Target Details
| UniProt AC | P11309 |
|---|---|
| Gene Symbol | PIM1 |
| Protein Name | Serine/threonine-protein kinase pim-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,647
- Clinical molecules 25
- Avg pChEMBL 8.21
KEGG Pathways (5)
Active Molecules (2,647)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OZAALIWIRMBCOR
|
8.2 | IC50 | 4 | — | |
PAVPZPCSAGSHHJ
|
8.2 | IC50 | 3 | — | |
PAWYDNPYJNAJHA
|
8.2 | IC50 | 3 | — | |
POZXOXRCXCUUSS
|
8.2 | IC50 | 3 | — | |
QISQRPRJLVQNKR
|
8.2 | IC50 | 4 | — | |
QNIVGJHTGPNPHG
|
8.2 | Ki | 2 | — | |
RJYKOWGBWXBBBA
|
8.2 | IC50 | 3 | — | |
UOOCRVJWAMBPLA
|
8.2 | IC50 | 2 | — | |
WCLBXMSWYPPACJ
|
8.2 | IC50 | 3 | — | |
WKKLGYBBGSOPSP
|
8.2 | IC50 | 2 | — | |
WNTHOTLXPLDFPC
|
8.2 | IC50 | 5 | — | |
XSIPCMUZGAGULD
|
8.2 | IC50 | 2 | — | |
YEGXHTKFBQFSNF
|
8.2 | IC50 | 3 | — | |
YNSGZPAZNHHVQL
|
8.2 | IC50 | 3 | — | |
ZQSFRZOCLWDZFX
|
8.2 | IC50 | 2 | — | |
AWUYXCAHTLGAMI
|
8.2 | IC50 | 2 | — | |
LRVOQVWUCGGLLL
|
8.2 | IC50 | 2 | — | |
UHRDRFKXJSSJHA
|
8.2 | IC50 | 2 | — | |
VPLXMHRCNSVLNX
|
8.2 | IC50 | 2 | — | |
CHTMRWQLNNRRFJ
|
8.2 | Ki | 70 | — | |
HMEPBBABMLMGIG
|
8.2 | IC50 | 2 | — | |
LSVPGWJBHBUSHL
|
8.2 | IC50 | 2 | — | |
RCZYLHFODBPYHX
|
8.2 | IC50 | 3 | — | |
VGHNUVDMAHSAAD
|
8.2 | IC50 | 2 | — | |
YXZSPNLYIYHRNS
|
8.2 | IC50 | 3 | — | |
CPZFYPWVXHFNAZ
|
8.2 | IC50 | 2 | — | |
FLUCKTIWFMWKNJ
|
8.2 | IC50 | 3 | — | |
FXKAJMTVSSOIMV
|
8.2 | IC50 | 2 | — | |
GVQAIMRPJCUOER
|
8.2 | IC50 | 2 | — | |
NVTPYRCDKQXUGU
|
8.2 | Ki | 3 | — | |
UIPGRKAAMDJZHQ
|
8.2 | IC50 | 2 | — | |
WSBXTXMVHFPAPA
|
8.2 | IC50 | 3 | — | |
DAGZBPRGFBEYDJ
|
8.2 | IC50 | 2 | — | |
DFKOCMIZZATJNQ
|
8.2 | IC50 | 2 | — | |
IYKWFKKDLTZONH
|
8.2 | IC50 | 3 | — | |
JCHKNLLUGJTBFB
|
8.2 | IC50 | 2 | — | |
KKVGPCFFNMHJHC
|
8.2 | IC50 | 3 | — | |
KPBPFEDQSSJBIT
|
8.2 | IC50 | 2 | — | |
NSUAVZRKGRVKNI
|
8.2 | IC50 | 2 | — | |
AVWIQATUPWLNJO
|
8.2 | IC50 | 3 | — | |
DTJDHZDARQGLCW
|
8.2 | IC50 | 4 | — | |
ODNOXJRRJVQZJF
|
8.2 | IC50 | 2 | — | |
PAWVEZOTRVPHRU
|
8.2 | IC50 | 2 | — | |
UYWOVNUCOZQXAD
|
8.2 | IC50 | 3 | — | |
YHICBQSUKWMZMG
|
8.2 | IC50 | 2 | — | |
BCPIVSDHNQBACL
|
8.2 | IC50 | 3 | — | |
BGKFEQIYJGJHTL
|
8.2 | IC50 | 2 | — | |
BKDLGAKRAHVMNP
|
8.2 | IC50 | 2 | — | |
BVXJGQKYALRJIJ
|
8.2 | IC50 | 3 | — | |
DECHCVMZNFKMLE
|
8.2 | IC50 | 3 | — |