Target Details
| UniProt AC | P11309 |
|---|---|
| Gene Symbol | PIM1 |
| Protein Name | Serine/threonine-protein kinase pim-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,647
- Clinical molecules 25
- Avg pChEMBL 8.21
KEGG Pathways (5)
Active Molecules (2,647)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JAMDNXUAYUHJLJ
|
6.9 | Ki | 40 | — | |
OVFDOYSALNWSNU
|
6.9 | IC50 | 2 | — | |
PLHUMPJXRHMFFR
|
6.9 | Ki | 28 | — | |
QQXBOOIPHBWOGC
|
6.9 | Ki | 4 | — | |
RUHYOXVTSYTTBT
|
6.9 | IC50 | 2 | — | |
SKKRZILJUKYLJS
|
6.9 | Ki | 25 | — | |
SQXSMLLCDWJNAC
|
6.9 | Ki | 20 | — | |
UFMAIBLTWQRHAK
|
6.9 | Ki | 10 | — | |
WDARYLSSWBWVCU
|
6.9 | Ki | 49 | — | |
XMFUGSRATNLPRM
|
6.9 | Ki | 19 | — | |
BGVLELSCIHASRV
|
6.9 | Kd | 12 | — | |
BGVLELSCIHASRV
|
6.9 | Kd | 12 | — | |
DFZRBXGBXWXXGB
|
6.9 | Ki | 2 | — | |
DJUSDFVEBBYFFL
|
6.9 | Ki | 27 | — | |
FHRKKLBIQCOIMF
|
6.9 | IC50 | 2 | — | |
OQAGQAIPXINVCL
|
6.9 | Ki | 2 | — | |
QXHXZOQHNCKQSX
|
6.9 | Ki | 2 | — | |
WXIKUAVDMWNARE
|
6.9 | IC50 | 3 | — | |
XFNCJVCQFOKSKF
|
6.9 | IC50 | 2 | — | |
ZJJQGBLVLDGPGZ
|
6.9 | IC50 | 2 | — | |
BZJVKWLOCYVMBE
|
6.9 | IC50 | 2 | — | |
IJFXPCHHRYCYMT
|
6.9 | IC50 | 2 | — | |
INEAQHZLYSEMPP
|
6.9 | IC50 | 2 | — | |
OMWYPFJWIVINCQ
|
6.9 | IC50 | 2 | — | |
PHNMDUIFDUSSMV
|
6.9 | IC50 | 2 | — | |
IBESYJMYJHCZDM
|
6.9 | IC50 | 2 | — | |
QJBCIQXUAPWXJF
|
6.9 | IC50 | 2 | — | |
UAPQZSZCXXFKCX
|
6.9 | Ki | 3 | — | |
AFHADFMYZXZAEV
|
6.8 | IC50 | 2 | — | |
NVEXZMGIURASMO
|
6.8 | IC50 | 3 | — | |
XQEZXMGUDOPHOF
|
6.8 | IC50 | 4 | — | |
AEHXIQDMWQDFQF
|
6.8 | IC50 | 3 | — | |
VPYGCTNEUKKPMV
|
6.8 | IC50 | 2 | — | |
XHSGYWPQERVYAH
|
6.8 | IC50 | 2 | — | |
YRYNGVLWTQYZJO
|
6.8 | IC50 | 2 | — | |
RXAMEJTTXXXMKB
|
6.8 | IC50 | 2 | — | |
GBWOSXZUTXXXQF
|
6.8 | IC50 | 2 | — | |
KOZFSFOOLUUIGY
|
6.8 | IC50 | 88 | Yes | |
MCZCAWWHZGEUFE
|
6.8 | IC50 | 2 | — | |
MXGVGSLEDSLTIC
|
6.8 | IC50 | 2 | — | |
PNOFQFZFLHUHOU
|
6.8 | IC50 | 2 | — | |
QPVVONUJDZMFFK
|
6.8 | IC50 | 3 | — | |
VWDOGNVHWKGFOS
|
6.8 | IC50 | 3 | — | |
WHOOZDLAJIKMBZ
|
6.8 | IC50 | 2 | — | |
XLSDQSUJJYRPJM
|
6.8 | IC50 | 2 | — | |
PZYHYOBAASYQAV
|
6.8 | IC50 | 2 | — | |
ULWOXNCGPLEIMP
|
6.8 | IC50 | 2 | — | |
UYLDCVPESWFMHG
|
6.8 | IC50 | 3 | — | |
WPIQMHAJTFSESE
|
6.8 | IC50 | 3 | — | |
BQWUBCRDJPIJAT
|
6.8 | Ki | 10 | — |