Target Details
| UniProt AC | P11309 |
|---|---|
| Gene Symbol | PIM1 |
| Protein Name | Serine/threonine-protein kinase pim-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,647
- Clinical molecules 25
- Avg pChEMBL 8.21
KEGG Pathways (5)
Active Molecules (2,647)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HJGKZOCLHWKVJH
|
6.3 | IC50 | 2 | — | |
JUYXBRKVOIMFID
|
6.3 | IC50 | 2 | — | |
LTDNKZSWXYPFSO
|
6.3 | IC50 | 2 | — | |
PKUBRJJJKVADPK
|
6.3 | IC50 | 2 | — | |
PNSNZHAESHMNMQ
|
6.3 | IC50 | 2 | — | |
TWDZDBZNJVDYIW
|
6.3 | IC50 | 2 | — | |
VVHKRQILCVGPQL
|
6.3 | IC50 | 2 | — | |
BIIVYFLTOXDAOV
|
6.2 | Kd | 29 | — | |
BIIVYFLTOXDAOV
|
6.2 | Kd | 82 | Yes | |
BMGQWWVMWDBQGC
|
6.2 | Kd | 147 | Yes | |
BMGQWWVMWDBQGC
|
6.2 | Kd | 91 | Yes | |
PZCSBWJSPSARQH
|
6.2 | IC50 | 3 | — | |
HEOZBPOPPDUPGK
|
6.2 | IC50 | 3 | — | |
KUIXBLRMWNOGNN
|
6.2 | IC50 | 2 | — | |
LASSUIXPGNSPGU
|
6.2 | IC50 | 5 | — | |
HXHFVYQPJRIKLE
|
6.2 | IC50 | 3 | — | |
LFTSGFILTZXQSJ
|
6.2 | IC50 | 2 | — | |
QNABDSWBQJKBHK
|
6.2 | IC50 | 45 | — | |
UODOVESKEUAVCH
|
6.2 | IC50 | 2 | — | |
DTXPSQFSJWKKSG
|
6.2 | IC50 | 2 | — | |
DZPOUCQZRNTFFR
|
6.2 | IC50 | 2 | — | |
WUPRAHSNJBLKQZ
|
6.2 | IC50 | 2 | — | |
AKNIGLLNHUTMPO
|
6.2 | IC50 | 9 | — | |
PTMADKDGOQDQEW
|
6.2 | IC50 | 2 | — | |
BRTHUECZMVKNMQ
|
6.2 | Ki | 31 | — | |
CHADTINFLWZSKR
|
6.2 | Ki | 26 | — | |
HHSVICUMCOBRPT
|
6.2 | Ki | 33 | — | |
HSKVRPZJBMXFDX
|
6.2 | Ki | 20 | — | |
IABDKYMGRMDGMM
|
6.2 | Ki | 10 | — | |
LCHCSKHPVCDXAU
|
6.2 | Ki | 30 | — | |
NWMPVMMGSHXANZ
|
6.2 | Ki | 58 | — | |
NXNQLECPAXXYTR
|
6.2 | Ki | 29 | — | |
ONNGIYXISLGYEJ
|
6.2 | IC50 | 2 | — | |
PNKALLUVKOKYHZ
|
6.2 | Ki | 32 | — | |
QGOIQRQXIWSNJF
|
6.2 | Ki | 6 | — | |
RVSKJUNTDGBSSS
|
6.2 | Ki | 25 | — | |
VGURQCQNQDZAOF
|
6.2 | Ki | 6 | — | |
VNDWQCSOSCCWIP
|
6.2 | Ki | 39 | Yes | |
XZONYYFHQICDAM
|
6.2 | Ki | 19 | — | |
ZGDYBJXDIXVTLV
|
6.2 | Ki | 54 | — | |
ZKLJKKASNXVQBZ
|
6.2 | Ki | 27 | — | |
ZNHQJXHYQWLGFE
|
6.2 | IC50 | 2 | — | |
IPQWMGNQGDHUJR
|
6.2 | IC50 | 2 | — | |
IWVAFPBIIPDZPF
|
6.2 | IC50 | 3 | — | |
MZXRFYLHTPTREK
|
6.2 | IC50 | 3 | — | |
UPDQDPHDALXCMH
|
6.2 | IC50 | 2 | — | |
BFWHRHJPPAUSLJ
|
6.2 | IC50 | 2 | — | |
DMNJQOOMCYGQDB
|
6.2 | IC50 | 2 | — | |
VLOOJWQZGAEEAD
|
6.2 | IC50 | 2 | — | |
ZTEGEMFKBZMGOF
|
6.2 | IC50 | 9 | — |