Target Details
| UniProt AC | P11309 |
|---|---|
| Gene Symbol | PIM1 |
| Protein Name | Serine/threonine-protein kinase pim-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,647
- Clinical molecules 25
- Avg pChEMBL 8.21
KEGG Pathways (5)
Active Molecules (2,647)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
USIJRQBCKOPRCW
|
10.7 | IC50 | 3 | — | |
XCLYLGWPWSZDDN
|
10.7 | IC50 | 3 | — | |
XKCUAIJHVDEELV
|
10.7 | Ki | 3 | — | |
YIECCVSVKBACNI
|
10.7 | IC50 | 3 | — | |
YYOYATJEOKTTDV
|
10.7 | IC50 | 3 | — | |
ZBIYVIOSDQBGRR
|
10.7 | IC50 | 3 | — | |
OZGQEEVEYNXVFZ
|
10.7 | Ki | 3 | — | |
REZOXLPEJRXIEV
|
10.7 | Ki | 3 | — | |
ZAMFTNWEACEFAR
|
10.7 | Ki | 3 | — | |
FPBWUTAWSOLPQI
|
10.7 | Ki | 3 | — | |
SVYHADKWCWQANW
|
10.7 | Ki | 3 | — | |
IWSDHPXZBHZPMC
|
10.6 | Ki | 3 | — | |
JEVIKKKBDOXJFA
|
10.6 | Ki | 3 | — | |
CDQXYOYHHLAARJ
|
10.6 | Ki | 3 | — | |
OOWGEGYPCQGHJZ
|
10.6 | Ki | 3 | — | |
VPGFPXLEFFWPKW
|
10.6 | Ki | 3 | — | |
JEVIKKKBDOXJFA
|
10.6 | Ki | 3 | — | |
UXRGJORUNNVPFQ
|
10.5 | IC50 | 2 | — | |
IBNILFRNVFTCBR
|
10.5 | IC50 | 2 | — | |
BNXXSPKXSUAPBT
|
10.5 | IC50 | 3 | — | |
BQWJQWNJLHDQHB
|
10.5 | IC50 | 3 | — | |
CHPLSEJPLSDICK
|
10.5 | IC50 | 3 | — | |
DGJWAGBAIDNRCG
|
10.5 | IC50 | 3 | — | |
FIWUALBYNQLBJL
|
10.5 | IC50 | 3 | — | |
FIWUALBYNQLBJL
|
10.5 | IC50 | 3 | — | |
GRBWTTRGGLFQRT
|
10.5 | IC50 | 3 | — | |
JNOBBFHKVJLMIK
|
10.5 | IC50 | 3 | — | |
KFEFAUXTDOPDKJ
|
10.5 | IC50 | 2 | — | |
KFEFAUXTDOPDKJ
|
10.5 | IC50 | 2 | — | |
KGZCVPZUCOCCCQ
|
10.5 | IC50 | 3 | — | |
KRXHIAQHNCEJEE
|
10.5 | IC50 | 3 | — | |
LFSINWPISNIWOR
|
10.5 | Ki | 3 | — | |
MXLKCGYBUFWTAU
|
10.5 | IC50 | 3 | — | |
MYFHTAWVDSNJJK
|
10.5 | IC50 | 3 | — | |
NPLDOTMTVQWXCF
|
10.5 | IC50 | 3 | — | |
NWDVLGCDUFSSHA
|
10.5 | IC50 | 3 | — | |
NYMXZZBYJOQYQM
|
10.5 | IC50 | 3 | — | |
ORIUYOMCIQSKDJ
|
10.5 | IC50 | 3 | — | |
OSBCYEMTQYPIMH
|
10.5 | Ki | 3 | — | |
PUOWLWZDSDPHDN
|
10.5 | IC50 | 3 | — | |
ROWCDUKNAFYOMJ
|
10.5 | IC50 | 3 | — | |
UFRGVTREMFYICD
|
10.5 | IC50 | 3 | — | |
VGTXZFMBNSOWGX
|
10.5 | IC50 | 3 | — | |
XFUKFDJFEAQRRG
|
10.5 | Ki | 3 | — | |
YBENUWLHUXAJFZ
|
10.5 | Ki | 3 | — | |
BKZIXMFZEWLONB
|
10.5 | Ki | 3 | — | |
AQFQLFWVDMMENJ
|
10.5 | Ki | 3 | — | |
CIHVZVQWPVPVHJ
|
10.5 | Ki | 3 | — | |
CTADVIUFFUGUBU
|
10.5 | IC50 | 2 | — | |
OHXQPUAQXWTIOM
|
10.5 | Ki | 3 | — |