Target Details
| UniProt AC | P11309 |
|---|---|
| Gene Symbol | PIM1 |
| Protein Name | Serine/threonine-protein kinase pim-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,647
- Clinical molecules 25
- Avg pChEMBL 8.21
KEGG Pathways (5)
Active Molecules (2,647)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LLPGSWBZJMRSKB
|
7.0 | IC50 | 2 | — | |
UMMNIAUFUJLWSP
|
7.0 | IC50 | 4 | — | |
VRQXRVAKPDCRCI
|
7.0 | IC50 | 3 | — | |
YRFCIKZEDHJVDM
|
7.0 | IC50 | 2 | — | |
CVEAXVOJZIHGML
|
7.0 | IC50 | 3 | — | |
DMYOZDHUHKTIQV
|
7.0 | IC50 | 2 | — | |
NEKWADPRTBLINN
|
7.0 | IC50 | 3 | — | |
PUOHSGKCNIZLIO
|
7.0 | IC50 | 2 | — | |
RVUJNEXOCBACNR
|
7.0 | IC50 | 2 | — | |
BGVLELSCIHASRV
|
7.0 | Kd | 11 | — | |
BPNUQXPIQBZCMR
|
7.0 | Ki | 60 | — | |
FMPKTXNCNJCHCC
|
7.0 | Ki | 25 | — | |
FNYHEMYACVRIOE
|
7.0 | IC50 | 3 | — | |
FSCBAXKYVITFPI
|
7.0 | IC50 | 2 | — | |
FSWFKKQQSQHIRZ
|
7.0 | Ki | 10 | — | |
RQFQZDREOKTQLS
|
7.0 | IC50 | 2 | — | |
VWVYILCFSYNJHF
|
7.0 | Ki | 49 | — | |
WAKGEHXTOOFEAE
|
7.0 | Ki | 27 | — | |
WGWOASUEIXPSEV
|
7.0 | IC50 | 2 | — | |
XMZSIICARYXABB
|
7.0 | IC50 | 2 | — | |
FZIXDSBXXBDCIU
|
7.0 | IC50 | 4 | — | |
PTCDBDLJIWEHCS
|
7.0 | IC50 | 2 | — | |
SLXLMYYURFOSRQ
|
7.0 | IC50 | 3 | — | |
UPQUIEZAMXWLIX
|
7.0 | IC50 | 3 | — | |
XJKLJBWCTWFTPQ
|
7.0 | IC50 | 3 | — | |
IFSZNNCMCGMAHD
|
7.0 | IC50 | 2 | — | |
JLODZLWVTOUEGJ
|
7.0 | IC50 | 2 | — | |
LPVAPMSEQYAFMQ
|
7.0 | IC50 | 2 | — | |
RPXPSOHJVFMQAQ
|
7.0 | IC50 | 2 | — | |
AKTIZWAVQKASGW
|
7.0 | IC50 | 2 | — | |
WDENWXDMHCFKSS
|
7.0 | IC50 | 2 | — | |
ZQGBFVDBBAKHCQ
|
7.0 | IC50 | 3 | — | |
LVBGEVIMGXRIPY
|
7.0 | IC50 | 3 | — | |
PUCCPIPNBMSAGL
|
7.0 | IC50 | 3 | — | |
QMLTXQZCXWHPPX
|
7.0 | IC50 | 2 | — | |
RXIQMLWEIBLNGH
|
7.0 | IC50 | 2 | — | |
UTWVEJOBAALHSL
|
7.0 | IC50 | 3 | — | |
ZINMQNQKXGNWQN
|
7.0 | IC50 | 2 | — | |
CPQINKSLOKLYSY
|
6.9 | IC50 | 2 | — | |
ZAOAKWGRHJIYTD
|
6.9 | Ki | 8 | — | |
HMTWWEPXQMGOSK
|
6.9 | IC50 | 3 | — | |
LCDAETYKSLPKDG
|
6.9 | IC50 | 2 | — | |
RJXWGPDMMDILGJ
|
6.9 | IC50 | 9 | — | |
SEAHTYRLTWEUCM
|
6.9 | IC50 | 2 | — | |
VWNCOFUKBTYAON
|
6.9 | IC50 | 3 | — | |
WHMWATJKBHTJIR
|
6.9 | IC50 | 3 | — | |
NOKZPPHIBFZGNL
|
6.9 | IC50 | 2 | — | |
PKIUWBSGVDRYIK
|
6.9 | Ki | 2 | — | |
GHHXRRBAWPYQTC
|
6.9 | IC50 | 2 | — | |
GQHSVFWCNBWKGM
|
6.9 | Ki | 3 | — |