Target Details
| UniProt AC | P11309 |
|---|---|
| Gene Symbol | PIM1 |
| Protein Name | Serine/threonine-protein kinase pim-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,647
- Clinical molecules 25
- Avg pChEMBL 8.21
KEGG Pathways (5)
Active Molecules (2,647)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DGAUZJLZJIGTFD
|
8.2 | IC50 | 2 | — | |
DOBBSPBMIKHNBX
|
8.2 | IC50 | 2 | — | |
FDOTVWCTNRPFBV
|
8.2 | IC50 | 3 | — | |
GKKURUBIEFRHRD
|
8.2 | IC50 | 3 | — | |
JFVYPLNMSLRVGZ
|
8.2 | IC50 | 3 | — | |
JSHFOHFQKWDTOB
|
8.2 | IC50 | 2 | — | |
KXRZQMBZXHBNTQ
|
8.2 | IC50 | 2 | — | |
LRZCLGRWOPGGBZ
|
8.2 | IC50 | 3 | — | |
MHXGEROHKGDZGO
|
8.2 | IC50 | 10 | — | |
OZZCHQRAYPMEEI
|
8.2 | IC50 | 2 | — | |
PKMITZKQGGMYHI
|
8.2 | IC50 | 4 | — | |
PSIMDRXAPBUVNE
|
8.2 | IC50 | 2 | — | |
QFEQLOZOUCTCFE
|
8.2 | IC50 | 3 | — | |
RLPRIAUIJLQFJH
|
8.2 | IC50 | 2 | — | |
WTGCKCDNZFLRCX
|
8.2 | IC50 | 2 | — | |
YCYQZQOOPFPJAO
|
8.2 | IC50 | 4 | — | |
YZAAXAWPNUWNKE
|
8.2 | IC50 | 2 | — | |
ZBDQLRFROCVCJP
|
8.2 | IC50 | 2 | — | |
ZOUDTZOMWZWKMO
|
8.2 | IC50 | 2 | — | |
ZVTHEZOGZZBRHH
|
8.2 | IC50 | 2 | — | |
ZWVHBACWMIHSNL
|
8.2 | IC50 | 2 | — | |
CAPRZSXGUIQKOH
|
8.1 | IC50 | 2 | — | |
JCHKNLLUGJTBFB
|
8.1 | IC50 | 2 | — | |
MPFTYTXJRHGYBP
|
8.1 | IC50 | 3 | — | |
OIHRVTLGUCLTFU
|
8.1 | IC50 | 2 | — | |
QUUBUYOWQZWVPC
|
8.1 | IC50 | 2 | — | |
SFMKWUZETRDDOW
|
8.1 | IC50 | 2 | — | |
SYPBNOXLIVCNCJ
|
8.1 | Ki | 3 | — | |
WSLDIDFQCRYHIJ
|
8.1 | IC50 | 2 | — | |
LPHDIQKURFDTPO
|
8.1 | IC50 | 2 | — | |
UPWSLCGFUGKUCL
|
8.1 | IC50 | 2 | — | |
AEWPQHXJYCZCLN
|
8.1 | IC50 | 2 | — | |
AVRMTBJBDHXUGZ
|
8.1 | IC50 | 2 | — | |
MLPJIYXHHVPOPK
|
8.1 | IC50 | 2 | — | |
NHZYQENPPFGWPW
|
8.1 | IC50 | 2 | — | |
NMOAVWCJECIOPM
|
8.1 | IC50 | 2 | — | |
NQJCNHBXICRIPG
|
8.1 | IC50 | 2 | — | |
UWKVKWLSOMBHTE
|
8.1 | Ki | 3 | — | |
YAJGELPVDBECTQ
|
8.1 | IC50 | 2 | — | |
FLPSOVPOQWHOJV
|
8.1 | IC50 | 3 | — | |
JKWRFEXKHMHWOO
|
8.1 | IC50 | 2 | — | |
KLIFVHOZCRYWKQ
|
8.1 | IC50 | 2 | — | |
MILQRCUVJFKCQR
|
8.1 | Ki | 3 | — | |
OTWLCRXTCIMBPE
|
8.1 | IC50 | 2 | — | |
QCKWETFAVPLIJH
|
8.1 | IC50 | 3 | — | |
AHTFFUBCDIKLDM
|
8.1 | IC50 | 3 | — | |
BAAFIGWSBYBAEO
|
8.1 | IC50 | 2 | — | |
BXKIPOGUQCAVMR
|
8.1 | IC50 | 3 | — | |
CPFUAFFNZAQNIL
|
8.1 | IC50 | 4 | — | |
DSXXEELGXBCYNQ
|
8.1 | Kd | 28 | Yes |