Target Details
| UniProt AC | P11309 |
|---|---|
| Gene Symbol | PIM1 |
| Protein Name | Serine/threonine-protein kinase pim-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,647
- Clinical molecules 25
- Avg pChEMBL 8.21
KEGG Pathways (5)
Active Molecules (2,647)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CMJKTDGFDREUGD
|
9.0 | IC50 | 2 | — | |
GDNKMWJOEGMBMT
|
9.0 | Ki | 3 | — | |
GEYAXZBDDHIAPF
|
9.0 | IC50 | 3 | — | |
JDVZPUBQXKOGSV
|
9.0 | IC50 | 2 | — | |
KCWAHDFNBQMGHB
|
9.0 | IC50 | 2 | — | |
KIPSRZQNNGSYJE
|
9.0 | IC50 | 3 | — | |
PWJMJGJCPRZTLY
|
9.0 | IC50 | 2 | — | |
QQCWPCSHFHPVFD
|
9.0 | IC50 | 2 | — | |
UCHPOAFBZQSXQS
|
9.0 | Ki | 3 | — | |
XDLZARQBWNHANQ
|
9.0 | IC50 | 2 | — | |
OBPOSYGZESRPFM
|
8.9 | IC50 | 3 | — | |
RMTGQRSHUXJNTH
|
8.9 | Ki | 3 | — | |
CJHZWEDFBINFAB
|
8.9 | Ki | 3 | — | |
YUJKLTZVCYEGQA
|
8.9 | Ki | 3 | — | |
BZUBDLKATGBRRF
|
8.9 | IC50 | 2 | — | |
DDALKELJNGHGGW
|
8.9 | IC50 | 2 | — | |
KIXOWPYWELTQEV
|
8.9 | IC50 | 2 | — | |
NOGKRZKIQYJCGB
|
8.9 | IC50 | 2 | — | |
OEXZILYFIBISBL
|
8.9 | IC50 | 2 | — | |
OLQLOEJZYFROOC
|
8.9 | IC50 | 2 | — | |
PJKHDASUTSMYOR
|
8.9 | IC50 | 2 | — | |
QQCWPCSHFHPVFD
|
8.9 | IC50 | 2 | — | |
SEZAIJZBNCLTIN
|
8.9 | IC50 | 2 | — | |
UIDMGDSJLAHUOJ
|
8.9 | Ki | 3 | — | |
VDJIRBSRWJZSCK
|
8.9 | Ki | 3 | — | |
ZBRMFNPKIONVTR
|
8.9 | IC50 | 3 | — | |
ZHCKQFBKXIHCHJ
|
8.9 | Ki | 3 | — | |
KWXMWYUQPYEECX
|
8.9 | IC50 | 2 | — | |
OEPCHHARAQRIEP
|
8.9 | Ki | 3 | — | |
VGHNUVDMAHSAAD
|
8.9 | IC50 | 2 | — | |
YKRVUDKGPNZLLY
|
8.9 | Ki | 3 | — | |
JJHPKDPBGCWUNR
|
8.9 | IC50 | 2 | — | |
MLMNRFXLMUJDHR
|
8.9 | IC50 | 2 | — | |
GIZDEODKRGICNS
|
8.9 | IC50 | 2 | — | |
HETPKWYRMKCRBF
|
8.9 | IC50 | 2 | — | |
HHWBOLGHDXDWCN
|
8.9 | IC50 | 2 | — | |
IXFNGWMOFJHECL
|
8.9 | IC50 | 2 | — | |
WFTKWNBPRXJBBC
|
8.9 | IC50 | 2 | — | |
XYDAVXLWFUQNSH
|
8.9 | IC50 | 7 | — | |
JIRRCQJZLNTIIP
|
8.9 | IC50 | 3 | — | |
LLNUQZVEPPOXBC
|
8.9 | IC50 | 2 | — | |
RBZKPGNGBLPBJZ
|
8.9 | IC50 | 2 | — | |
UVJRFPDIIZDNQE
|
8.9 | IC50 | 3 | — | |
BRWANDFSFFFOPJ
|
8.9 | IC50 | 3 | — | |
FUOLJDPZDKQMEX
|
8.9 | IC50 | 2 | — | |
XNQLYGHTCMOZRQ
|
8.9 | IC50 | 3 | — | |
BMRHAWSJNXXRJI
|
8.8 | IC50 | 2 | — | |
CUEWSGPOORVNOX
|
8.8 | IC50 | 2 | — | |
DFPNYFLFFOGKAB
|
8.8 | IC50 | 2 | — | |
RDWOPOGQJJCJBX
|
8.8 | IC50 | 3 | — |