Target Details
| UniProt AC | P11309 |
|---|---|
| Gene Symbol | PIM1 |
| Protein Name | Serine/threonine-protein kinase pim-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,647
- Clinical molecules 25
- Avg pChEMBL 8.21
KEGG Pathways (5)
Active Molecules (2,647)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WXIKUAVDMWNARE
|
7.7 | IC50 | 3 | — | |
XLHVTKIMNYRMGW
|
7.7 | IC50 | 2 | — | |
ZQGMAEVBUDWZSM
|
7.7 | IC50 | 2 | — | |
CUWAPHLUSJWBCU
|
7.7 | IC50 | 2 | — | |
RLFQVKISFLTJNU
|
7.7 | IC50 | 3 | — | |
CQOAYBZZYRBDJZ
|
7.7 | IC50 | 2 | — | |
GOKWYLQQNCJARE
|
7.7 | Ki | 2 | — | |
GVUXAQWOKREQBF
|
7.7 | IC50 | 4 | — | |
HXWWNIUEVOHPKT
|
7.7 | Ki | 3 | — | |
NLIRZAJMWQYPLA
|
7.7 | IC50 | 2 | — | |
QWCZNBVUCFOLSB
|
7.7 | IC50 | 2 | — | |
UOMPPOVQMYNXST
|
7.7 | IC50 | 2 | — | |
YVTVCGFWYNABGD
|
7.7 | Ki | 3 | — | |
WHJIHZSXTQRCNX
|
7.7 | IC50 | 10 | — | |
ANAOYTVZYSRWRF
|
7.6 | Ki | 3 | — | |
DEDZRZXSRZHUAQ
|
7.6 | IC50 | 2 | — | |
FGFBVVWWRFZMMR
|
7.6 | IC50 | 2 | — | |
FSVMVFNAUYVDDY
|
7.6 | IC50 | 2 | — | |
GZUBPRPQRRXDTP
|
7.6 | IC50 | 2 | — | |
HIRGJKYVLHTQTI
|
7.6 | IC50 | 3 | — | |
KKYRWGKJFKLPFO
|
7.6 | IC50 | 2 | — | |
QRVJKXOAMVIRHV
|
7.6 | IC50 | 2 | — | |
QWEBKNRGVXJIKS
|
7.6 | IC50 | 3 | — | |
USPNCTNCYQFTGT
|
7.6 | IC50 | 3 | — | |
AMFKEKUSTBMIEA
|
7.6 | IC50 | 3 | — | |
BHWVHQCCGNUXHH
|
7.6 | IC50 | 2 | — | |
MEGWNHRJENCAAU
|
7.6 | IC50 | 2 | — | |
AWLKBZZAGUKGIX
|
7.6 | IC50 | 2 | — | |
HPXHJTNCJPAWOK
|
7.6 | IC50 | 2 | — | |
KDRBBKILEOZBCW
|
7.6 | IC50 | 2 | — | |
NCUSDXPQLMTWTR
|
7.6 | IC50 | 3 | — | |
NGJLOFCOEOHFKQ
|
7.6 | IC50 | 4 | — | |
OLWSXGZFLPJRBT
|
7.6 | IC50 | 3 | — | |
PDRYKKBDIUESOF
|
7.6 | IC50 | 5 | — | |
QLPGKDRTCLALRP
|
7.6 | IC50 | 2 | — | |
RCBCKGFUIXSXGK
|
7.6 | IC50 | 2 | — | |
SGQNOLAVVZNJKI
|
7.6 | IC50 | 2 | — | |
ZDHNAPJCCZPPCX
|
7.6 | IC50 | 2 | — | |
DGBIUYHHQKNLEE
|
7.6 | IC50 | 3 | — | |
LEFJKUQAFOHMGV
|
7.6 | IC50 | 3 | — | |
ZCCPLJOKGAACRT
|
7.6 | Kd | 599 | — | |
AYUREZCMYVPMPV
|
7.6 | IC50 | 2 | — | |
CNWMKSDNKYKWRI
|
7.6 | Ki | 2 | — | |
DFHQXRLKAFZKPB
|
7.6 | IC50 | 3 | — | |
DRAKVWYEJUJMPG
|
7.6 | IC50 | 2 | — | |
FCGLYPSBPNFQRF
|
7.6 | IC50 | 3 | — | |
GVOOEMLKTIRYCO
|
7.6 | Ki | 7 | — | |
IVHFBERBIURXGC
|
7.6 | IC50 | 2 | — | |
PFFNHXNHPCGMCF
|
7.6 | IC50 | 2 | — | |
PGBRENJGANITFP
|
7.6 | IC50 | 2 | — |