Target Details
| UniProt AC | P11309 |
|---|---|
| Gene Symbol | PIM1 |
| Protein Name | Serine/threonine-protein kinase pim-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,647
- Clinical molecules 25
- Avg pChEMBL 8.21
KEGG Pathways (5)
Active Molecules (2,647)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
YUSLVKTWCYEISD
|
7.2 | IC50 | 2 | — | |
BWMLQQFMYWLLTA
|
7.2 | IC50 | 2 | — | |
DTBFDAJNODVUMF
|
7.2 | IC50 | 4 | — | |
NGYJMRVHIXLDET
|
7.2 | IC50 | 2 | — | |
OQAGQAIPXINVCL
|
7.2 | Ki | 3 | — | |
QXXPMOWWTZPKON
|
7.2 | IC50 | 3 | — | |
VJWOOBJEGKYLAB
|
7.2 | IC50 | 2 | — | |
VQNVMWNZONLRRO
|
7.2 | IC50 | 5 | — | |
WBSAJBTWVPKTJT
|
7.2 | IC50 | 2 | — | |
XDPJTYJYUSGOBW
|
7.2 | IC50 | 3 | — | |
ZBCKBGNGRYQRDG
|
7.2 | IC50 | 3 | — | |
HGGDKROMZVBKPS
|
7.2 | Ki | 2 | — | |
PGRHMLHEMDGMJC
|
7.2 | IC50 | 3 | — | |
FKXULRCNBDSLOP
|
7.2 | IC50 | 2 | — | |
IPFSIVVOJSEJOL
|
7.2 | IC50 | 5 | — | |
BWVXJRCNKNGHQO
|
7.2 | IC50 | 2 | — | |
FVBZRBVWVRMHGP
|
7.2 | IC50 | 4 | — | |
MEEVFCYRSMGEPY
|
7.2 | Ki | 2 | — | |
PRQMWOGCLLGXFR
|
7.2 | IC50 | 3 | — | |
QDWLLJBVOXFDPM
|
7.2 | IC50 | 3 | — | |
DASFSPDIWCMVRW
|
7.2 | Ki | 21 | — | |
GCBJDOWIQHMCMR
|
7.2 | Ki | 84 | — | |
IPKHSYHXXAIZDD
|
7.2 | Ki | 18 | — | |
PUYIXDDMOUMMRR
|
7.2 | Ki | 27 | — | |
LFARYXBOQBLUCT
|
7.2 | IC50 | 4 | — | |
LMKPQMOEIJCWGT
|
7.2 | Ki | 2 | — | |
ONHQPZWMSNCSPQ
|
7.2 | IC50 | 4 | — | |
PRGPHFAZQFQXGO
|
7.2 | IC50 | 3 | — | |
SBIZDCXHNTXPFJ
|
7.2 | IC50 | 2 | — | |
ICHMDGWTFDJDKG
|
7.2 | IC50 | 3 | — | |
NTSRRTDSNYXRJQ
|
7.2 | IC50 | 2 | — | |
SJHSISOAEIVKHQ
|
7.2 | Ki | 2 | — | |
VOMLURQXSWZQTM
|
7.2 | IC50 | 2 | — | |
ZRRGYYZOLYHGAW
|
7.2 | IC50 | 2 | — | |
AAXDVSTZQJTQAT
|
7.2 | IC50 | 2 | — | |
ALBGFVLKMMXQOA
|
7.2 | IC50 | 2 | — | |
HDYFVAJZXGMYBL
|
7.2 | IC50 | 2 | — | |
JNBVAICFZXTBFR
|
7.2 | IC50 | 2 | — | |
JPELSCGIWMCOQI
|
7.2 | IC50 | 3 | — | |
UGKGADDXINSGDU
|
7.2 | IC50 | 2 | — | |
UMGDPWHBQYJXAW
|
7.2 | IC50 | 2 | — | |
USWKUNURYXQEGK
|
7.2 | IC50 | 3 | — | |
AOIQLUCEVDVFMD
|
7.2 | IC50 | 2 | — | |
APORZEWICVAJLV
|
7.2 | IC50 | 2 | — | |
CIWKLGOVYCXUEM
|
7.2 | IC50 | 2 | — | |
JKBYIWGVODPSLG
|
7.2 | IC50 | 2 | — | |
KGBVDJBWYKPEQH
|
7.2 | IC50 | 2 | — | |
KLARKHWRPZGSDO
|
7.2 | IC50 | 4 | — | |
PRLYAWMVWDZNRR
|
7.2 | IC50 | 2 | — | |
REDBALFMTAGWMV
|
7.2 | IC50 | 2 | — |