Target Details
| UniProt AC | P11309 |
|---|---|
| Gene Symbol | PIM1 |
| Protein Name | Serine/threonine-protein kinase pim-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,647
- Clinical molecules 25
- Avg pChEMBL 8.21
KEGG Pathways (5)
Active Molecules (2,647)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SEAHTYRLTWEUCM
|
6.7 | IC50 | 2 | — | |
UIARLYUEJFELEN
|
6.7 | Kd | 289 | Yes | |
ULCBWFFBEDGJOB
|
6.7 | IC50 | 3 | — | |
VLAUCAGVICCIPT
|
6.7 | IC50 | 2 | — | |
XCOSAQGGGZDYJN
|
6.7 | IC50 | 11 | — | |
XXSPHNFKLDJDAK
|
6.7 | Ki | 26 | — | |
YXLMZHOMTDRUPU
|
6.7 | IC50 | 2 | — | |
ZCBUQCWBWNUWSU
|
6.7 | Kd | 59 | — | |
ZJKIGHOTHYACFW
|
6.7 | Kd | 6 | — | |
ZKHDDJKHTPLPOQ
|
6.7 | Ki | 62 | — | |
QDITZBLZQQZVEE
|
6.7 | Kd | 19 | — | |
RQFQZDREOKTQLS
|
6.7 | IC50 | 2 | — | |
XXHMHUZOEHCANX
|
6.7 | IC50 | 2 | — | |
FRWQFENAPABQKD
|
6.7 | IC50 | 2 | — | |
NHMJTDONHQHMSX
|
6.7 | IC50 | 2 | — | |
NXSJMRCTGYTSTK
|
6.7 | Kd | 200 | — | |
PWLTUXUDBOARFK
|
6.7 | IC50 | 2 | — | |
MUOKSQABCJCOPU
|
6.7 | IC50 | 2 | — | |
NZRNMCARUJZDNV
|
6.7 | IC50 | 2 | — | |
GBYGWVVFPYTZJX
|
6.7 | IC50 | 4 | — | |
GIMGRIKBHQXFGE
|
6.7 | IC50 | 3 | — | |
JUYNMCTUZPLCCS
|
6.7 | IC50 | 2 | — | |
LRJIEZPKWFBSEJ
|
6.7 | IC50 | 6 | — | |
IZPVJWBTUYHIEP
|
6.7 | IC50 | 2 | — | |
PUALMDIOHBZAKU
|
6.7 | IC50 | 2 | — | |
WWFCQWLROPCPMS
|
6.7 | IC50 | 3 | — | |
XUXVOLMDSBESRR
|
6.7 | IC50 | 3 | — | |
IEFSYAIPOMVBKO
|
6.6 | IC50 | 2 | — | |
JLPYFPFLXZSGDS
|
6.6 | IC50 | 3 | — | |
RATNMNKEUJOIEP
|
6.6 | IC50 | 2 | — | |
GWSMWULJBQJZOT
|
6.6 | IC50 | 2 | — | |
KKEFRYYBQOMKLR
|
6.6 | IC50 | 2 | — | |
MZBVCDVHYWIHEK
|
6.6 | IC50 | 2 | — | |
PIQQGEFPKANVCP
|
6.6 | IC50 | 2 | — | |
QNDDTEOQJSXYGY
|
6.6 | IC50 | 2 | — | |
DYSRECIVMDGUQU
|
6.6 | Ki | 29 | — | |
ICMWGEHZAFFUFB
|
6.6 | IC50 | 2 | — | |
IVGLUWWICIQZOH
|
6.6 | IC50 | 2 | — | |
MZQFDJIZQKRSCS
|
6.6 | IC50 | 3 | — | |
ORCAYCBKCKHOLI
|
6.6 | IC50 | 2 | — | |
YHBLEBHGDWHESZ
|
6.6 | IC50 | 2 | — | |
ADMFLILDQJSEIK
|
6.6 | Ki | 72 | — | |
AGYZUONRISUOIK
|
6.6 | Ki | 10 | — | |
DPRGOXVMSNDADU
|
6.6 | Ki | 16 | — | |
DPUAZEZKRZGPNA
|
6.6 | IC50 | 2 | — | |
DTMZXHDQZQLTHA
|
6.6 | Ki | 21 | — | |
DWXUTKBSWVUPBE
|
6.6 | Ki | 8 | — | |
HKRUFMXPSVYVMY
|
6.6 | Ki | 4 | — | |
HOYRWTWZUFFACV
|
6.6 | Ki | 28 | — | |
KYACBMRLQMEIAI
|
6.6 | Ki | 30 | — |