Target Details
| UniProt AC | P11309 |
|---|---|
| Gene Symbol | PIM1 |
| Protein Name | Serine/threonine-protein kinase pim-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,647
- Clinical molecules 25
- Avg pChEMBL 8.21
KEGG Pathways (5)
Active Molecules (2,647)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KDKNXCUSRALRIT
|
9.0 | IC50 | 3 | — | |
KKLILNOZODIJCA
|
9.0 | IC50 | 3 | — | |
KMEWOQDIZJORND
|
9.0 | IC50 | 3 | — | |
LCPFTSAYXQZOCT
|
9.0 | IC50 | 3 | — | |
LHUASYMEOPGJLS
|
9.0 | IC50 | 3 | — | |
LQASHUDUJOBHMP
|
9.0 | IC50 | 3 | — | |
LRQKBAQIKBSJAJ
|
9.0 | IC50 | 3 | — | |
MBDRYNIIESDGQW
|
9.0 | IC50 | 2 | — | |
MFQHDSGLLLJSPV
|
9.0 | IC50 | 3 | — | |
MHYXMWPAQOHZQD
|
9.0 | IC50 | 3 | — | |
MQUXRVLSWBLTHR
|
9.0 | IC50 | 3 | — | |
MXGJFGVAPMJHRD
|
9.0 | IC50 | 3 | — | |
NENYUFKIMYPYBK
|
9.0 | IC50 | 3 | — | |
NEORABJLFZZFEQ
|
9.0 | IC50 | 2 | — | |
NHIRQUMDHFNSGY
|
9.0 | IC50 | 3 | — | |
NLKQVIFMDOOBRW
|
9.0 | IC50 | 3 | — | |
NPIIOAIPYXDRBZ
|
9.0 | IC50 | 3 | — | |
NTFBHHYDVVRATP
|
9.0 | IC50 | 2 | — | |
NYJVWPXVQNSSLU
|
9.0 | IC50 | 2 | — | |
ODZZYKUYGVLOTQ
|
9.0 | IC50 | 3 | — | |
PAWYDNPYJNAJHA
|
9.0 | IC50 | 3 | — | |
PAWYDNPYJNAJHA
|
9.0 | IC50 | 3 | — | |
PBYQNLORWAKJIE
|
9.0 | IC50 | 2 | — | |
PKHXAHNPTNZSSF
|
9.0 | IC50 | 3 | — | |
POOGYHHHUWNODC
|
9.0 | IC50 | 2 | — | |
PPYABCSZOJIKBY
|
9.0 | IC50 | 3 | — | |
PYVZMEJFWXPRBE
|
9.0 | IC50 | 3 | — | |
QBDOORMZDCRUOU
|
9.0 | IC50 | 3 | — | |
QFGXSSFSKIVBOP
|
9.0 | IC50 | 3 | — | |
QGXLCQREBIFJLA
|
9.0 | IC50 | 3 | — | |
QJWGSVNGDURFSA
|
9.0 | IC50 | 3 | — | |
QKUWPBOCGZKIAG
|
9.0 | IC50 | 2 | — | |
QLEWJDQBRAZQMH
|
9.0 | IC50 | 3 | — | |
QPKIGRQFGZEZBT
|
9.0 | IC50 | 2 | — | |
QQKNGMZFTNVAKG
|
9.0 | IC50 | 2 | — | |
QSNACFYJEZLGIS
|
9.0 | IC50 | 3 | — | |
QTLYBRKPIYULQQ
|
9.0 | IC50 | 3 | — | |
QVAKUYTZVMRSAG
|
9.0 | IC50 | 3 | — | |
QVCLVTVRXGXXOR
|
9.0 | Ki | 4 | — | |
QYKGYRLGHZIFTF
|
9.0 | IC50 | 3 | — | |
QZYGPBINVRPXPJ
|
9.0 | IC50 | 2 | — | |
RDPIVXMVUFXNIS
|
9.0 | Ki | 2 | — | |
ROJUIQFJWVBSKO
|
9.0 | IC50 | 3 | — | |
SBJPEYLIYCCZOA
|
9.0 | IC50 | 3 | — | |
SDSSZBQMUURFEC
|
9.0 | IC50 | 3 | — | |
SKRRMVNHSWITRS
|
9.0 | IC50 | 2 | — | |
SKYIOLUXCWYHKN
|
9.0 | IC50 | 3 | — | |
SMKDKOFQQMLFPP
|
9.0 | IC50 | 3 | — | |
SMKDKOFQQMLFPP
|
9.0 | IC50 | 3 | — | |
SOVGWUJZYLFKDZ
|
9.0 | Ki | 3 | — |