Target Details
| UniProt AC | P11309 |
|---|---|
| Gene Symbol | PIM1 |
| Protein Name | Serine/threonine-protein kinase pim-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,647
- Clinical molecules 25
- Avg pChEMBL 8.21
KEGG Pathways (5)
Active Molecules (2,647)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
CTMMAHRPYPQKSU
|
9.0 | IC50 | 3 | — | |
CYDDMCKGRSYSNW
|
9.0 | IC50 | 2 | — | |
DDPVTMQONNFZAJ
|
9.0 | IC50 | 3 | — | |
DFIJYMKITRKPIH
|
9.0 | IC50 | 3 | — | |
DFXMBRWAQKZCBG
|
9.0 | IC50 | 2 | — | |
DOFPZEPZLPYGKA
|
9.0 | IC50 | 3 | — | |
DQUAKDWLLPATPK
|
9.0 | IC50 | 3 | — | |
DRSGGAHSPDXOOW
|
9.0 | IC50 | 3 | — | |
DSUSEZJHVSEHGF
|
9.0 | IC50 | 2 | — | |
DSUSEZJHVSEHGF
|
9.0 | IC50 | 2 | — | |
FAHDUHMZUVZGJA
|
9.0 | IC50 | 3 | — | |
FCGLYPSBPNFQRF
|
9.0 | IC50 | 3 | — | |
FDCZCIGFGKWALA
|
9.0 | Ki | 2 | — | |
FLESDXZVGOIBKK
|
9.0 | IC50 | 3 | — | |
FNKRKMGPGVJYDC
|
9.0 | IC50 | 3 | — | |
FTEJBTVRJIRRSV
|
9.0 | IC50 | 3 | — | |
FUCDNRWEBGAXAG
|
9.0 | IC50 | 3 | — | |
FUGPTCJAZZYCRJ
|
9.0 | IC50 | 2 | — | |
FXKAJMTVSSOIMV
|
9.0 | IC50 | 2 | — | |
GACLTRJMGHVCIN
|
9.0 | IC50 | 2 | — | |
GACLTRJMGHVCIN
|
9.0 | IC50 | 2 | — | |
GHBOTNLUBMTSJO
|
9.0 | IC50 | 3 | — | |
GNTIXZIMEPMGMD
|
9.0 | IC50 | 3 | — | |
GOYXKJXQXYESKZ
|
9.0 | IC50 | 3 | — | |
GXZGFGZOTUWEPA
|
9.0 | IC50 | 2 | — | |
HDYFVAJZXGMYBL
|
9.0 | IC50 | 2 | — | |
HFUZHVLXCKATBR
|
9.0 | IC50 | 3 | — | |
HIPDXMYHALNOCD
|
9.0 | IC50 | 3 | — | |
HIRGJKYVLHTQTI
|
9.0 | IC50 | 3 | — | |
HIRGJKYVLHTQTI
|
9.0 | IC50 | 3 | — | |
HMFMRXDOISLKHG
|
9.0 | IC50 | 3 | — | |
HQZZLYFXAGRMNB
|
9.0 | IC50 | 3 | — | |
HSAKWLGNZJVJCZ
|
9.0 | IC50 | 3 | — | |
IBJNNOBWKBCHNX
|
9.0 | IC50 | 2 | — | |
IDHYALMZKJRNKP
|
9.0 | IC50 | 2 | — | |
IDPLHVZCGVXEDH
|
9.0 | IC50 | 3 | — | |
IFDWSONRKKYDJB
|
9.0 | IC50 | 3 | — | |
ISSQSUGBRMTNBJ
|
9.0 | IC50 | 3 | — | |
IUBIAVFVWYAABB
|
9.0 | IC50 | 3 | — | |
IZLJTEJHPGSEBB
|
9.0 | IC50 | 3 | — | |
JAIGOJJTHHSCML
|
9.0 | IC50 | 3 | — | |
JDXDVNMKQNFAFD
|
9.0 | IC50 | 3 | — | |
JDXDVNMKQNFAFD
|
9.0 | IC50 | 3 | — | |
JPLWJJBURUCINP
|
9.0 | IC50 | 2 | — | |
JRMXORAYSQPTMU
|
9.0 | IC50 | 3 | — | |
JSWXHRIKDWHCOW
|
9.0 | IC50 | 3 | — | |
JVFOBBPBZAGJLA
|
9.0 | IC50 | 3 | — | |
JVTKKKZABXBICW
|
9.0 | IC50 | 3 | — | |
JXINSHNJIUKPKA
|
9.0 | IC50 | 3 | — | |
JXVXKOPUJQFJEO
|
9.0 | Ki | 3 | — |