Target Details
| UniProt AC | P11309 |
|---|---|
| Gene Symbol | PIM1 |
| Protein Name | Serine/threonine-protein kinase pim-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,647
- Clinical molecules 25
- Avg pChEMBL 8.21
KEGG Pathways (5)
Active Molecules (2,647)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NTBQVSFBQPCPSN
|
7.3 | IC50 | 2 | — | |
QYHNDVSXGOYYML
|
7.3 | IC50 | 2 | — | |
WMRKCEAEBWUZOS
|
7.3 | IC50 | 2 | — | |
HETRNUQWOLKNPR
|
7.3 | Ki | 2 | — | |
XCOFVVDVCWPAKU
|
7.3 | IC50 | 3 | — | |
YNACXPCSBHKFII
|
7.3 | Ki | 3 | — | |
BLWKVHOHRHEESG
|
7.3 | IC50 | 2 | — | |
HNZBELVVHGZHII
|
7.3 | Ki | 5 | — | |
IBHWJOWTGROPBE
|
7.3 | IC50 | 2 | — | |
NKGLJTITEFZKAN
|
7.3 | Ki | 35 | — | |
OAVGBZOFDPFGPJ
|
7.3 | IC50 | 42 | Yes | |
PUOHSGKCNIZLIO
|
7.3 | IC50 | 2 | — | |
UOXLVUGEYRRGOI
|
7.3 | IC50 | 2 | — | |
WPKXXVMGORDACP
|
7.3 | IC50 | 2 | — | |
ZLBGPWHOXABCIP
|
7.3 | Ki | 3 | — | |
CBHIHNZQLLGLIM
|
7.3 | IC50 | 3 | — | |
NRLTZCOPEPALOW
|
7.3 | IC50 | 2 | — | |
SIJKOQWJVVMYBK
|
7.3 | IC50 | 2 | — | |
UMWOBMRFTWBYTM
|
7.3 | IC50 | 2 | — | |
UYQKRAKNSZLAGM
|
7.3 | IC50 | 3 | — | |
ZUBJROMQSSOPHK
|
7.3 | IC50 | 2 | — | |
ZWDQRWWMKAKDAQ
|
7.3 | IC50 | 2 | — | |
ASMLDRAEBPYENO
|
7.3 | IC50 | 10 | — | |
BOIHZJDLVMPWRM
|
7.3 | IC50 | 2 | — | |
GQGBNSOWWUUWLC
|
7.3 | IC50 | 2 | — | |
JLQSMFNIARXKCU
|
7.3 | IC50 | 3 | — | |
LBKHGMSDKVXRDB
|
7.3 | IC50 | 2 | — | |
LBKHGMSDKVXRDB
|
7.3 | IC50 | 2 | — | |
PKEFFRGRYXIQIF
|
7.3 | IC50 | 2 | — | |
UCPHIHXQZQEBRG
|
7.3 | IC50 | 2 | — | |
ITUYHNBWFITURV
|
7.3 | IC50 | 2 | — | |
LUJRXDRGQWULDY
|
7.3 | IC50 | 2 | — | |
XBXBORDUPDOLCE
|
7.3 | IC50 | 2 | — | |
XLYVQVWMTOLDNL
|
7.3 | IC50 | 21 | — | |
XLYVQVWMTOLDNL
|
7.3 | IC50 | 21 | — | |
ACGIDZCOGGWWNN
|
7.3 | IC50 | 3 | — | |
CQZYFTGZTQNFBI
|
7.3 | IC50 | 2 | — | |
GENMMDLXJLCFEL
|
7.3 | IC50 | 3 | — | |
OBNFJKLGXLFJKC
|
7.3 | IC50 | 3 | — | |
POCZBHBFCIWCCV
|
7.3 | IC50 | 5 | — | |
RLKAUHPQJBOSEB
|
7.3 | IC50 | 2 | — | |
RYSQBFTZOVSXES
|
7.3 | IC50 | 2 | — | |
SGBJKPOASLHDBO
|
7.3 | IC50 | 2 | — | |
SIDJSVHZOQKDIN
|
7.3 | IC50 | 2 | — | |
VHXQWLMFJNVBML
|
7.3 | IC50 | 2 | — | |
XRNVABDYQLHODA
|
7.3 | IC50 | 3 | — | |
DHNGJAGYNYNKKJ
|
7.2 | IC50 | 3 | — | |
JZBBTWBWAAABLO
|
7.2 | IC50 | 2 | — | |
KJQXCNJCWBIKFK
|
7.2 | Ki | 3 | — | |
RXDFGEFKYADZNK
|
7.2 | Ki | 3 | — |