Target Details
| UniProt AC | P11309 |
|---|---|
| Gene Symbol | PIM1 |
| Protein Name | Serine/threonine-protein kinase pim-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,647
- Clinical molecules 25
- Avg pChEMBL 8.21
KEGG Pathways (5)
Active Molecules (2,647)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GXLUWERWHDKAIH
|
8.6 | IC50 | 2 | — | |
LIWYTDUPDUJNJU
|
8.6 | IC50 | 2 | — | |
NYYSUURQWPBBLY
|
8.6 | IC50 | 2 | — | |
YAJGELPVDBECTQ
|
8.6 | IC50 | 3 | — | |
YYOMMRYHXLZQAT
|
8.6 | IC50 | 2 | — | |
DDQXBYGNFGPJRL
|
8.6 | IC50 | 3 | — | |
WEXPEOSYSQAIMZ
|
8.6 | IC50 | 2 | — | |
DTQJEAKNKGKTFD
|
8.6 | IC50 | 2 | — | |
FISXIELUYFZCMF
|
8.6 | IC50 | 2 | — | |
GYTXVBJMXPKSOG
|
8.6 | IC50 | 2 | — | |
UYOVRFLWHXLTBC
|
8.6 | IC50 | 3 | — | |
XUKBGDSNMIGPJV
|
8.6 | IC50 | 2 | — | |
YAJGELPVDBECTQ
|
8.6 | IC50 | 2 | — | |
YHUIWRYXTNQCAQ
|
8.6 | IC50 | 2 | — | |
DWJRVXUXEZICSB
|
8.5 | IC50 | 3 | — | |
GWILJQBMYLXBHZ
|
8.5 | Kd | 4 | — | |
LODPYXJMYAQIRB
|
8.5 | IC50 | 2 | — | |
UQNXDCLXUSCERQ
|
8.5 | IC50 | 2 | — | |
NUMGAHMZNWRORP
|
8.5 | Ki | 3 | — | |
SDHRADPEFDLIKD
|
8.5 | IC50 | 3 | — | |
SJVQOMGMHYJTEW
|
8.5 | IC50 | 2 | — | |
AQEZXJQHJXDUQL
|
8.5 | Ki | 3 | — | |
ATEORQMBWPIYQV
|
8.5 | IC50 | 3 | — | |
ATEORQMBWPIYQV
|
8.5 | IC50 | 3 | — | |
AXPHZYUNEZZRPW
|
8.5 | IC50 | 3 | — | |
AZSRVVPUAZTMAY
|
8.5 | IC50 | 2 | — | |
BKUXTVCORRDHGA
|
8.5 | IC50 | 3 | — | |
CDTJUEGCVWKCSA
|
8.5 | Ki | 3 | — | |
CPSNZCXBWOPDKW
|
8.5 | IC50 | 2 | — | |
CQOGWJPRIVQKRD
|
8.5 | IC50 | 2 | — | |
CUNYNKMLNKLFMN
|
8.5 | IC50 | 3 | — | |
FVGBFIJGKRDTEZ
|
8.5 | IC50 | 4 | — | |
GUTPGVLUDRSUIK
|
8.5 | IC50 | 2 | — | |
HFWFTPAPYFCKSG
|
8.5 | IC50 | 2 | — | |
HJJCPVZAEJNRGD
|
8.5 | IC50 | 3 | — | |
HJUNBWFLNSCJJH
|
8.5 | IC50 | 2 | — | |
HQWHAKOOAUIEHY
|
8.5 | IC50 | 3 | — | |
HWIDISMNBLRQNP
|
8.5 | IC50 | 3 | — | |
HZMQZYRYZGLOKJ
|
8.5 | IC50 | 3 | — | |
IMBMKCJXFZCZIB
|
8.5 | IC50 | 3 | — | |
INVWNQRXSPFOJI
|
8.5 | IC50 | 2 | — | |
JMHGWOVBMIFUIZ
|
8.5 | IC50 | 3 | — | |
JRBXRMRBIAPYOW
|
8.5 | IC50 | 3 | — | |
JXHFSTVXTDOYNC
|
8.5 | IC50 | 3 | — | |
KDDDVGDVYWKNOE
|
8.5 | IC50 | 2 | — | |
KEGTZWAXCSFQBQ
|
8.5 | Ki | 2 | — | |
KUFLSJFOFGKCHC
|
8.5 | IC50 | 3 | — | |
LLIAUBZSOICLJD
|
8.5 | IC50 | 2 | — | |
OMJQNHQCUDWRDZ
|
8.5 | IC50 | 2 | — | |
ORPOKTQAISYRIO
|
8.5 | IC50 | 5 | — |