Target Details
| UniProt AC | P11309 |
|---|---|
| Gene Symbol | PIM1 |
| Protein Name | Serine/threonine-protein kinase pim-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,647
- Clinical molecules 25
- Avg pChEMBL 8.21
KEGG Pathways (5)
Active Molecules (2,647)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RTBZFULAXSZFTC
|
7.6 | IC50 | 2 | — | |
RUGJASFMGVWDAX
|
7.6 | IC50 | 2 | — | |
SNBKWZURQXFUQV
|
7.6 | IC50 | 2 | — | |
TWESPFOMZINAFH
|
7.6 | IC50 | 2 | — | |
VNGYQBMDQMDALH
|
7.6 | Ki | 25 | — | |
WHSNSKLEZGKYLB
|
7.6 | IC50 | 2 | — | |
AHFVIIAVAVUYKX
|
7.6 | IC50 | 3 | — | |
DKQVDFIPXRLAHK
|
7.6 | IC50 | 3 | — | |
LCPPDMKTNXVYBC
|
7.6 | IC50 | 2 | — | |
ZJVSOYXGSBGVDG
|
7.6 | IC50 | 3 | — | |
BVFUBYDIYASTFC
|
7.6 | IC50 | 2 | — | |
DQHDWRILUICKSN
|
7.6 | IC50 | 2 | — | |
HEMOXCULECZESD
|
7.6 | IC50 | 2 | — | |
JVSVOIZZHBUDNG
|
7.6 | IC50 | 2 | — | |
KFBFNFWYBBFFDY
|
7.6 | IC50 | 2 | — | |
KJZOQUBRACKVFA
|
7.6 | IC50 | 2 | — | |
MOZUWJVTBZTPTJ
|
7.6 | IC50 | 3 | — | |
WMRKCEAEBWUZOS
|
7.6 | IC50 | 2 | — | |
ZDGGLAZWYAXWTN
|
7.6 | Ki | 3 | — | |
ATMAGFPFVYJWHA
|
7.6 | IC50 | 3 | — | |
DAELCQFOTJBMKB
|
7.6 | IC50 | 2 | — | |
DKGRYLGTOXMKFX
|
7.6 | IC50 | 2 | — | |
DQYBRTASHMYDJG
|
7.6 | Kd | 13 | Yes | |
HIQSWPMUNKYMHE
|
7.6 | IC50 | 4 | — | |
LTUJVSFHKWFNCG
|
7.6 | IC50 | 2 | — | |
OOINHKLROPYETD
|
7.6 | IC50 | 3 | — | |
QMGUOJYZJKLOLH
|
7.6 | IC50 | 21 | Yes | |
WYRRPQWTIXERBJ
|
7.6 | IC50 | 2 | — | |
YOXRHHNVUJXJFA
|
7.6 | IC50 | 3 | — | |
DSXHSERBBFHDMQ
|
7.6 | IC50 | 3 | — | |
GXSHWBSAHCQKFV
|
7.6 | IC50 | 2 | — | |
DNXZIJKGPFJRAA
|
7.5 | IC50 | 3 | — | |
DOERTQQDUFOAOA
|
7.5 | IC50 | 2 | — | |
ITKWGXVYWSDMPF
|
7.5 | Ki | 3 | — | |
KWTSXUHMAHLNMY
|
7.5 | IC50 | 2 | — | |
OOYZNZPKFQSWHZ
|
7.5 | IC50 | 3 | — | |
PHERSJGVHFLHAP
|
7.5 | IC50 | 5 | — | |
PYLMTZUQBJXIQJ
|
7.5 | IC50 | 3 | — | |
RAALJCORRJVBNY
|
7.5 | IC50 | 2 | — | |
RRXLHFUTCAGGON
|
7.5 | IC50 | 2 | — | |
VHAIPPXUMKWXIR
|
7.5 | IC50 | 2 | — | |
YQOPMWZYUDDIAP
|
7.5 | IC50 | 2 | — | |
AJEKKBSRNRYYET
|
7.5 | IC50 | 3 | — | |
CZZCAOGIEGXMBZ
|
7.5 | IC50 | 10 | — | |
DCLLXJAPIKAKPL
|
7.5 | IC50 | 2 | — | |
GVJNYUQTRLLCQS
|
7.5 | IC50 | 3 | — | |
IPHOLKTXQVULGA
|
7.5 | IC50 | 9 | — | |
LWHTZTIHIFBTMB
|
7.5 | IC50 | 3 | — | |
RRHKBGWLQRCEFH
|
7.5 | Ki | 2 | — | |
ZZQKMYABUGJCHQ
|
7.5 | IC50 | 2 | — |