Target Details
| UniProt AC | P11309 |
|---|---|
| Gene Symbol | PIM1 |
| Protein Name | Serine/threonine-protein kinase pim-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,647
- Clinical molecules 25
- Avg pChEMBL 8.21
KEGG Pathways (5)
Active Molecules (2,647)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PQLFXCXWQSZFCU
|
8.5 | IC50 | 3 | — | |
QECUEJIBDRRTOL
|
8.5 | IC50 | 3 | — | |
QGIFMDZYUIQIRA
|
8.5 | IC50 | 5 | — | |
QVLFSPWFBBQTFA
|
8.5 | IC50 | 3 | — | |
QWCBDDMORRCKOO
|
8.5 | IC50 | 2 | — | |
QYEZWOQHLCHEFN
|
8.5 | Ki | 3 | — | |
RVEDMOLIJBWGQX
|
8.5 | Ki | 3 | — | |
SCIQGAHHNPDKAJ
|
8.5 | Ki | 2 | — | |
STWDLMHONRHMTF
|
8.5 | IC50 | 3 | — | |
SYPBNOXLIVCNCJ
|
8.5 | Ki | 3 | — | |
TUKQVKODBBLMSY
|
8.5 | IC50 | 2 | — | |
UGCCFJQVUHNGIM
|
8.5 | IC50 | 2 | — | |
UPYHXTVTHXTKNF
|
8.5 | IC50 | 3 | — | |
USAPQYPKDFTEMB
|
8.5 | IC50 | 2 | — | |
UUIYNZNVNQVZOT
|
8.5 | IC50 | 5 | — | |
VCGNDPLDVLHZGK
|
8.5 | IC50 | 2 | — | |
VQNRDEXAKNAZTQ
|
8.5 | IC50 | 4 | — | |
ZGMKDXQXTMYRAS
|
8.5 | IC50 | 3 | — | |
ZPIVTGDIMHFXKE
|
8.5 | IC50 | 3 | — | |
ZWERZKRFVLXPIK
|
8.5 | IC50 | 3 | — | |
ZXQIHLJIAWEHOF
|
8.5 | IC50 | 2 | — | |
CHPLSEJPLSDICK
|
8.5 | IC50 | 3 | — | |
ITQFRPBHRRDOKY
|
8.5 | IC50 | 3 | — | |
JTAMJXTXUVCVAP
|
8.5 | IC50 | 2 | — | |
JXTNSWUVLITLAJ
|
8.5 | IC50 | 2 | — | |
NQGMOQOKDFPUAO
|
8.5 | IC50 | 2 | — | |
OSOUOUSXPWWDON
|
8.5 | IC50 | 2 | — | |
RRSYIVJLGUPYPY
|
8.5 | IC50 | 2 | — | |
UTNCOKVXILEJCJ
|
8.5 | IC50 | 2 | — | |
WUWGDDJIQSVRRK
|
8.5 | IC50 | 2 | — | |
YYXJSPFGMAXZGZ
|
8.5 | IC50 | 2 | — | |
ILVKLFOUGPBUMK
|
8.5 | IC50 | 3 | — | |
RRCCIDQPUXDUMY
|
8.5 | IC50 | 4 | — | |
HKSZLNNOFSGOKW
|
8.5 | Kd | 213 | — | |
XQPKIOMITKLVFI
|
8.5 | IC50 | 2 | — | |
YZAQSGMOAYQDAV
|
8.5 | IC50 | 3 | — | |
JCHKNLLUGJTBFB
|
8.5 | IC50 | 2 | — | |
JEIAIOKPHBZXMK
|
8.5 | IC50 | 2 | — | |
QIMHWUWINRBUSR
|
8.5 | Ki | 3 | — | |
SCMFHYFEMLZBFQ
|
8.5 | IC50 | 2 | — | |
VBXJPSXXVSLXSF
|
8.5 | IC50 | 2 | — | |
VMKWYFBQMNYWFN
|
8.5 | IC50 | 2 | — | |
FHAPDLVADXCIGY
|
8.5 | Ki | 3 | — | |
RRSYIVJLGUPYPY
|
8.5 | IC50 | 2 | — | |
SMYZVTZPMXEMEO
|
8.5 | IC50 | 2 | — | |
UEPZXHSQXVBLNH
|
8.5 | IC50 | 2 | — | |
XBUJJWKSFWVCRV
|
8.5 | IC50 | 3 | — | |
GHJCZGQHMLEEKQ
|
8.5 | IC50 | 3 | — | |
SAJBFQXKSKYUNF
|
8.5 | IC50 | 2 | — | |
SAWCQUAVBDKEJR
|
8.5 | IC50 | 2 | — |