Target Details
| UniProt AC | P11309 |
|---|---|
| Gene Symbol | PIM1 |
| Protein Name | Serine/threonine-protein kinase pim-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,647
- Clinical molecules 25
- Avg pChEMBL 8.21
KEGG Pathways (5)
Active Molecules (2,647)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SEWSVZNGUQAMFX
|
8.5 | Ki | 3 | — | |
FINRCSOWWRQIKA
|
8.4 | IC50 | 2 | — | |
WYCYQOYGEREIMC
|
8.4 | Ki | 3 | — | |
YHEKLPCGOWOJKE
|
8.4 | IC50 | 2 | — | |
CMCGBWKSQYENCR
|
8.4 | IC50 | 2 | — | |
FSUPHBZWCKRZOA
|
8.4 | IC50 | 2 | — | |
XRZKMAHDTNYENT
|
8.4 | IC50 | 2 | — | |
YKRWZGXTOYQHJI
|
8.4 | IC50 | 3 | — | |
BTAOJMVOLXGTQG
|
8.4 | IC50 | 2 | — | |
MDXOTNRTTAMQJG
|
8.4 | IC50 | 2 | — | |
QCWLXJUMRLWMRQ
|
8.4 | IC50 | 2 | — | |
SSUVSBRBZXJBQT
|
8.4 | Ki | 3 | — | |
UOMPPOVQMYNXST
|
8.4 | IC50 | 2 | — | |
CPBODKOJHSDKCU
|
8.4 | IC50 | 2 | — | |
HSKRSIYBQAHFCE
|
8.4 | Ki | 3 | — | |
NXDFPMRJOPOBGD
|
8.4 | IC50 | 2 | — | |
PPKOMRSAECKGDB
|
8.4 | IC50 | 2 | — | |
SMXUSZSYBNSJDM
|
8.4 | IC50 | 3 | — | |
FALXVTLWNUJCKA
|
8.4 | Ki | 3 | — | |
HNIDDGUBRPIXPG
|
8.4 | IC50 | 7 | — | |
RYSAKMOLNKFGCG
|
8.4 | IC50 | 2 | — | |
UZWDCWONPYILKI
|
8.4 | IC50 | 47 | — | |
ADQZWDPCIBFHEH
|
8.4 | IC50 | 3 | — | |
ANSIRGLMUHWNPB
|
8.4 | IC50 | 3 | — | |
AVHYIXDAOCBQIU
|
8.4 | IC50 | 2 | — | |
AZSRVVPUAZTMAY
|
8.4 | IC50 | 2 | — | |
BAJBJWWXJSZEDI
|
8.4 | IC50 | 2 | — | |
BFDYPWZGYIYZPW
|
8.4 | IC50 | 2 | — | |
CXZABFFSXIOBBA
|
8.4 | Ki | 2 | — | |
DAGZBPRGFBEYDJ
|
8.4 | IC50 | 2 | — | |
FCQKXMKELLUTAY
|
8.4 | IC50 | 4 | — | |
FVRMTRYCXIUJEB
|
8.4 | IC50 | 3 | — | |
FVRMTRYCXIUJEB
|
8.4 | IC50 | 3 | — | |
GBPGFWBSOAIUBT
|
8.4 | Ki | 3 | — | |
GDARJPADPPAMKE
|
8.4 | IC50 | 3 | — | |
GMLWQFRZINHDEH
|
8.4 | IC50 | 3 | — | |
GUNWLRDFSJIUEI
|
8.4 | IC50 | 4 | — | |
GZBBGJRQPGJEEE
|
8.4 | IC50 | 2 | — | |
HAJKKQIGRJNJJQ
|
8.4 | IC50 | 3 | — | |
HGARXRXLHSFNEX
|
8.4 | IC50 | 5 | — | |
HKOWJFORUXHTHX
|
8.4 | IC50 | 4 | — | |
HNODKCFEFLQKBO
|
8.4 | Ki | 6 | — | |
HPGYBULDKFXBFU
|
8.4 | IC50 | 3 | — | |
HSBXTJAEFSRBOW
|
8.4 | IC50 | 4 | — | |
ITEIREYZTCHMHP
|
8.4 | Ki | 3 | — | |
JIORTDOUIQMVEG
|
8.4 | IC50 | 2 | — | |
KOARITDFMAWYET
|
8.4 | IC50 | 3 | — | |
KSFKMCQSTBWUED
|
8.4 | Ki | 3 | — | |
LIVUQZJIYLMRNO
|
8.4 | IC50 | 2 | — | |
LRPIEIXQEJCTBD
|
8.4 | IC50 | 3 | — |