Target Details
| UniProt AC | P11309 |
|---|---|
| Gene Symbol | PIM1 |
| Protein Name | Serine/threonine-protein kinase pim-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,647
- Clinical molecules 25
- Avg pChEMBL 8.21
KEGG Pathways (5)
Active Molecules (2,647)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
VWHVWERPKXPYFT
|
8.7 | Ki | 3 | — | |
AJMRXXHYVHTIEV
|
8.7 | IC50 | 2 | — | |
FEIGOJWLHHRBHZ
|
8.7 | IC50 | 3 | — | |
LNIXAFUYUNLOOW
|
8.7 | Ki | 3 | — | |
LSRFJFLUAZLYAC
|
8.7 | IC50 | 2 | — | |
OFVSBWPTAOVFMJ
|
8.7 | IC50 | 2 | — | |
WAGFUTAXHIKUFA
|
8.7 | IC50 | 3 | — | |
YMZURUFTCLYPGO
|
8.7 | IC50 | 4 | — | |
ZTSKLXVSNKQDEN
|
8.7 | IC50 | 2 | — | |
DETSRRVOAOWTKK
|
8.7 | IC50 | 3 | — | |
KFQYYKRUXDSCRR
|
8.7 | Ki | 3 | — | |
SYEYZQUZNVVCNN
|
8.7 | IC50 | 3 | — | |
VMTDEYJXDXLJNT
|
8.7 | IC50 | 3 | — | |
ZZPSHDYFXGODPI
|
8.7 | Ki | 3 | — | |
ABUQYEHMIDSXIU
|
8.7 | IC50 | 2 | — | |
AHEMFHZQUVEVBH
|
8.7 | IC50 | 3 | — | |
AISMIGRIJQYZHW
|
8.7 | IC50 | 3 | — | |
ANXPRWZUQDZBMG
|
8.7 | IC50 | 2 | — | |
APHDIFQMSHEHKR
|
8.7 | IC50 | 2 | — | |
BQHHQEYEYHRNQA
|
8.7 | IC50 | 2 | — | |
BUHFIGHCARUNTG
|
8.7 | IC50 | 3 | — | |
BUMNKOYIRRNDAN
|
8.7 | IC50 | 2 | — | |
CAZNIOSROXHNKZ
|
8.7 | IC50 | 2 | — | |
CGBJYLPDYMUGJF
|
8.7 | IC50 | 3 | — | |
CGBJYLPDYMUGJF
|
8.7 | IC50 | 3 | — | |
CHSSIQHQGBQIEV
|
8.7 | IC50 | 2 | — | |
CNSKFROODZMZLE
|
8.7 | IC50 | 2 | — | |
CSYNBNGKBZGJAV
|
8.7 | IC50 | 3 | — | |
CUWBXIFJTGMJHU
|
8.7 | IC50 | 2 | — | |
DEIMIMRYYMEUNQ
|
8.7 | IC50 | 3 | — | |
DVZDOOQBSLUYLR
|
8.7 | IC50 | 2 | — | |
DZGZWWIIVUJLHY
|
8.7 | IC50 | 2 | — | |
FMYNFWDKPWRVHK
|
8.7 | Ki | 2 | — | |
FOCOGYAYQMQYQQ
|
8.7 | IC50 | 3 | — | |
GACLTRJMGHVCIN
|
8.7 | IC50 | 2 | — | |
GHBOTNLUBMTSJO
|
8.7 | IC50 | 3 | — | |
GXVGZXNLFFDMQG
|
8.7 | Ki | 2 | — | |
GZGLZFSLPIMAQV
|
8.7 | IC50 | 3 | — | |
GZGLZFSLPIMAQV
|
8.7 | IC50 | 3 | — | |
HIRGJKYVLHTQTI
|
8.7 | IC50 | 3 | — | |
HLVXBQWAULZBSW
|
8.7 | IC50 | 2 | — | |
HWNZDLXOJIRFFD
|
8.7 | IC50 | 3 | — | |
IRJSEURWZYHEFR
|
8.7 | IC50 | 3 | — | |
IXGVTTDCWVKAIV
|
8.7 | IC50 | 3 | — | |
JLGPSJZWENLOLE
|
8.7 | IC50 | 3 | — | |
KBIGMPDPPRLJPK
|
8.7 | IC50 | 3 | — | |
KOXBMECFAXSCGM
|
8.7 | IC50 | 3 | — | |
LFCJJXBBLSJUTJ
|
8.7 | IC50 | 4 | — | |
LQASHUDUJOBHMP
|
8.7 | IC50 | 3 | — | |
LYAZTMOXEBYWIS
|
8.7 | IC50 | 3 | — |