Target Details
| UniProt AC | P11309 |
|---|---|
| Gene Symbol | PIM1 |
| Protein Name | Serine/threonine-protein kinase pim-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,647
- Clinical molecules 25
- Avg pChEMBL 8.21
KEGG Pathways (5)
Active Molecules (2,647)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MYUKMNGTJODGDO
|
6.3 | Ki | 2 | — | |
BUWKEFCPLBPYPS
|
6.3 | IC50 | 3 | — | |
FXFHRANPUZFDHI
|
6.3 | IC50 | 2 | — | |
IDNJKMAZNUUVIO
|
6.3 | IC50 | 9 | — | |
JVWTTWRBGWZCTC
|
6.3 | IC50 | 2 | — | |
CJCNVDWBDYXQMZ
|
6.3 | IC50 | 3 | — | |
NSJSUQKRPXMKFM
|
6.3 | IC50 | 3 | — | |
YFFJZYDSWBTDHO
|
6.3 | IC50 | 2 | — | |
DFIYULDPYGDCHT
|
6.3 | IC50 | 2 | — | |
QCTMVDQWYGRUJK
|
6.3 | IC50 | 9 | — | |
FOIOWDZKEWEOQP
|
6.3 | IC50 | 2 | — | |
MQSVIANYXKTUMS
|
6.3 | IC50 | 2 | — | |
VCVQQLOILLJUOV
|
6.3 | Ki | 2 | — | |
AWJPVXSHMIELNJ
|
6.3 | Ki | 23 | — | |
AZCMGIZOUJMZKI
|
6.3 | IC50 | 2 | — | |
BQPLWJRDSDNGNE
|
6.3 | Ki | 16 | — | |
CTQIQHVVPQICIK
|
6.3 | Ki | 7 | — | |
FSLDLBJGAMZARH
|
6.3 | IC50 | 3 | — | |
GLWBITRHFXSHPS
|
6.3 | IC50 | 2 | — | |
GPSRFACTNSQKSI
|
6.3 | Ki | 2 | — | |
JBRASADWXDKCLJ
|
6.3 | Ki | 22 | — | |
JMHQUQCLIVNTHT
|
6.3 | Ki | 24 | — | |
KRIUNPBAQZGFQA
|
6.3 | Ki | 76 | — | |
LHQWPYOYDRVMFI
|
6.3 | Ki | 21 | — | |
MQAKXLBEDXFDMV
|
6.3 | Ki | 5 | — | |
MTDOMZCSLNXWQL
|
6.3 | IC50 | 2 | — | |
NAGOZOOVQLAGAY
|
6.3 | IC50 | 2 | — | |
PJUVRETYCLPAFV
|
6.3 | Ki | 20 | — | |
PNAPQQCRNHMIER
|
6.3 | Ki | 12 | — | |
PTZQSGFNHIVQKV
|
6.3 | Ki | 8 | — | |
PWIKZIKRKUUHRB
|
6.3 | Ki | 9 | — | |
RQJIDUOCLNMUHR
|
6.3 | Ki | 15 | — | |
RXQXACYMRVINQU
|
6.3 | IC50 | 5 | — | |
SHENEEFOURUIBP
|
6.3 | Ki | 29 | — | |
SLKCVFPEQGHNSI
|
6.3 | Ki | 29 | — | |
VUDAXHCEPITOSW
|
6.3 | Ki | 4 | — | |
VVEGARMQKNYDID
|
6.3 | Ki | 24 | — | |
XOJQJDHWKVZUAT
|
6.3 | Ki | 9 | — | |
XPHWIERLJBFPFV
|
6.3 | Ki | 69 | — | |
SLCNIAWQMQCAFR
|
6.3 | IC50 | 8 | — | |
XDJFHHCDOHCTAP
|
6.3 | IC50 | 2 | — | |
YBNMHABOJIFTIT
|
6.3 | IC50 | 2 | — | |
ZCEUQTPCLMOQAN
|
6.3 | IC50 | 2 | — | |
LCWIMYAVOHBYBI
|
6.3 | IC50 | 2 | — | |
NZRSCXANLQLBGL
|
6.3 | IC50 | 2 | — | |
UKRBSFMZVQRMFR
|
6.3 | Ki | 2 | — | |
NVAMEDJVKXMJQB
|
6.3 | IC50 | 2 | — | |
BACDVSQDOPKJRZ
|
6.3 | IC50 | 2 | — | |
BUTIQIJGJAAJDE
|
6.3 | IC50 | 3 | — | |
GOAQEBHGPZLMLL
|
6.3 | IC50 | 3 | — |