Target Details
| UniProt AC | P11309 |
|---|---|
| Gene Symbol | PIM1 |
| Protein Name | Serine/threonine-protein kinase pim-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,647
- Clinical molecules 25
- Avg pChEMBL 8.21
KEGG Pathways (5)
Active Molecules (2,647)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WNOHFJIMKSDPHP
|
8.3 | IC50 | 4 | — | |
WPMKCHOCXWTADK
|
8.3 | IC50 | 2 | — | |
YLJCMWKIAARCQT
|
8.3 | Ki | 2 | — | |
YQHNAPALHYCHHP
|
8.3 | Ki | 2 | — | |
KXHNUSUTHSYUGC
|
8.3 | IC50 | 2 | — | |
OXNIZFDZFYTTAF
|
8.3 | IC50 | 3 | — | |
RMWWTXNOTVLFAD
|
8.3 | IC50 | 2 | — | |
SMWFSPOWWDSJEB
|
8.3 | IC50 | 3 | — | |
AFGSEIPIIRAHRL
|
8.3 | IC50 | 2 | — | |
CNMCULKLLKXKPE
|
8.3 | IC50 | 2 | — | |
IDGZWDPYDQBXHU
|
8.3 | IC50 | 2 | — | |
ILKOWNVFKVGQKA
|
8.3 | IC50 | 2 | — | |
CVTRYARXXBAMAJ
|
8.3 | IC50 | 2 | — | |
FSXGCPFKFZBVFO
|
8.3 | IC50 | 3 | — | |
KRBNQISTMITIOJ
|
8.3 | IC50 | 2 | — | |
VKGQNHBAFASGIN
|
8.3 | IC50 | 2 | — | |
YXBOQTUJWONSJX
|
8.3 | IC50 | 3 | — | |
AWPOFKRPERMOIK
|
8.2 | IC50 | 3 | — | |
DJYGBVVTIRVFKI
|
8.2 | Ki | 3 | — | |
HUQIGUWVDJPJBU
|
8.2 | IC50 | 2 | — | |
JHCXRIDGVGVKMB
|
8.2 | IC50 | 3 | — | |
VXKHZVAIDVDYAH
|
8.2 | Ki | 3 | — | |
XKTURFXRMNBNAV
|
8.2 | Ki | 3 | — | |
FAZMPKDPEUFZHA
|
8.2 | IC50 | 3 | — | |
GOURHBOOQWGQNN
|
8.2 | Ki | 3 | — | |
JVRVCXNNVPBKQF
|
8.2 | IC50 | 2 | — | |
KOEBLNVZIKWEAL
|
8.2 | IC50 | 2 | — | |
POHFVNMGAPNFAB
|
8.2 | IC50 | 2 | — | |
ROJNKYJPUZLUTF
|
8.2 | IC50 | 2 | — | |
UDHXHJAZPMOTOA
|
8.2 | IC50 | 3 | — | |
UKOFGJPVBBRSGO
|
8.2 | IC50 | 2 | — | |
WNIIXCCZBNUGMW
|
8.2 | IC50 | 3 | — | |
BNJGTWDHTFBYQR
|
8.2 | IC50 | 3 | — | |
KYVNDWJWKGXGDI
|
8.2 | IC50 | 2 | — | |
TZQSDHCSGGGNSR
|
8.2 | IC50 | 3 | — | |
UXBAIRNMPUPDFK
|
8.2 | IC50 | 2 | — | |
YUZSKZGDSMZEFD
|
8.2 | IC50 | 3 | — | |
YYOMMRYHXLZQAT
|
8.2 | IC50 | 2 | — | |
ZIUGHJPWIKKQNX
|
8.2 | IC50 | 2 | — | |
AQLVNFYJDCDILG
|
8.2 | IC50 | 2 | — | |
BIKSJBQYLXGSCK
|
8.2 | IC50 | 2 | — | |
CYOIVDLXCFCOCJ
|
8.2 | IC50 | 4 | — | |
DADGQFMQIHDYTQ
|
8.2 | IC50 | 2 | — | |
DRMHBTZKBJCWJJ
|
8.2 | Ki | 3 | — | |
FOMQAXLFFZQXNC
|
8.2 | IC50 | 2 | — | |
GTHLJKKDZJPZLZ
|
8.2 | IC50 | 3 | — | |
HNIDDGUBRPIXPG
|
8.2 | IC50 | 7 | — | |
IRUULFBKQJRPEH
|
8.2 | IC50 | 2 | — | |
MHHJJHVQXDCGDG
|
8.2 | IC50 | 3 | — | |
MSUFNCHTJLZAPS
|
8.2 | IC50 | 2 | — |