Target Details
| UniProt AC | P11309 |
|---|---|
| Gene Symbol | PIM1 |
| Protein Name | Serine/threonine-protein kinase pim-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,647
- Clinical molecules 25
- Avg pChEMBL 8.21
KEGG Pathways (5)
Active Molecules (2,647)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FBEUTZRQCSCWQM
|
8.1 | IC50 | 2 | — | |
FDKSNPXUVSQPQD
|
8.1 | IC50 | 2 | — | |
FOPGQICEKPAAOV
|
8.1 | IC50 | 2 | — | |
FRRLLRQAGKSVMU
|
8.1 | IC50 | 7 | — | |
GAXARIICIJOJOY
|
8.1 | IC50 | 3 | — | |
GQQFTUPPVDKXOP
|
8.1 | IC50 | 2 | — | |
HCDKRSHCTHPMMG
|
8.1 | IC50 | 3 | — | |
HGRGBTOFFWBXHE
|
8.1 | Ki | 3 | — | |
HMSVYVJNUGHJAR
|
8.1 | IC50 | 2 | — | |
HUUCRJKCBZDCKY
|
8.1 | IC50 | 4 | — | |
KTRXAKKECRZQCO
|
8.1 | IC50 | 2 | — | |
KXDUVJWVGXIEPX
|
8.1 | IC50 | 2 | — | |
LIFFFTHJTYXQFZ
|
8.1 | IC50 | 2 | — | |
OFVISGBWWVXCGV
|
8.1 | Ki | 2 | — | |
PCRTYXJARRBTQP
|
8.1 | Ki | 2 | — | |
QPDFWFQRIFSVFV
|
8.1 | IC50 | 2 | — | |
RDBQZAOHLXXDCN
|
8.1 | IC50 | 3 | — | |
UENAANOOJPBPBW
|
8.1 | IC50 | 3 | — | |
URLSXEUWUQRQEM
|
8.1 | IC50 | 5 | — | |
WLPJPVKABBJIAP
|
8.1 | IC50 | 3 | — | |
YJNHMIYBHYMVLJ
|
8.1 | Ki | 2 | — | |
YJVVLQUVYXOXOT
|
8.1 | IC50 | 2 | — | |
YSUUUMYLQMWZMR
|
8.1 | IC50 | 2 | — | |
YWTBGJGMTBHQTM
|
8.1 | Ki | 65 | — | |
BJWZYPUXMABVIE
|
8.1 | IC50 | 3 | — | |
FAUDAQJUMHDILO
|
8.1 | IC50 | 2 | — | |
KDYCRHVPKRGNNL
|
8.1 | IC50 | 2 | — | |
MHDPLRBCBJTFPZ
|
8.1 | IC50 | 2 | — | |
LDOPSNXYWCQDJY
|
8.1 | IC50 | 2 | — | |
REOXYDROSGGGDW
|
8.1 | IC50 | 2 | — | |
MBDXCSSBRAZUJO
|
8.1 | Ki | 2 | — | |
OLIOBBIZJBFLQG
|
8.1 | IC50 | 3 | — | |
WQLUNJCVHZPXEC
|
8.1 | IC50 | 2 | — | |
CTUHVBQMEHYEQH
|
8.1 | IC50 | 2 | — | |
PNQLIJJPVOBSQU
|
8.1 | IC50 | 4 | — | |
QERPWVWLRMKUFA
|
8.1 | IC50 | 2 | — | |
XTWLLGKUEJXNPC
|
8.1 | IC50 | 3 | — | |
YUOMNHIIJUOCOA
|
8.1 | IC50 | 2 | — | |
BLPVXPWSPTYNPS
|
8.1 | IC50 | 4 | — | |
CLDXOKMGNYBJKR
|
8.1 | IC50 | 2 | — | |
DGLXOJMLPNCUDE
|
8.1 | IC50 | 7 | Yes | |
DSUSQUXNJRQJMI
|
8.1 | Ki | 2 | — | |
GIHUWFBQWLLTIZ
|
8.1 | IC50 | 4 | — | |
HEZINGLKAUOZKD
|
8.1 | IC50 | 3 | — | |
HNPPTJBBFAGSJD
|
8.1 | IC50 | 3 | — | |
HXRPIJWBXRRJAP
|
8.1 | IC50 | 4 | — | |
IMFKOPJGEHGUDY
|
8.1 | IC50 | 3 | — | |
JGKMXEWZXLSBRF
|
8.1 | IC50 | 2 | — | |
JYUCZTGADIKZPX
|
8.1 | IC50 | 3 | — | |
KZLQFLHBCDGIBH
|
8.1 | IC50 | 5 | — |