Target Details
| UniProt AC | P11309 |
|---|---|
| Gene Symbol | PIM1 |
| Protein Name | Serine/threonine-protein kinase pim-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,647
- Clinical molecules 25
- Avg pChEMBL 8.21
KEGG Pathways (5)
Active Molecules (2,647)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
AECUWGQUPZABQT
|
7.7 | IC50 | 2 | — | |
BLBAWGODFTZAEY
|
7.7 | IC50 | 2 | — | |
DUFBPFBIIKCZOK
|
7.7 | IC50 | 2 | — | |
FCQWHYNQCKOSRV
|
7.7 | IC50 | 3 | — | |
NHWNYDXOYLBMJG
|
7.7 | IC50 | 2 | — | |
NKXSGMQFDUZNPT
|
7.7 | IC50 | 3 | — | |
OZFLDPINWWCZMD
|
7.7 | IC50 | 3 | — | |
SUWUBTVCKQZMPW
|
7.7 | IC50 | 4 | — | |
UPTADSCUUNQNDI
|
7.7 | IC50 | 2 | — | |
YCKUAKXRPAUDMQ
|
7.7 | IC50 | 2 | — | |
ZZQKMYABUGJCHQ
|
7.7 | IC50 | 2 | — | |
RMTAUHCHXYNQOT
|
7.7 | IC50 | 3 | — | |
RTFAQLBYFHKCPR
|
7.7 | IC50 | 2 | — | |
BUZDEHLSGHZEBZ
|
7.7 | Ki | 2 | — | |
CNGZGBQVACJCTJ
|
7.7 | IC50 | 2 | — | |
DZPWHGFOCWIUKE
|
7.7 | Ki | 3 | — | |
FGQCVFKIQHFEDF
|
7.7 | IC50 | 2 | — | |
GJSKIXCETHIGQQ
|
7.7 | IC50 | 3 | — | |
HYSKVGJVSDFOHZ
|
7.7 | IC50 | 2 | — | |
JCYRBMWQKSQMPU
|
7.7 | IC50 | 2 | — | |
JPSRNNAKSXAWPL
|
7.7 | IC50 | 2 | — | |
KLGUOFQVXLDGTK
|
7.7 | IC50 | 2 | — | |
KPYXZOZRPALMPX
|
7.7 | IC50 | 2 | — | |
LCOVSYDTOHZUSS
|
7.7 | IC50 | 5 | — | |
MBDNHHKZEBJSRM
|
7.7 | IC50 | 2 | — | |
MCKDPRWMNDLDPP
|
7.7 | IC50 | 2 | — | |
OOKQFYPMRWKVRB
|
7.7 | IC50 | 3 | — | |
PHWHNHYZZNJPLB
|
7.7 | Ki | 16 | — | |
UDGYUGQHPSWDMW
|
7.7 | IC50 | 2 | — | |
VHNDENLQTFRWOM
|
7.7 | IC50 | 2 | — | |
VSYLYSOTCDFRSM
|
7.7 | IC50 | 2 | — | |
WJEUVIUVISQACN
|
7.7 | IC50 | 2 | — | |
WPQVIQXQVLVSIJ
|
7.7 | IC50 | 2 | — | |
ZCBUQCWBWNUWSU
|
7.7 | Ki | 11 | — | |
ZLDXTUTZYPVCKG
|
7.7 | IC50 | 3 | — | |
DJNAAVCOMOYFNT
|
7.7 | IC50 | 3 | — | |
NGHKXECWEKEJAN
|
7.7 | Ki | 3 | — | |
OUKYCHWOBSPIBT
|
7.7 | IC50 | 2 | — | |
BEGMGTVTJSZGTO
|
7.7 | IC50 | 3 | — | |
BMYXNSDMYMRNAW
|
7.7 | IC50 | 3 | — | |
CHYPUQGSRVSROE
|
7.7 | IC50 | 2 | — | |
HDECOLDRAJGUTB
|
7.7 | IC50 | 3 | — | |
HVQKSMUBAKDZPC
|
7.7 | IC50 | 2 | — | |
HYTFYLWLSNWHGV
|
7.7 | IC50 | 2 | — | |
JWYMKPOZFIRRBB
|
7.7 | IC50 | 3 | — | |
KBYVWOCCWQCSGX
|
7.7 | IC50 | 2 | — | |
LHJWKHNEQQVHNI
|
7.7 | IC50 | 2 | — | |
PSBYBDMPXANZIE
|
7.7 | IC50 | 2 | — | |
SENFEQVLOFSJFU
|
7.7 | Ki | 3 | Yes | |
UCSBUXYSZFPGSI
|
7.7 | IC50 | 3 | — |