Target Details
| UniProt AC | P11309 |
|---|---|
| Gene Symbol | PIM1 |
| Protein Name | Serine/threonine-protein kinase pim-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,647
- Clinical molecules 25
- Avg pChEMBL 8.21
KEGG Pathways (5)
Active Molecules (2,647)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GPAPAMNDJCEOJQ
|
7.8 | IC50 | 2 | — | |
HDYFVAJZXGMYBL
|
7.8 | IC50 | 2 | — | |
HKOKUJNLAMXOED
|
7.8 | IC50 | 3 | — | |
JKSFANMDRYVNBI
|
7.8 | IC50 | 4 | — | |
JTUMZSSZJKUTNF
|
7.8 | IC50 | 2 | — | |
LHKDWQFFBVATPU
|
7.8 | IC50 | 2 | — | |
LRUMZQFUWNWSQL
|
7.8 | IC50 | 2 | — | |
LVKVPSJZKQLBMV
|
7.8 | IC50 | 5 | — | |
OTLXPFZNAMLUDF
|
7.8 | Ki | 2 | — | |
PRPKIYKNDIOAEU
|
7.8 | Ki | 2 | — | |
ULDSFJCLLURBJV
|
7.8 | IC50 | 4 | — | |
UWWMNBSTTVYINO
|
7.8 | IC50 | 4 | — | |
VZZLTWZEAQOFRD
|
7.8 | Ki | 3 | — | |
WFPLKANBSQGCJH
|
7.8 | IC50 | 2 | — | |
WZIZMFJEBARBSY
|
7.8 | IC50 | 2 | — | |
ZZFSRGVIDIVGQO
|
7.8 | IC50 | 4 | — | |
ZXQIHLJIAWEHOF
|
7.8 | IC50 | 2 | — | |
IICNWQTVBNJGKW
|
7.8 | IC50 | 2 | — | |
JLBPJFGCWQRFTF
|
7.8 | IC50 | 2 | — | |
SJQWLZPINZQQNC
|
7.8 | IC50 | 2 | — | |
BTTJTCLIZBSDNP
|
7.8 | IC50 | 8 | — | |
DAJUQGQQWWXBPE
|
7.8 | IC50 | 3 | — | |
FUGVOKHOINFPBY
|
7.8 | IC50 | 3 | — | |
FZFVXBALMLDUDW
|
7.8 | Ki | 3 | — | |
GIFPOJWPSWZZCJ
|
7.8 | IC50 | 4 | — | |
JBFFDNABQNAJAB
|
7.8 | IC50 | 4 | — | |
KLGUOFQVXLDGTK
|
7.8 | IC50 | 3 | — | |
PNAYFCPGKVJMMN
|
7.8 | IC50 | 3 | — | |
POINNGFQYFKPBA
|
7.8 | IC50 | 3 | — | |
PRLYAWMVWDZNRR
|
7.8 | IC50 | 3 | — | |
QNUFZYZRLJGZJL
|
7.8 | IC50 | 10 | — | |
QSTDMPARCWMFIJ
|
7.8 | IC50 | 4 | — | |
RQILRUHUVGWBAL
|
7.8 | IC50 | 2 | — | |
RZVRZDUJJWCVMN
|
7.8 | IC50 | 3 | — | |
SBDJADVTLNKDBC
|
7.8 | Ki | 3 | — | |
UWQLIXURTCXRJT
|
7.8 | Ki | 2 | — | |
YRVVLUIFOUTBGD
|
7.8 | Ki | 2 | — | |
AZPAUNKZBWYQME
|
7.8 | IC50 | 3 | — | |
CKASJUOAZZSCTR
|
7.8 | Ki | 3 | — | |
PAOXVIIJQNGJQF
|
7.8 | IC50 | 2 | — | |
CZXVLEKLKBMPNR
|
7.8 | IC50 | 2 | — | |
GAZLCQLGBUPWQG
|
7.8 | IC50 | 4 | — | |
GNGHBXZAZFETNZ
|
7.8 | IC50 | 2 | — | |
GPUYNLZUUOVRON
|
7.8 | IC50 | 2 | — | |
HBIPPWQOAJGLJC
|
7.8 | IC50 | 4 | — | |
HKCQYVZLEUOAFO
|
7.8 | IC50 | 3 | — | |
JCICCACMYITOCI
|
7.8 | IC50 | 3 | — | |
JIQHIGWAELIAMV
|
7.8 | IC50 | 2 | — | |
JMNGRHJERIBAHK
|
7.8 | Ki | 3 | — | |
LVPUPCZWFVIOGD
|
7.8 | IC50 | 2 | — |