Target Details
| UniProt AC | P11309 |
|---|---|
| Gene Symbol | PIM1 |
| Protein Name | Serine/threonine-protein kinase pim-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,647
- Clinical molecules 25
- Avg pChEMBL 8.21
KEGG Pathways (5)
Active Molecules (2,647)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SIJCUIFJKVCQLY
|
7.5 | IC50 | 2 | — | |
VKEUENNFSYBBIP
|
7.5 | IC50 | 2 | — | |
XFOBAYGKLHISDN
|
7.5 | IC50 | 2 | — | |
ZWJAIKDUVQVDKA
|
7.5 | IC50 | 2 | — | |
CSMZHIBTZOWELW
|
7.5 | IC50 | 3 | — | |
IGHMJKWWOGRBRK
|
7.5 | IC50 | 2 | — | |
JTSLALYXYSRPGW
|
7.5 | Kd | 8 | — | |
KLSMNUWOPFTNED
|
7.5 | IC50 | 4 | — | |
RRJABROJIAQAMF
|
7.5 | IC50 | 2 | — | |
VPOWFKFQCPHERH
|
7.5 | IC50 | 2 | — | |
VXHZPRIZADWWCX
|
7.5 | IC50 | 3 | — | |
ZZXFFCMCDXONOF
|
7.5 | IC50 | 4 | — | |
AERKBGXWIRADDM
|
7.5 | IC50 | 2 | — | |
UUGYRWZDBLILPN
|
7.5 | IC50 | 2 | — | |
AOOOVPXXJPJQMK
|
7.4 | IC50 | 2 | — | |
FBWNNWKXBOZFGD
|
7.4 | IC50 | 2 | — | |
GQZLEGHBRKPDDJ
|
7.4 | IC50 | 2 | — | |
JTQIPRFASTWFSP
|
7.4 | Ki | 2 | — | |
MRNSXEQVKISUCA
|
7.4 | IC50 | 3 | — | |
OINUTZGUCFIHAF
|
7.4 | IC50 | 3 | — | |
TWVUWPGFFNHEDT
|
7.4 | Ki | 2 | — | |
WRWXDAAODUAFDL
|
7.4 | Ki | 2 | — | |
XUBFCYANDUSCNL
|
7.4 | IC50 | 2 | — | |
PHIHTBDQZOPXAF
|
7.4 | IC50 | 3 | — | |
AEFFENQISAXIKE
|
7.4 | IC50 | 9 | — | |
ATOJNTJIPUYZJC
|
7.4 | IC50 | 3 | — | |
CSNKQXLBFBGYCU
|
7.4 | Ki | 3 | — | |
DWRQBWXBAGAKJH
|
7.4 | IC50 | 4 | — | |
HSCGIZGJUXQGHW
|
7.4 | IC50 | 2 | — | |
KGFURSRTCYARCY
|
7.4 | IC50 | 3 | — | |
KRZFOHDWKJHXLR
|
7.4 | IC50 | 3 | — | |
LNPQKOKBBJUSNM
|
7.4 | IC50 | 2 | — | |
MESZFHDSIOYFJC
|
7.4 | IC50 | 3 | — | |
MWKSRKSEWLRPBL
|
7.4 | Kd | 1075 | — | |
XQXCEKIWYGDQJP
|
7.4 | IC50 | 2 | — | |
YBSGHQWNCMWAPW
|
7.4 | IC50 | 2 | — | |
AJYJGZPVGQOKOB
|
7.4 | IC50 | 2 | — | |
JBAKTVVTRACTOI
|
7.4 | IC50 | 2 | — | |
JRYFWOLNIOKGSO
|
7.4 | IC50 | 2 | — | |
OEJMEIAMVNPZBT
|
7.4 | Ki | 3 | — | |
ORIZHSWHRATWPB
|
7.4 | IC50 | 2 | — | |
QLQXQPDNKGTPIA
|
7.4 | IC50 | 2 | — | |
WAISNUDWNYJNMT
|
7.4 | IC50 | 3 | — | |
XODCTWLLGVOGFI
|
7.4 | IC50 | 4 | — | |
AOOOSENPXVAGON
|
7.4 | IC50 | 2 | — | |
BXADXKNHUSVYFU
|
7.4 | Ki | 2 | — | |
CTANUMSASKECMC
|
7.4 | IC50 | 2 | — | |
JAXWDNNZTVFOMJ
|
7.4 | IC50 | 2 | — | |
KAKGFGCTONHQJW
|
7.4 | Ki | 25 | — | |
OEZGLXNWDIQDMU
|
7.4 | IC50 | 2 | — |