Target Details
| UniProt AC | P11309 |
|---|---|
| Gene Symbol | PIM1 |
| Protein Name | Serine/threonine-protein kinase pim-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,647
- Clinical molecules 25
- Avg pChEMBL 8.21
KEGG Pathways (5)
Active Molecules (2,647)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LOMGAGWJYPGDLT
|
6.6 | Ki | 8 | — | |
OBZHLULOFFWAJX
|
6.6 | Ki | 8 | — | |
OWDRQHVEJIYVOI
|
6.6 | Ki | 47 | — | |
RJZDECGDCKOHBV
|
6.6 | Ki | 70 | — | |
SDBOIBYRBWPIEL
|
6.6 | Ki | 31 | — | |
SHNZBTHVGXHLLD
|
6.6 | Ki | 2 | — | |
SNZAMISUNWKHPW
|
6.6 | IC50 | 2 | — | |
SRONQUHCRFZABC
|
6.6 | Ki | 28 | — | |
WCAKSXQRFBVWDG
|
6.6 | Ki | 10 | — | |
XUFLBSMTYMFOQH
|
6.6 | Ki | 43 | — | |
ZAZHHFGHOUJWKE
|
6.6 | IC50 | 2 | — | |
ZHJGWYRLJUCMRT
|
6.6 | Kd | 18 | — | |
ZYTFPHRVOZXPGZ
|
6.6 | Ki | 30 | — | |
LDOFQWMCMLOLPB
|
6.6 | IC50 | 2 | — | |
OUFYOWHGJCSWTJ
|
6.6 | IC50 | 2 | — | |
QKGJXCXUJSSLBQ
|
6.6 | IC50 | 2 | — | |
ASXDLQKYJZCCLE
|
6.6 | IC50 | 3 | — | |
JNOYDDQBVMUSBF
|
6.6 | IC50 | 2 | — | |
QWRKVKFVRKHBNP
|
6.6 | IC50 | 2 | — | |
FKOFSCFFWGHTPP
|
6.6 | IC50 | 3 | — | |
FMJPDZXMKIOBKX
|
6.6 | IC50 | 3 | — | |
GHPFSYCYZJKVDZ
|
6.6 | Ki | 18 | Yes | |
LNTZYZOAYALYHB
|
6.6 | IC50 | 2 | — | |
MITSRVMYKFVRJP
|
6.6 | Ki | 2 | — | |
VEXHSPQZXZWAJJ
|
6.6 | IC50 | 3 | — | |
GAYLCUTUNZYVAU
|
6.5 | IC50 | 2 | — | |
VIJAADBVHYURKM
|
6.5 | IC50 | 3 | — | |
ZGYIJLHCURUFFT
|
6.5 | IC50 | 2 | — | |
ZTWXZFSVBMVSQW
|
6.5 | IC50 | 2 | — | |
KYQQIKNSNCDVJK
|
6.5 | Ki | 2 | — | |
OSVUGUHRKMMBSE
|
6.5 | Kd | 170 | — | |
FOKXPYMCQHYPFQ
|
6.5 | Ki | 2 | — | |
UWZJKUPJAFEETI
|
6.5 | IC50 | 2 | — | |
ANJVMJRVHWNWEU
|
6.5 | IC50 | 2 | — | |
BJBDVWJMRSHUFX
|
6.5 | IC50 | 3 | — | |
MPJZDLDOQBVNLJ
|
6.5 | Ki | 3 | — | |
QLJZRTOWAKEAEW
|
6.5 | IC50 | 2 | — | |
CALAEFSQWBJMDU
|
6.5 | Ki | 21 | — | |
DRKMVSXBCWCKMW
|
6.5 | IC50 | 2 | — | |
GILNGUYOGYOZMP
|
6.5 | IC50 | 6 | — | |
GIYCJABQEROMOM
|
6.5 | IC50 | 2 | — | |
GXZFDXZCJALHRF
|
6.5 | IC50 | 6 | — | |
FLEAYYMORDPWAJ
|
6.5 | Ki | 90 | — | |
HKTZXBYEGIFWTQ
|
6.5 | IC50 | 2 | — | |
IRQBQPNOWKSJBR
|
6.5 | IC50 | 2 | — | |
KHGPYYFCIAISBU
|
6.5 | Ki | 31 | — | |
LEKFNUHVYFCLDC
|
6.5 | IC50 | 2 | — | |
OBHMNLIBIPFXCY
|
6.5 | Ki | 15 | — | |
QNZJDYVERIAXAI
|
6.5 | Ki | 7 | — | |
QZIVKBVZTKZHCY
|
6.5 | Ki | 2 | — |