Target Details
| UniProt AC | P11309 |
|---|---|
| Gene Symbol | PIM1 |
| Protein Name | Serine/threonine-protein kinase pim-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,647
- Clinical molecules 25
- Avg pChEMBL 8.21
KEGG Pathways (5)
Active Molecules (2,647)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UCESDNAOCAZCCC
|
6.5 | IC50 | 2 | — | |
WKYMGORXOQPTTO
|
6.5 | IC50 | 9 | — | |
YBTSMEPVYOMDST
|
6.5 | IC50 | 2 | — | |
YOVNFNXUCOWYSG
|
6.5 | Ki | 33 | Yes | |
HHKWNBHZPMNYAO
|
6.5 | IC50 | 3 | — | |
WHFMKTUASWKIEL
|
6.5 | IC50 | 3 | — | |
WXCIWTZRWIINEJ
|
6.5 | IC50 | 2 | — | |
GHXXZGKRRQQPIS
|
6.5 | IC50 | 2 | — | |
MHPMAOLCNNEBOA
|
6.5 | IC50 | 6 | — | |
AMEIMZMBRNKSJG
|
6.5 | IC50 | 2 | — | |
KSDORXSBAJOQKH
|
6.5 | Ki | 3 | — | |
QXMXIHBLICGPMG
|
6.5 | IC50 | 9 | — | |
SWIVJTVGOIXUKC
|
6.5 | IC50 | 9 | — | |
FYTKRHWUZSNWFH
|
6.5 | IC50 | 3 | — | |
MOGPAEFTHZLUGU
|
6.4 | IC50 | 2 | — | |
OSEXMPOYORIWSM
|
6.4 | IC50 | 2 | — | |
OWHMMNCEQSPPJR
|
6.4 | IC50 | 5 | — | |
UBGUCDLLEIGHHP
|
6.4 | IC50 | 6 | — | |
JGWXTXMXVIFIMG
|
6.4 | IC50 | 3 | — | |
UOTWZVLZNWFPOS
|
6.4 | IC50 | 2 | — | |
HGIQFKFKNNUPOP
|
6.4 | IC50 | 2 | — | |
HNIFOTFIRDDPLT
|
6.4 | IC50 | 2 | — | |
MENVSADYTLLXLP
|
6.4 | IC50 | 6 | — | |
FVMQSKYNSZUZOQ
|
6.4 | IC50 | 3 | — | |
MRMWXHSKVZBHNM
|
6.4 | IC50 | 2 | — | |
XTGFWKBHSZHXMC
|
6.4 | IC50 | 2 | — | |
CBZZSUSDNUHUEI
|
6.4 | IC50 | 2 | — | |
CFBADDSSFSYJPF
|
6.4 | Ki | 23 | — | |
HDRLAVNNWSHSOA
|
6.4 | Ki | 19 | — | |
LACOMQAWPSFXQC
|
6.4 | Ki | 27 | — | |
LYNBNVBMAGDJRW
|
6.4 | Ki | 81 | — | |
NIUJTENHSPPCKO
|
6.4 | Ki | 9 | — | |
OSHXOLFPPORXMW
|
6.4 | IC50 | 2 | — | |
QVNZKVACBBTKSL
|
6.4 | Ki | 38 | — | |
RRAMBEGOYIJQHY
|
6.4 | Ki | 11 | — | |
SGHXFHRRWFLILP
|
6.4 | Ki | 29 | — | |
UDFDIIVNIYWXDM
|
6.4 | Ki | 74 | — | |
UYGYYOIUVFMGKQ
|
6.4 | Ki | 30 | — | |
VUWOSKCPLJROAK
|
6.4 | Ki | 6 | — | |
WKOWIUGYPIXNRD
|
6.4 | IC50 | 2 | — | |
YMIJUBCSOKSFRU
|
6.4 | Ki | 87 | — | |
ZDXCUVXIHVTLEU
|
6.4 | Ki | 3 | — | |
ZGGIYFOLDBTZIL
|
6.4 | Ki | 27 | — | |
OAYLGJMFKMEJKI
|
6.4 | IC50 | 2 | — | |
PPMGWZOVBXDTHU
|
6.4 | IC50 | 4 | — | |
VDXGLZJPQRGNLY
|
6.4 | IC50 | 10 | — | |
YNJSOFSKQGYIDB
|
6.4 | IC50 | 2 | — | |
KYRUZUVASMOUCI
|
6.4 | IC50 | 2 | — | |
ACPNKTFJVNAQNM
|
6.3 | IC50 | 2 | — | |
LRSMQMIQOQCOJQ
|
6.3 | IC50 | 2 | — |