Target Details
| UniProt AC | P11309 |
|---|---|
| Gene Symbol | PIM1 |
| Protein Name | Serine/threonine-protein kinase pim-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,647
- Clinical molecules 25
- Avg pChEMBL 8.21
KEGG Pathways (5)
Active Molecules (2,647)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LBMWUDHQCZLSHO
|
8.1 | IC50 | 2 | — | |
LGCIOVKFCKDKRB
|
8.1 | Ki | 2 | — | |
MZUPUZSATAUNBG
|
8.1 | IC50 | 2 | — | |
NLOZLPYLNHZXJD
|
8.1 | IC50 | 3 | — | |
NSYYGKLWUGNCHP
|
8.1 | IC50 | 4 | — | |
RZEHXAGBPVZUII
|
8.1 | IC50 | 2 | — | |
WTGCKCDNZFLRCX
|
8.1 | IC50 | 2 | — | |
XHQCKTYOEPETON
|
8.1 | IC50 | 3 | — | |
XSOGQUXEVBPTQF
|
8.1 | IC50 | 4 | — | |
XXSRLUNTWYTWGT
|
8.1 | IC50 | 2 | — | |
YLYOPFUNIKCBEG
|
8.1 | IC50 | 3 | — | |
GWBUKZMEQCEWRK
|
8.0 | IC50 | 2 | — | |
HTMBVCFZCSVVSW
|
8.0 | IC50 | 3 | — | |
WUTCYYSJWLOLPF
|
8.0 | IC50 | 3 | — | |
YJOIGTLSOAMPHW
|
8.0 | IC50 | 3 | — | |
BSFGKWICIAYJPQ
|
8.0 | IC50 | 2 | — | |
DHICUKZZXJZLPW
|
8.0 | IC50 | 2 | — | |
GWRLSNACWTZFNG
|
8.0 | IC50 | 3 | — | |
QTIQZQUAJDJRAA
|
8.0 | IC50 | 2 | — | |
SAMUUOQCTGFAPT
|
8.0 | IC50 | 3 | — | |
XJLLCFIQDIZPNO
|
8.0 | IC50 | 2 | — | |
DHZAZLLWSFQYML
|
8.0 | IC50 | 3 | — | |
HIOLHQVNMHVRKB
|
8.0 | IC50 | 2 | — | |
JOOLQZAACBCCFW
|
8.0 | IC50 | 2 | — | |
OQULQTMKDZGXOL
|
8.0 | Ki | 3 | — | |
QWIPSLMHCCVXCL
|
8.0 | IC50 | 2 | — | |
AYZUBCLOFTTWJJ
|
8.0 | IC50 | 3 | — | |
DCHLKSOMTRDQCG
|
8.0 | IC50 | 4 | — | |
FRTFBLDBKLPEEG
|
8.0 | IC50 | 2 | — | |
FRVOCFJDZQHLPC
|
8.0 | IC50 | 3 | — | |
FZKGUWWNNSQWJG
|
8.0 | IC50 | 2 | — | |
GHPFQRTVUDXWCC
|
8.0 | Ki | 35 | — | |
HKSZLNNOFSGOKW
|
8.0 | IC50 | 408 | — | |
HKSZLNNOFSGOKW
|
8.0 | IC50 | 49 | Yes | |
HPHKSCVZUSQYGD
|
8.0 | IC50 | 5 | — | |
IUFOLPOPTPIBRL
|
8.0 | IC50 | 2 | — | |
MESLRIMNHFRXEO
|
8.0 | IC50 | 2 | — | |
PYWZTKODXYPZLR
|
8.0 | IC50 | 3 | — | |
UHYACKXUWYSKIU
|
8.0 | IC50 | 2 | — | |
UQQRRLPBVIAHKF
|
8.0 | IC50 | 5 | — | |
UXEVZFRUXSMUKW
|
8.0 | IC50 | 2 | — | |
YPGUAMCIYVJFOJ
|
8.0 | IC50 | 3 | — | |
YSWMGTNULRMHFF
|
8.0 | IC50 | 2 | — | |
FZTSRAGTHKAPKA
|
8.0 | Ki | 3 | — | |
GFNSSGCOEONQCH
|
8.0 | IC50 | 2 | — | |
LRHALWOPMLQBBG
|
8.0 | IC50 | 2 | — | |
LLQIYQUPTCRRAL
|
8.0 | Ki | 3 | — | |
NLOZLPYLNHZXJD
|
8.0 | IC50 | 3 | — | |
DAGZBPRGFBEYDJ
|
8.0 | IC50 | 3 | — | |
HCTNDZZYSZKDDR
|
8.0 | IC50 | 3 | — |