHGD
|
6.1 | Ki | 4 | — | |
DKTMRIORKQEKMU
|
6.1 | Ki | 10 | — | |
FPQHXFMYXQZPSV
|
6.1 | Ki | 23 | — | |
GHMRUNOHAHJNNA
|
6.1 | Ki | 29 | — | |
GXFGHUNNGNQSMQ
|
6.1 | Ki | 19 | — | |
HBZTVQKHXVDIDE
|
6.1 | Ki | 9 | — | |
HGLWPJISHDLCTE
|
6.1 | IC50 | 7 | — | |
HRJWTAWVFDCTGO
|
6.1 | Ki | 13 | Yes | |
INJUVNWOFHYUIN
|
6.1 | Ki | 9 | Yes | |
JEYMTHFRFGDBSF
|
6.1 | IC50 | 3 | — | |
JPYQFPGTGGLOMD
|
6.1 | IC50 | 4 | — | |
KEBMSGAJMPWLNS
|
6.1 | IC50 | 7 | Yes | |
KTRGYJLQTZDGPX
|
6.1 | Ki | 9 | — | |
LXVBELDBJGYFEM
|
6.1 | Ki | 20 | — | |
MONUZQWCBUZODF
|
6.1 | Ki | 3 | — | |
NFKMFNBKEOQNPZ
|
6.1 | Ki | 43 | — | |
OKCNACDPDSQZSE
|
6.1 | Ki | 7 | — | |
RYSOFKOEVPNDDI
|
6.1 | Ki | 9 | — | |
SMRWVXLSRJWVBF
|
6.1 | Ki | 25 | — | |
UPPYTUNUGKDPSA
|
6.1 | Ki | 7 | — | |
UXUQVXDYXKMCGA
|
6.1 | Ki | 21 | — | |
VABVHJXJMHPWJC
|
6.1 | IC50 | 3 | — | |
VIZWJTHWUUQVGO
|
6.1 | Ki | 9 | — | |
VLEFVPMCVJDTHZ
|
6.1 | Ki | 13 | — | |
VYACUCWGDYRIAG
|
6.1 | Ki | 7 | — | |
WICLISNBDMGFST
|
6.1 | Ki | 10 | — | |
WNJPSYHJVTYTBP
|
6.1 | Ki | 9 | — | |
WZBMMJKAHHOXRG
|
6.1 | Ki | 16 | — | |
XJJYJNMNYDNXNO
|
6.1 | Ki | 23 | — | |
XNWKXXIGSPPPBH
|
6.1 | Ki | 31 | — | |
ZCAOFAAOUBUUBJ
|
6.1 | Ki | 9 | — | |
CZQHHVNHHHRRDU
|
6.1 | IC50 | 12 | Yes | |
NXBHOGUUOJAZBN
|
6.1 | IC50 | 4 | — | |
RFSBAWKLQHFSAF
|
6.1 | Ki | 2 | — | |
TXXUEHVGHOFRGC
|
6.1 | IC50 | 2 | — | |
ZJNQYXSEANTVCY
|
6.1 | IC50 | 2 | — | |
DEIFYFMWJVRUHV
|
6.1 | IC50 | 2 | — |