Target Details
| UniProt AC | P11309 |
|---|---|
| Gene Symbol | PIM1 |
| Protein Name | Serine/threonine-protein kinase pim-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,647
- Clinical molecules 25
- Avg pChEMBL 8.21
KEGG Pathways (5)
Active Molecules (2,647)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DBDYEQWRFONQEP
|
7.2 | IC50 | 2 | — | |
HHEMFVAUZWKILQ
|
7.2 | IC50 | 3 | — | |
QQWAYVLBNKWVHL
|
7.2 | Ki | 2 | — | |
CNVDRXITZNMNTP
|
7.1 | IC50 | 4 | — | |
CQJNXVJJHWGYQQ
|
7.1 | IC50 | 3 | — | |
CYARIWRQUWGCTF
|
7.1 | IC50 | 3 | — | |
KKBGGKFCFCEFRX
|
7.1 | IC50 | 2 | — | |
LGRJHSGKEBRDHI
|
7.1 | IC50 | 4 | — | |
WISHLJZJMNBRMX
|
7.1 | IC50 | 9 | — | |
AZWJVNNXHBOAKD
|
7.1 | IC50 | 2 | — | |
QMBHNDOJNFNUMI
|
7.1 | IC50 | 3 | — | |
QZODUKPIHBQCBB
|
7.1 | IC50 | 2 | — | |
UTCSFSCIISEIJY
|
7.1 | IC50 | 2 | — | |
DXEUSDFBCOEFHQ
|
7.1 | IC50 | 2 | — | |
VGZNWCWWERCEPK
|
7.1 | IC50 | 2 | — | |
ASLGQVPNOSGBQR
|
7.1 | IC50 | 10 | — | |
OSCGVQOTNNOXNM
|
7.1 | IC50 | 2 | — | |
PSJHTNRKPOXZIN
|
7.1 | IC50 | 4 | — | |
QOHJZKISICESGE
|
7.1 | IC50 | 3 | — | |
YANNSWWYRMATEM
|
7.1 | IC50 | 4 | — | |
YUKFVIAVKMQRBS
|
7.1 | IC50 | 3 | — | |
AEYLJTAIDDIOBA
|
7.1 | Ki | 53 | — | |
AVLYNJZZQYEFEA
|
7.1 | IC50 | 8 | Yes | |
BWRQNVDGLTUELI
|
7.1 | IC50 | 5 | — | |
CEOGUGIFKNBDAK
|
7.1 | Ki | 5 | — | |
DBFCGNXJRISFMI
|
7.1 | Ki | 4 | — | |
GWJHMRBQEUHFOC
|
7.1 | Ki | 42 | — | |
OWFLADWRSCINST
|
7.1 | Ki | 30 | — | |
RCYPVQCPYKNSTG
|
7.1 | IC50 | 7 | — | |
RGNHKJWHFIPHIM
|
7.1 | Ki | 66 | — | |
BPRSGQHMNJDRQL
|
7.1 | IC50 | 2 | — | |
MRDMBHMNISKFJZ
|
7.1 | IC50 | 3 | — | |
QPMFXQPTRYIZIM
|
7.1 | IC50 | 3 | — | |
YTBNWMZWTXFXLR
|
7.1 | IC50 | 2 | — | |
JUICDMKIEODAIP
|
7.1 | IC50 | 2 | — | |
LUFUSDUYKFHLLN
|
7.1 | IC50 | 3 | — | |
CMWRPDHVGMHLSZ
|
7.1 | IC50 | 22 | — | |
LVYDNZIZBIQXIS
|
7.1 | IC50 | 2 | — | |
NKIQMYXRVCWNGC
|
7.1 | IC50 | 2 | — | |
RCYKJOARDMHTPJ
|
7.1 | IC50 | 2 | — | |
DZWWBGNMJMTMJH
|
7.0 | IC50 | 3 | — | |
PJOIFMZNPPOQBO
|
7.0 | IC50 | 2 | — | |
GZVLKFFYCJUAPT
|
7.0 | IC50 | 2 | — | |
KRKGTVKFVGNHRA
|
7.0 | IC50 | 2 | — | |
MOSRYOLZKZQPJM
|
7.0 | IC50 | 4 | — | |
XPDNPGNUQDMFOW
|
7.0 | Ki | 2 | — | |
CVBIOKGKBZUACK
|
7.0 | IC50 | 2 | — | |
FMPZTFZITBVOOF
|
7.0 | IC50 | 3 | — | |
GWPJORJJIDSOOC
|
7.0 | IC50 | 3 | — | |
WNYGUIMINVSVMX
|
7.0 | IC50 | 2 | — |