Target Details
| UniProt AC | P11309 |
|---|---|
| Gene Symbol | PIM1 |
| Protein Name | Serine/threonine-protein kinase pim-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,647
- Clinical molecules 25
- Avg pChEMBL 8.21
KEGG Pathways (5)
Active Molecules (2,647)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
HQRWFKUVQLFJSA
|
8.0 | IC50 | 2 | — | |
NPLDOTMTVQWXCF
|
8.0 | IC50 | 3 | — | |
AYZUBCLOFTTWJJ
|
8.0 | IC50 | 3 | — | |
AZBLJXRSEYELKU
|
8.0 | IC50 | 2 | — | |
BNLHKRKGCKUVHA
|
8.0 | IC50 | 4 | — | |
DBFVYHGYASQAJI
|
8.0 | Ki | 3 | — | |
DYYJJDFSLFXRAV
|
8.0 | Ki | 2 | — | |
FRRLLRQAGKSVMU
|
8.0 | IC50 | 7 | — | |
GWRQOSDZGCDBHH
|
8.0 | IC50 | 3 | — | |
HTDBXCBZQPTDQB
|
8.0 | IC50 | 4 | — | |
ISYNRKKNWPXOCT
|
8.0 | Ki | 2 | — | |
JDUUXRFAIVVJFT
|
8.0 | IC50 | 2 | — | |
KBQOSTHTFJGZBY
|
8.0 | IC50 | 2 | — | |
KEJAEPZICPHNOE
|
8.0 | IC50 | 2 | — | |
MBFRJIPAANIXOT
|
8.0 | Ki | 2 | — | |
MDBOHSQFSGLDSX
|
8.0 | Ki | 2 | — | |
MEFXTBWNNFVIHA
|
8.0 | IC50 | 2 | — | |
NRHBVVQSMCFGOS
|
8.0 | IC50 | 4 | — | |
PAVPZPCSAGSHHJ
|
8.0 | IC50 | 3 | — | |
PAWYOAJXAZJAQU
|
8.0 | IC50 | 3 | — | |
RWNSOGBUKTYZJZ
|
8.0 | IC50 | 3 | — | |
SCHVVSMHPGRYLE
|
8.0 | IC50 | 2 | — | |
VJAFLWYXUBIIJD
|
8.0 | IC50 | 3 | — | |
WIPBIZXEEPHOTH
|
8.0 | IC50 | 3 | — | |
WTJOTLCUSWSEMH
|
8.0 | IC50 | 3 | — | |
WZTOVDHYAYCPOP
|
8.0 | IC50 | 5 | — | |
XLKGJWHZQCXAIX
|
8.0 | IC50 | 2 | — | |
XZFRNJKDMFEUTK
|
8.0 | IC50 | 2 | — | |
YUYSIGQIXVQKCJ
|
8.0 | IC50 | 3 | — | |
VBZISNIVQBAKDD
|
8.0 | Ki | 3 | — | |
CRDMJKIEIKHCSZ
|
7.9 | IC50 | 2 | — | |
DRQCVGYHMOTKEO
|
7.9 | Ki | 3 | — | |
KBGGFQXKCDNJOX
|
7.9 | Ki | 2 | — | |
LWAINAQZGRZKTJ
|
7.9 | IC50 | 2 | — | |
MAHUZUBWHKQCIH
|
7.9 | IC50 | 3 | — | |
OPYBFXSLCXMZGR
|
7.9 | IC50 | 2 | — | |
FZTSRAGTHKAPKA
|
7.9 | Ki | 3 | — | |
IXLHWDDKCRTAAT
|
7.9 | IC50 | 4 | — | |
OSAJYFUYGLKCLG
|
7.9 | IC50 | 2 | — | |
PKUYPRFEWPYLAU
|
7.9 | IC50 | 2 | — | |
YYOZRZRSLJUTAW
|
7.9 | IC50 | 2 | — | |
BKDNXYLZMURERH
|
7.9 | IC50 | 3 | — | |
CNJCQHGFLOVMGJ
|
7.9 | IC50 | 3 | — | |
DJOXKKRRSXGVNT
|
7.9 | Ki | 2 | — | |
KREARTJFHWAQOG
|
7.9 | IC50 | 2 | — | |
LVJGPCQGQKMJHE
|
7.9 | IC50 | 3 | — | |
MSOLNCSVZOTSMV
|
7.9 | IC50 | 2 | — | |
NBZYCEPNLRVSAP
|
7.9 | IC50 | 3 | — | |
NEJSXCPIDIEJKT
|
7.9 | IC50 | 4 | — | |
NLQUZLBPOZVPHA
|
7.9 | IC50 | 3 | — |