Target Details
| UniProt AC | P11309 |
|---|---|
| Gene Symbol | PIM1 |
| Protein Name | Serine/threonine-protein kinase pim-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,647
- Clinical molecules 25
- Avg pChEMBL 8.21
KEGG Pathways (5)
Active Molecules (2,647)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
BGNRMTUXZUCPDO
|
7.5 | IC50 | 3 | — | |
PBLUDSMVIHVGIX
|
7.5 | IC50 | 2 | — | |
ARNUKQRNOOIEGV
|
7.5 | IC50 | 2 | — | |
DDANOGFWWHHVPP
|
7.5 | IC50 | 2 | — | |
DLVABOPQYSXZPM
|
7.5 | IC50 | 2 | — | |
DVANQYCQWXMWPM
|
7.5 | IC50 | 2 | — | |
FZEITOZYNXRCOT
|
7.5 | IC50 | 2 | — | |
GLYWPANTIWPDCD
|
7.5 | IC50 | 2 | — | |
HWMYTSVQLOTTGQ
|
7.5 | IC50 | 2 | — | |
JBJTUZIBTZMMOG
|
7.5 | IC50 | 2 | — | |
JHWKXDBSEDXRAD
|
7.5 | IC50 | 2 | — | |
JZMTWKROJYCQEE
|
7.5 | IC50 | 3 | — | |
NIFSXAKUQWXUEQ
|
7.5 | IC50 | 2 | — | |
OXTPERZFYREBFH
|
7.5 | IC50 | 3 | — | |
PITNXTPXOPNHEK
|
7.5 | IC50 | 2 | — | |
QQCWPCSHFHPVFD
|
7.5 | IC50 | 2 | — | |
RDPUEIZFSORAPJ
|
7.5 | IC50 | 2 | — | |
SGUNCNYHPYXQNG
|
7.5 | IC50 | 2 | — | |
UGOKMGYEFGBJST
|
7.5 | Ki | 2 | — | |
VFFKOUSSVDBQAF
|
7.5 | IC50 | 5 | Yes | |
WLJWSUVXFQUAHY
|
7.5 | IC50 | 3 | — | |
CMILZUZLXJQSGJ
|
7.5 | IC50 | 2 | — | |
DGJWAGBAIDNRCG
|
7.5 | IC50 | 2 | — | |
HIRGJKYVLHTQTI
|
7.5 | IC50 | 3 | — | |
IFSZNNCMCGMAHD
|
7.5 | IC50 | 4 | — | |
KIBZGUOKQUDIFC
|
7.5 | Ki | 3 | — | |
KPCHRAXFURQEBV
|
7.5 | IC50 | 5 | — | |
NDNWVNFWIGICKO
|
7.5 | Ki | 3 | — | |
NPHICJWCOYEVRI
|
7.5 | IC50 | 2 | — | |
PHJNQZCUTKCIGD
|
7.5 | IC50 | 2 | — | |
UAQJGBPGZKYVKD
|
7.5 | IC50 | 2 | — | |
UFARADZVZUVRAW
|
7.5 | IC50 | 2 | — | |
YNQGEMKAJKCOIP
|
7.5 | IC50 | 3 | — | |
YWJGVHDHQUUQEH
|
7.5 | IC50 | 3 | — | |
BGYVWFZMYBWCNY
|
7.5 | Ki | 30 | — | |
DPEXRCOBPACFOO
|
7.5 | Ki | 36 | — | |
DWLRROMENORWQU
|
7.5 | IC50 | 3 | — | |
HBJGQSLQQKVOJA
|
7.5 | Ki | 2 | — | |
HMKKDSBJGMESJD
|
7.5 | Ki | 10 | — | |
JEYOQYMSSQZLJL
|
7.5 | Ki | 7 | — | |
LKXSICYXJDCMQF
|
7.5 | IC50 | 3 | — | |
SLCZMHSSTXGLFD
|
7.5 | IC50 | 2 | — | |
UVGKRGCBYGNVGI
|
7.5 | IC50 | 2 | — | |
XPRWPAHCXZUIPP
|
7.5 | IC50 | 5 | — | |
DNTVXDZWVOVLOD
|
7.5 | IC50 | 5 | — | |
ZJOSEGOSWVWPDQ
|
7.5 | IC50 | 3 | — | |
KCXFEPOPVGRWEO
|
7.5 | IC50 | 2 | — | |
NIRJXKZEFQTBIC
|
7.5 | IC50 | 2 | — | |
ONBYHZKTWDQADU
|
7.5 | IC50 | 2 | — | |
BVWMTYDPXCWJOP
|
7.5 | IC50 | 2 | — |