Target Details
| UniProt AC | P11309 |
|---|---|
| Gene Symbol | PIM1 |
| Protein Name | Serine/threonine-protein kinase pim-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,647
- Clinical molecules 25
- Avg pChEMBL 8.21
KEGG Pathways (5)
Active Molecules (2,647)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MEQUDKNTYPMAEZ
|
7.8 | IC50 | 2 | — | |
MPKGZYZIJRTCNU
|
7.8 | IC50 | 4 | — | |
NJUKVCLHVLPDAP
|
7.8 | Ki | 3 | — | |
PKUDLMDWOHMCHC
|
7.8 | Ki | 3 | — | |
PRHPCWAJDWRBJW
|
7.8 | IC50 | 3 | — | |
PZGOKNURFTXNGH
|
7.8 | IC50 | 2 | — | |
QBGYLZQNONTKJL
|
7.8 | IC50 | 2 | — | |
SARSRHFTCLKGJD
|
7.8 | Ki | 2 | — | |
SLRQWILFIQMPFZ
|
7.8 | IC50 | 3 | — | |
WQCAIEFWZIYFLE
|
7.8 | IC50 | 2 | — | |
ZFJYBIDCQXNLFR
|
7.8 | IC50 | 2 | — | |
PDVZWQUTIFENGJ
|
7.8 | IC50 | 2 | — | |
UMFRMBNWQDGSCQ
|
7.8 | IC50 | 2 | — | |
FPUFRVZXLSMBNG
|
7.8 | IC50 | 3 | — | |
NTBQVSFBQPCPSN
|
7.8 | IC50 | 2 | — | |
PKFIEHJDQBPPOI
|
7.8 | IC50 | 3 | — | |
VWNWDNDEKMMIHM
|
7.8 | IC50 | 3 | — | |
BHNFVXISRPMSCV
|
7.8 | IC50 | 4 | — | |
CMNCIJKGYUUTDZ
|
7.8 | IC50 | 3 | — | |
DUIYQEGWIKOTCS
|
7.8 | Ki | 3 | — | |
FPGQJZNMSHOCKW
|
7.8 | IC50 | 4 | — | |
FSQNGXYJUMATLF
|
7.8 | IC50 | 3 | — | |
GQCFPBDBAMWOAP
|
7.8 | IC50 | 2 | — | |
GQCHSJRNLCGUAC
|
7.8 | IC50 | 3 | — | |
IAYHXSKNPQYTOD
|
7.8 | IC50 | 3 | — | |
OCDUTTRLHDUQLY
|
7.8 | IC50 | 2 | — | |
RKJBOGXNNPWZEW
|
7.8 | Ki | 2 | — | |
UGRPNQCFWPYERM
|
7.8 | IC50 | 5 | — | |
USZMAOOUNPYUGA
|
7.8 | IC50 | 2 | — | |
VCOMCNXJZDHONQ
|
7.8 | IC50 | 2 | — | |
YOXRHHNVUJXJFA
|
7.8 | IC50 | 3 | — | |
OAFRMXFROSZIEC
|
7.8 | IC50 | 3 | — | |
QWCWGAZSLRLOPF
|
7.8 | IC50 | 3 | — | |
ACWWBXAGCBHIGJ
|
7.8 | IC50 | 2 | — | |
MABMEAYNQCJUKG
|
7.8 | IC50 | 3 | — | |
RCQQWKQETBJWOO
|
7.8 | IC50 | 3 | — | |
APMKLXLBNBDHBU
|
7.7 | IC50 | 2 | — | |
BQEKYURMJHGZAW
|
7.7 | IC50 | 2 | — | |
CXGNKWVDMVOVTL
|
7.7 | Ki | 3 | — | |
HNXYPVWPNANYAO
|
7.7 | IC50 | 5 | — | |
JCHKNLLUGJTBFB
|
7.7 | IC50 | 2 | — | |
LPJAKJUVEMSSSX
|
7.7 | IC50 | 9 | — | |
MSNPLCILYPRIGG
|
7.7 | IC50 | 2 | — | |
ODHWZXUUXOFUQZ
|
7.7 | IC50 | 3 | — | |
OQMBYFPSIKELDN
|
7.7 | IC50 | 3 | — | |
OZGYSJHDOKWOOY
|
7.7 | IC50 | 3 | — | |
SHXZNKIVNYEJBF
|
7.7 | IC50 | 2 | — | |
VYHCLYDDXNTHAU
|
7.7 | IC50 | 4 | — | |
ZRPRPAYPNUQSQH
|
7.7 | IC50 | 2 | — | |
WIAJWDVLVSAMRU
|
7.7 | IC50 | 2 | — |