Target Details
| UniProt AC | P11309 |
|---|---|
| Gene Symbol | PIM1 |
| Protein Name | Serine/threonine-protein kinase pim-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,647
- Clinical molecules 25
- Avg pChEMBL 8.21
KEGG Pathways (5)
Active Molecules (2,647)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UJBRJYXRVHBJQM
|
8.3 | IC50 | 2 | — | |
VDFWYILSYHAMNU
|
8.3 | IC50 | 2 | — | |
WFKZLRQOFSFNJO
|
8.3 | IC50 | 4 | — | |
DSFJTSSJSJDOGO
|
8.3 | IC50 | 2 | — | |
GPLPYBDISWCAQW
|
8.3 | IC50 | 2 | — | |
KTWRUVPDMFAYQD
|
8.3 | IC50 | 3 | — | |
PMUBHUYTMZZLML
|
8.3 | IC50 | 3 | — | |
QVHWRVHLJFUJKP
|
8.3 | Ki | 3 | — | |
ALFMWZJOROWWPA
|
8.3 | IC50 | 2 | — | |
FISCYPDTCXZXLZ
|
8.3 | IC50 | 2 | — | |
RAGDOJKYCQWMLT
|
8.3 | IC50 | 2 | — | |
SKDNYSOXNQDPRX
|
8.3 | IC50 | 2 | — | |
VUSIBGXJGOLGIN
|
8.3 | IC50 | 2 | — | |
FMCHSBJRGSMUTQ
|
8.3 | IC50 | 2 | — | |
ANPJHKVBDUXPEB
|
8.3 | IC50 | 2 | — | |
JIPAVNODPHBEFL
|
8.3 | IC50 | 2 | — | |
XPMXMSKJKVFHSA
|
8.3 | IC50 | 2 | — | |
YUDHKJJAUQNWBR
|
8.3 | IC50 | 2 | — | |
AKRXLINEJRYTHQ
|
8.3 | IC50 | 3 | — | |
ANSIRGLMUHWNPB
|
8.3 | IC50 | 3 | — | |
BGYKECRMNHZETP
|
8.3 | IC50 | 3 | — | |
BRAYMNJVFKIQLD
|
8.3 | IC50 | 2 | — | |
CWRBSZWGCCMVST
|
8.3 | IC50 | 2 | — | |
DIMWPKIMCQOTSC
|
8.3 | Ki | 3 | — | |
DNXZIJKGPFJRAA
|
8.3 | IC50 | 3 | — | |
DOERTQQDUFOAOA
|
8.3 | IC50 | 2 | — | |
DSUSEZJHVSEHGF
|
8.3 | IC50 | 2 | — | |
DSUSQUXNJRQJMI
|
8.3 | Ki | 2 | — | |
GNXBPOKOBOXVEM
|
8.3 | IC50 | 3 | — | |
GOFOMUKPTQCOQX
|
8.3 | Ki | 3 | — | |
IFKCLLHUGZYAPV
|
8.3 | IC50 | 4 | — | |
IRPPYJZDFMMBBV
|
8.3 | IC50 | 3 | — | |
IVDRVWFOHOJDBW
|
8.3 | IC50 | 3 | — | |
IXPYOFCXANNZML
|
8.3 | IC50 | 4 | — | |
JSOJYCSDBKJYSB
|
8.3 | Ki | 3 | — | |
JXGOFCNAXBWAJO
|
8.3 | IC50 | 4 | — | |
JZJFOEZBTQXBKQ
|
8.3 | Ki | 2 | — | |
KGBPLKOPSFDBOX
|
8.3 | IC50 | 4 | — | |
LIVUQZJIYLMRNO
|
8.3 | IC50 | 2 | — | |
NFMGQYVXXDIVFX
|
8.3 | IC50 | 2 | — | |
NJPWCTYVEJIQBM
|
8.3 | Ki | 72 | — | |
NNXJGFIMOCXDNA
|
8.3 | Ki | 2 | — | |
OPXDNPAGMKMBTA
|
8.3 | IC50 | 2 | — | |
PZACVAVZCMGALO
|
8.3 | Ki | 3 | — | |
QBBDBUVPJDYPLQ
|
8.3 | IC50 | 4 | — | |
QRVJKXOAMVIRHV
|
8.3 | IC50 | 2 | — | |
QUKALHWYSNHRNQ
|
8.3 | IC50 | 2 | — | |
RWRRKKBGTAZXGP
|
8.3 | IC50 | 3 | — | |
VJZFGXCKDFGGEU
|
8.3 | Ki | 2 | — | |
VXYDJXMHISGSDA
|
8.3 | Ki | 59 | — |