Target Details
| UniProt AC | P11309 |
|---|---|
| Gene Symbol | PIM1 |
| Protein Name | Serine/threonine-protein kinase pim-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,647
- Clinical molecules 25
- Avg pChEMBL 8.21
KEGG Pathways (5)
Active Molecules (2,647)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HTFKYUIYCWNLNL
|
6.8 | IC50 | 3 | — | |
JOIUJUJSHIHBDT
|
6.8 | Ki | 18 | — | |
KAICHBSRWFIESE
|
6.8 | Ki | 14 | — | |
RNGUAWHIYIYTKR
|
6.8 | IC50 | 3 | — | |
RQIKEJKQGQDFHA
|
6.8 | IC50 | 2 | — | |
TURIRIIGEMCNAC
|
6.8 | IC50 | 2 | — | |
UMYBAQLXZPEUQW
|
6.8 | Ki | 15 | — | |
UPITUWGOTMBQLX
|
6.8 | Ki | 13 | — | |
USHMNZBDAOGLMB
|
6.8 | Ki | 26 | — | |
WHKWRDQKKUPBMN
|
6.8 | Ki | 7 | — | |
WLLUQXGGNFUQGM
|
6.8 | Ki | 4 | — | |
XFWUTMHVDGPWLH
|
6.8 | Ki | 75 | — | |
YJBNTRQKJQHMTM
|
6.8 | Ki | 11 | — | |
YRWZRNPWLKELTF
|
6.8 | Ki | 2 | — | |
YYPKOMNJRZRWIC
|
6.8 | Ki | 26 | — | |
ZNOHZAFAPWYALF
|
6.8 | IC50 | 2 | — | |
PVVXLUMJFJECFG
|
6.8 | IC50 | 3 | — | |
WXHGHAQKEZKCNT
|
6.8 | IC50 | 2 | — | |
LUIWEOHKWIYVQO
|
6.8 | IC50 | 2 | — | |
HNEODCCAWZXTMR
|
6.8 | Ki | 2 | — | |
LMXYVLFTZRPNRV
|
6.8 | IC50 | 8 | — | |
NPIDXFQGHNFEQU
|
6.8 | IC50 | 3 | — | |
UFKSWYKDQZBJTH
|
6.8 | IC50 | 5 | — | |
MVLOBPPFCUCBHT
|
6.8 | IC50 | 9 | — | |
XKDSMPCDGPJCLX
|
6.8 | IC50 | 2 | — | |
LHBDFSZOARHGLZ
|
6.8 | IC50 | 3 | — | |
UQZFPLZZLBNFOS
|
6.8 | IC50 | 3 | — | |
ZIRFPDLVDBRJHO
|
6.8 | IC50 | 3 | — | |
BPNUQXPIQBZCMR
|
6.7 | Kd | 83 | Yes | |
UUXDJIVNVOOKFQ
|
6.7 | IC50 | 9 | — | |
WAISNUDWNYJNMT
|
6.7 | IC50 | 3 | — | |
LIUBFLOZGTYGQV
|
6.7 | IC50 | 2 | — | |
URZDNZCJPNIWLN
|
6.7 | IC50 | 2 | — | |
YRKXZCVFINEWAZ
|
6.7 | IC50 | 2 | — | |
OEZSDKKFOOLHKE
|
6.7 | Ki | 3 | — | |
RXAMEJTTXXXMKB
|
6.7 | IC50 | 2 | — | |
UQUBWQXJXQJXPB
|
6.7 | Ki | 3 | — | |
WEPFOMSXGUEDJU
|
6.7 | IC50 | 2 | — | |
BKLXEFIQIATWPR
|
6.7 | IC50 | 2 | — | |
GZPFCSWSXRQYKX
|
6.7 | IC50 | 2 | — | |
AXRCEOKUDYDWLF
|
6.7 | Kd | 31 | — | |
CFIBXVQLBVNOHW
|
6.7 | Ki | 64 | — | |
HDIIEJQPCDNNML
|
6.7 | Ki | 2 | — | |
KTWBYGUSEYSRND
|
6.7 | Ki | 28 | — | |
LSLPDHNUWRDOGC
|
6.7 | Ki | 25 | — | |
MDJCUXFFMNEBHG
|
6.7 | Ki | 13 | — | |
NSFWLIYQFQEQDW
|
6.7 | IC50 | 6 | — | |
PLGUCBXOJHSJEN
|
6.7 | IC50 | 2 | — | |
PWNFEFRGKMPFSG
|
6.7 | Ki | 2 | — | |
QLBROIYTIICCKT
|
6.7 | IC50 | 2 | — |