Target Details
| UniProt AC | P11309 |
|---|---|
| Gene Symbol | PIM1 |
| Protein Name | Serine/threonine-protein kinase pim-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,647
- Clinical molecules 25
- Avg pChEMBL 8.21
KEGG Pathways (5)
Active Molecules (2,647)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MACWFODIYDAOMY
|
8.4 | Ki | 2 | — | |
MGOSXKXPLHPFEB
|
8.4 | IC50 | 3 | — | |
MOYQBNCJLIJEOA
|
8.4 | IC50 | 3 | — | |
NOJHQUZCNBPNPS
|
8.4 | IC50 | 2 | — | |
NZRCHCMMQGWKLZ
|
8.4 | IC50 | 3 | — | |
ODOJDGPBPYYKKL
|
8.4 | Ki | 2 | — | |
ODZZYKUYGVLOTQ
|
8.4 | IC50 | 3 | — | |
OUPLDKOZBSMDAA
|
8.4 | IC50 | 2 | — | |
PBLFJZCOGVJGGN
|
8.4 | IC50 | 2 | — | |
PQACSMVQKDXJMY
|
8.4 | IC50 | 2 | — | |
PSFMCOGQKUBLKM
|
8.4 | IC50 | 3 | — | |
PUUIFRIHCXPFEM
|
8.4 | IC50 | 4 | — | |
PZOMINBBFNQNAN
|
8.4 | IC50 | 2 | — | |
QKRLKEOSBXNMGP
|
8.4 | Ki | 3 | — | |
QUQCDJVOANWCBN
|
8.4 | IC50 | 4 | — | |
RHIDXFBMAIUIMQ
|
8.4 | IC50 | 2 | — | |
RUJLVOBTFPKXGV
|
8.4 | IC50 | 2 | — | |
RVDVNYIESZTRRB
|
8.4 | IC50 | 2 | — | |
SOUGKZTUMVEVDD
|
8.4 | IC50 | 2 | — | |
SVDDKCFDTZXPLV
|
8.4 | IC50 | 3 | — | |
UJCZXEMKGRZREN
|
8.4 | IC50 | 5 | — | |
URCZAWFHBYABKR
|
8.4 | IC50 | 2 | — | |
UXKHBSKXYJUFJH
|
8.4 | Ki | 3 | — | |
WFKSOSWVYIZSKO
|
8.4 | IC50 | 2 | — | |
WQTAETIAWLTMKZ
|
8.4 | Ki | 2 | — | |
WSTRRKGONYVANU
|
8.4 | IC50 | 3 | — | |
WVOATLASLUXFNF
|
8.4 | IC50 | 2 | — | |
ZXQIHLJIAWEHOF
|
8.4 | IC50 | 2 | — | |
APMKLXLBNBDHBU
|
8.4 | IC50 | 2 | — | |
OGTWUWZXWAVZHO
|
8.4 | IC50 | 2 | — | |
OXJMFQVRMWSKKM
|
8.4 | IC50 | 2 | — | |
RJQJFTUVYNAFRC
|
8.4 | IC50 | 2 | — | |
JTESMRSKGHICMR
|
8.4 | IC50 | 3 | — | |
KOQXLXUOIGXSIW
|
8.4 | IC50 | 2 | — | |
SMFLEXPDEWVLCB
|
8.4 | IC50 | 2 | — | |
VLWWSFAMFACJRL
|
8.4 | IC50 | 2 | — | |
YNYGYKNLVMLFSO
|
8.4 | IC50 | 3 | — | |
YTBQJCHZAHBGOV
|
8.4 | IC50 | 3 | — | |
GHYCXGADCHFASP
|
8.4 | IC50 | 2 | — | |
MDZQPPYWTULKAT
|
8.4 | IC50 | 2 | — | |
SDWLMNIERCYSEQ
|
8.4 | IC50 | 2 | — | |
GAFQWVCMOUDTGJ
|
8.4 | Ki | 3 | — | |
INYRWBVCPQQSGE
|
8.4 | IC50 | 2 | — | |
JBUOFUIXSMJURC
|
8.4 | IC50 | 3 | — | |
MVCMGBIAYBTDLE
|
8.4 | Ki | 3 | — | |
PVPKHHBPGARBMQ
|
8.4 | IC50 | 2 | — | |
DRSGTFRMJJUHTO
|
8.3 | IC50 | 2 | — | |
FRGSBCXYFDKJNS
|
8.3 | IC50 | 2 | — | |
NOVOUDRJIQLPML
|
8.3 | IC50 | 3 | — | |
RWNZWAMJEWYARJ
|
8.3 | IC50 | 2 | — |