Target Details
| UniProt AC | P11309 |
|---|---|
| Gene Symbol | PIM1 |
| Protein Name | Serine/threonine-protein kinase pim-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,647
- Clinical molecules 25
- Avg pChEMBL 8.21
KEGG Pathways (5)
Active Molecules (2,647)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GXDSAAYOXDQSQT
|
8.7 | Ki | 3 | — | |
HYYSIISVZBZUCM
|
8.7 | IC50 | 3 | — | |
VQGGQIGYLGHRNK
|
8.7 | IC50 | 3 | — | |
WIEJYJKDNYOPRH
|
8.7 | IC50 | 2 | — | |
WXBFQEMPNLLMNB
|
8.7 | Ki | 3 | — | |
BAOKFBOYECPWHF
|
8.7 | IC50 | 2 | — | |
BJSRODNZIHDLGO
|
8.7 | IC50 | 2 | — | |
LWXHKBKAMIELTQ
|
8.7 | IC50 | 2 | — | |
QVKCJELFCURCFY
|
8.7 | IC50 | 2 | — | |
WFTKWNBPRXJBBC
|
8.7 | IC50 | 2 | — | |
ZCZUSZGYIKHCLA
|
8.7 | IC50 | 2 | — | |
JEIAIOKPHBZXMK
|
8.7 | IC50 | 2 | — | |
OLFNLUGZKOQDEV
|
8.7 | IC50 | 9 | — | |
GDXMDKRKEIKPLW
|
8.6 | IC50 | 3 | — | |
JJMUWUXKLXIKLX
|
8.6 | IC50 | 2 | — | |
JMXDXNXSONBWNR
|
8.6 | IC50 | 2 | — | |
NFWRERNMTFKQTQ
|
8.6 | IC50 | 3 | — | |
PKGOHWVMPQTAGB
|
8.6 | IC50 | 2 | — | |
RJSJQDPTJIRVMZ
|
8.6 | IC50 | 2 | — | |
SYEYZQUZNVVCNN
|
8.6 | IC50 | 3 | — | |
BCAJPBKAVYTBSA
|
8.6 | IC50 | 2 | — | |
FUHMQPKEAAESFF
|
8.6 | IC50 | 2 | — | |
LYKLXICYCIJMAH
|
8.6 | IC50 | 2 | — | |
JFRTUZNKHJJSEH
|
8.6 | Ki | 3 | — | |
JRPMCVBHTMZOFM
|
8.6 | IC50 | 2 | — | |
OCLNGTQPTBNGKK
|
8.6 | IC50 | 2 | — | |
PVFFECNHTDFMJH
|
8.6 | IC50 | 3 | — | |
ISRJLVCSRJCNHO
|
8.6 | Ki | 3 | — | |
KDCYTTGIKIQSNT
|
8.6 | IC50 | 2 | — | |
QTQGVCAJBPUCSI
|
8.6 | IC50 | 2 | — | |
ANEQDQCTWAKZMN
|
8.6 | Ki | 3 | — | |
DRZARKMSKHYBNU
|
8.6 | IC50 | 2 | — | |
IVRNZICLBSEICC
|
8.6 | IC50 | 3 | — | |
JILYBMJSGXWKEA
|
8.6 | IC50 | 2 | — | |
MHDDMEQPCVULAB
|
8.6 | IC50 | 2 | — | |
PFJLWRBNOCAYMG
|
8.6 | IC50 | 2 | — | |
ROWCDUKNAFYOMJ
|
8.6 | IC50 | 3 | — | |
RRSYIVJLGUPYPY
|
8.6 | IC50 | 2 | — | |
UBPWEHJKADMOAV
|
8.6 | Ki | 2 | — | |
UKKVYNLBAIKQRV
|
8.6 | IC50 | 2 | — | |
WWECFSFDKPKNDT
|
8.6 | IC50 | 3 | — | |
XFXGUOSEGMYBDJ
|
8.6 | IC50 | 2 | — | |
HYYSIISVZBZUCM
|
8.6 | IC50 | 3 | — | |
LZPLMBTYKYAPPN
|
8.6 | IC50 | 2 | — | |
SKLNJZRVHSSOOX
|
8.6 | IC50 | 2 | — | |
IMRPDFHFPGNLBK
|
8.6 | IC50 | 2 | — | |
YIZTXYBSHMFWTH
|
8.6 | IC50 | 3 | — | |
BAPPLHACLUEZGL
|
8.6 | IC50 | 2 | — | |
CRDMJKIEIKHCSZ
|
8.6 | IC50 | 2 | — | |
DFKOCMIZZATJNQ
|
8.6 | IC50 | 3 | — |