Target Details
| UniProt AC | P11309 |
|---|---|
| Gene Symbol | PIM1 |
| Protein Name | Serine/threonine-protein kinase pim-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,647
- Clinical molecules 25
- Avg pChEMBL 8.21
KEGG Pathways (5)
Active Molecules (2,647)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CKRMSGUCWWVREC
|
10.3 | IC50 | 3 | — | |
DFRBAIKCWZMMMO
|
10.3 | IC50 | 3 | — | |
DXLJDEPUAKIDEU
|
10.3 | IC50 | 3 | — | |
IWHCZHJFBABLPW
|
10.3 | IC50 | 3 | — | |
KCTVGDJYWANSPP
|
10.3 | IC50 | 3 | — | |
KJJNLSMGLGFZKA
|
10.3 | IC50 | 3 | — | |
KKTIVBUXNOFPPA
|
10.3 | IC50 | 3 | — | |
KYXJMCQQNZDWIT
|
10.3 | IC50 | 3 | — | |
PCYKKOGKWQRTHA
|
10.3 | IC50 | 3 | — | |
QXAYUMXTGXOKMA
|
10.3 | IC50 | 3 | — | |
SRRKWAYGAFFJAH
|
10.3 | IC50 | 3 | — | |
UEPBAYVBVVMZEN
|
10.3 | IC50 | 3 | — | |
UNUIYTCZSVJTMB
|
10.3 | IC50 | 3 | — | |
UORSWGPLCPBYOP
|
10.3 | IC50 | 3 | — | |
WDZRXBBDZLKEFS
|
10.3 | IC50 | 3 | — | |
WPKXXVMGORDACP
|
10.3 | IC50 | 2 | — | |
XEQARXMAIVALIC
|
10.3 | IC50 | 3 | — | |
YNWQVSDBNPDGBY
|
10.3 | IC50 | 3 | — | |
ZCTSKEOHMXXIST
|
10.3 | IC50 | 3 | — | |
DSEZYCNDQGVNMS
|
10.3 | Ki | 3 | — | |
SLOPAQZOFGEXBY
|
10.3 | Ki | 3 | — | |
JIEGLKQWELHCHA
|
10.3 | Ki | 3 | — | |
QBMHBUSZNODSPS
|
10.2 | Ki | 3 | — | |
CDQXYOYHHLAARJ
|
10.2 | Ki | 3 | — | |
NZMKTUOUHOLJCW
|
10.2 | Ki | 3 | — | |
VFYCNKMVBINXBE
|
10.2 | IC50 | 2 | — | |
BVSPZNRNBYKDLE
|
10.2 | Ki | 3 | — | |
BZGCHCBKEVJNKB
|
10.2 | Ki | 3 | — | |
CBXHYUCLQVWOJZ
|
10.2 | IC50 | 2 | — | |
DTOJGRXBNXZBHP
|
10.2 | IC50 | 3 | — | |
DWZMCUJAYLNSOB
|
10.2 | IC50 | 2 | — | |
JVMZLXCDQMDOEH
|
10.2 | IC50 | 3 | — | |
MMOSRHUYBPJLSR
|
10.2 | IC50 | 3 | — | |
QMBLOFSJYILYLC
|
10.2 | IC50 | 3 | — | |
SMKDKOFQQMLFPP
|
10.2 | IC50 | 3 | — | |
UXHFURUISHIEFX
|
10.2 | IC50 | 3 | — | |
UZSKGLPUMSUOBY
|
10.2 | Ki | 3 | — | |
XXTLQVLGJWHTST
|
10.2 | Ki | 3 | — | |
UMPRJLHPSRTEEA
|
10.2 | Ki | 3 | — | |
ZSSJFQNBWZACGS
|
10.2 | Ki | 3 | — | |
NZEBBXTUICPDQF
|
10.2 | Ki | 3 | — | |
AVOZYOVWQGVLHZ
|
10.2 | Ki | 3 | — | |
OLFGXMCJTMYBMY
|
10.2 | IC50 | 2 | — | |
MHBGRNASPWNGMV
|
10.2 | Ki | 3 | — | |
OIZRMKSUYVZCDN
|
10.2 | Ki | 3 | — | |
OSJCCDKQCYGFSD
|
10.2 | Ki | 3 | — | |
NAXPQDDUXNEVAM
|
10.2 | Ki | 3 | — | |
CRQPGRMAMXKTSC
|
10.2 | Ki | 3 | — | |
LDCFHYFYINOQIH
|
10.2 | IC50 | 2 | — | |
MLAWVMHISKOVHW
|
10.2 | IC50 | 3 | — |