Target Details
| UniProt AC | P11309 |
|---|---|
| Gene Symbol | PIM1 |
| Protein Name | Serine/threonine-protein kinase pim-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,647
- Clinical molecules 25
- Avg pChEMBL 8.21
KEGG Pathways (5)
Active Molecules (2,647)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OLONVMXDIIPFOK
|
7.9 | IC50 | 2 | — | |
PACWQXXFANARIG
|
7.9 | IC50 | 2 | — | |
PMKXIEFCLZIQLZ
|
7.9 | IC50 | 2 | — | |
PQKSGKOVSKUOPB
|
7.9 | IC50 | 3 | — | |
RCBIRPOKYRSUDB
|
7.9 | IC50 | 2 | — | |
STJQTLCHUQJELE
|
7.9 | Ki | 2 | — | |
UPTADSCUUNQNDI
|
7.9 | IC50 | 2 | — | |
UQHKJRCFSLMWIA
|
7.9 | Kd | 3 | — | |
XCFKWUCNYGYTAY
|
7.9 | Ki | 3 | — | |
XFKAPHNFSNSIFR
|
7.9 | IC50 | 3 | — | |
JTXMDYASUVCZMQ
|
7.9 | IC50 | 2 | — | |
LYSVYDGAEVIKAF
|
7.9 | IC50 | 3 | — | |
UDSJMCNBYOMONW
|
7.9 | Ki | 2 | — | |
VLCAXVDVDRCYLY
|
7.9 | IC50 | 2 | — | |
WDOAVCPYTBBYJE
|
7.9 | Ki | 2 | — | |
WUTCYYSJWLOLPF
|
7.9 | IC50 | 3 | — | |
ZUUYCPKOPFRHGK
|
7.9 | IC50 | 2 | — | |
FTQIZXVNFDCIQI
|
7.9 | Ki | 3 | — | |
GESRYDOMZCMGNO
|
7.9 | IC50 | 4 | — | |
IIFMWBFXGMFSOH
|
7.9 | IC50 | 3 | — | |
LVAZMNBKXWCIMF
|
7.9 | IC50 | 3 | — | |
STCFUYVDTGGZPT
|
7.9 | IC50 | 2 | — | |
AKOHJQLWPFONMJ
|
7.9 | IC50 | 2 | — | |
BSXBVSWEULDBKN
|
7.9 | IC50 | 2 | — | |
CSNVUBRZPKUAIT
|
7.9 | IC50 | 2 | — | |
DSIUXAXVFGLHPR
|
7.9 | IC50 | 2 | — | |
FCZYYBANBFQRMS
|
7.9 | IC50 | 2 | — | |
GFVZLOMZOSEUPY
|
7.9 | IC50 | 2 | — | |
GPICQYUBSFLTRN
|
7.9 | IC50 | 2 | — | |
LMUQPBXEPPNVJF
|
7.9 | IC50 | 2 | — | |
MCZCAWWHZGEUFE
|
7.9 | IC50 | 2 | — | |
OPRSJJZSXUUJLS
|
7.9 | IC50 | 2 | — | |
QETFAMKONUZFSO
|
7.9 | IC50 | 2 | — | |
WSZGOCPQOSHGAF
|
7.9 | IC50 | 7 | — | |
XHEYSFJJPSXTHP
|
7.9 | IC50 | 3 | — | |
XKBJDTIYSQFHST
|
7.9 | IC50 | 2 | — | |
ZXWCVIPMPJIAAK
|
7.9 | IC50 | 2 | — | |
GDPZLMJSLZTJBB
|
7.9 | IC50 | 3 | — | |
MQKXIAMASIXWJH
|
7.9 | IC50 | 2 | — | |
OLKXVDKTEYJKPA
|
7.9 | IC50 | 3 | — | |
SRRKWAYGAFFJAH
|
7.9 | IC50 | 2 | — | |
WSKIIQILRYHQCK
|
7.9 | IC50 | 2 | — | |
SNHNWCQKOINDPL
|
7.9 | IC50 | 3 | — | |
SOEBVEZGKJJGMP
|
7.9 | IC50 | 2 | — | |
QPOKFUGFTPMYSP
|
7.9 | IC50 | 2 | — | |
XQGPDQSRBACGPU
|
7.9 | IC50 | 2 | — | |
ZJOSEGOSWVWPDQ
|
7.9 | IC50 | 2 | — | |
AUPKOEHUXGYASA
|
7.8 | IC50 | 2 | — | |
DKGRYLGTOXMKFX
|
7.8 | IC50 | 2 | — | |
DKZYXHCYPUVGAF
|
7.8 | Kd | 112 | — |