Target Details
| UniProt AC | P11309 |
|---|---|
| Gene Symbol | PIM1 |
| Protein Name | Serine/threonine-protein kinase pim-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,647
- Clinical molecules 25
- Avg pChEMBL 8.21
KEGG Pathways (5)
Active Molecules (2,647)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NJSRSTOIFDINEP
|
10.2 | IC50 | 3 | — | |
OIZRMKSUYVZCDN
|
10.2 | Ki | 3 | — | |
OJACGGVADSBVKM
|
10.2 | IC50 | 2 | — | |
XQMOXTIXSKOQJT
|
10.2 | IC50 | 3 | — | |
YGGVNGYTDSWNCC
|
10.2 | IC50 | 3 | — | |
ZBNXMASDPWDPMD
|
10.2 | IC50 | 3 | — | |
BVEIZVVTRHJPMZ
|
10.1 | Ki | 3 | — | |
KTRUDSZOTYPXRK
|
10.1 | Ki | 3 | — | |
RJVAYMWLBAJIOR
|
10.1 | Ki | 3 | — | |
SJECHZVGJJSCJC
|
10.1 | Ki | 3 | — | |
CDQXYOYHHLAARJ
|
10.1 | Ki | 3 | — | |
JTYPMPKUWKZGBR
|
10.1 | IC50 | 2 | — | |
PUJNJBCBFYLKKR
|
10.1 | Ki | 3 | — | |
YMMNFBQYTKNEGM
|
10.1 | Ki | 3 | — | |
ACVVOPWTQGINNG
|
10.1 | Ki | 3 | — | |
AWSQCMGUEHCTJL
|
10.1 | IC50 | 2 | — | |
CHHIPMRGGGEDHC
|
10.1 | IC50 | 3 | — | |
JLRFGUCJKRWAIB
|
10.1 | IC50 | 3 | — | |
MLPJIYXHHVPOPK
|
10.1 | IC50 | 3 | — | |
OGPYGXDCCOBKSO
|
10.1 | Ki | 3 | — | |
OSSMVZDTZQMDKR
|
10.1 | IC50 | 3 | — | |
VNFMQMVCRRHLOL
|
10.1 | IC50 | 3 | — | |
YGEIOFPNCMIFRQ
|
10.1 | IC50 | 3 | — | |
BRUNMKAHHCQBLZ
|
10.1 | IC50 | 2 | — | |
RLVWGBLSDHEDOU
|
10.1 | Ki | 3 | — | |
BCKKTEZAIGOQBN
|
10.1 | Ki | 3 | — | |
NCCOUWIBICXQSL
|
10.1 | Ki | 3 | — | |
AZUDXPDVDQXJJH
|
10.1 | Ki | 3 | — | |
IGYTYDLTGAZLER
|
10.1 | IC50 | 3 | — | |
IGYZGYVIMRJJRJ
|
10.1 | Ki | 3 | — | |
IIYNOYBNJALAMM
|
10.1 | IC50 | 3 | — | |
KRMOAWBSZVZSIA
|
10.1 | IC50 | 3 | — | |
QVRUMXAVDBYHBP
|
10.1 | IC50 | 3 | — | |
RLVXEHCCQLTFMJ
|
10.1 | IC50 | 2 | — | |
WRMQNETYMUMXMG
|
10.1 | IC50 | 3 | — | |
FHESSCZVRQCSRX
|
10.0 | Ki | 3 | — | |
UEYONFUBMMGJIX
|
10.0 | Ki | 3 | — | |
IWDUWWSSLHPWJZ
|
10.0 | Ki | 3 | — | |
NBUDKNPONYZRBZ
|
10.0 | Ki | 3 | — | |
OUBKTSCIYLAKMV
|
10.0 | Ki | 3 | — | |
AENSKLYNJAPICQ
|
10.0 | IC50 | 2 | — | |
ASZCABSVZBJTKA
|
10.0 | IC50 | 3 | — | |
BHBIGGOODMPQTA
|
10.0 | IC50 | 2 | — | |
BYFQNMWZRKKFRI
|
10.0 | IC50 | 4 | — | |
FJZQCIBDBNRACD
|
10.0 | IC50 | 2 | — | |
FPIJQPCUMVUNOE
|
10.0 | IC50 | 2 | — | |
GTKNYUJNLDGSDF
|
10.0 | IC50 | 3 | — | |
HRAGREQODMBNFS
|
10.0 | Ki | 3 | — | |
IOOVJBGMLHBOOX
|
10.0 | IC50 | 2 | — | |
ISSQSUGBRMTNBJ
|
10.0 | IC50 | 3 | — |