Target Details
| UniProt AC | P11309 |
|---|---|
| Gene Symbol | PIM1 |
| Protein Name | Serine/threonine-protein kinase pim-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,647
- Clinical molecules 25
- Avg pChEMBL 8.21
KEGG Pathways (5)
Active Molecules (2,647)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RQGHKTDVDKITFW
|
9.1 | IC50 | 2 | — | |
SLGWCOFFSAFFES
|
9.1 | Ki | 3 | — | |
SNCXKOCIPWPVQA
|
9.1 | Ki | 3 | — | |
TXTDGNUYTBBPSP
|
9.1 | IC50 | 3 | — | |
XQTDEFZROIJVJH
|
9.1 | IC50 | 2 | — | |
ZTITWEKKRIDSCW
|
9.1 | IC50 | 2 | — | |
AWBJVQCGEWMAGP
|
9.1 | Ki | 3 | — | |
OSHOEUXWOYAJAL
|
9.1 | IC50 | 2 | — | |
URRUOKGGTGKOSU
|
9.1 | Ki | 3 | — | |
PDIITFZVMNMSSW
|
9.1 | IC50 | 2 | — | |
DUROCBBMWRCUSH
|
9.1 | IC50 | 3 | — | |
QEULBJUCNBXCDE
|
9.1 | Ki | 3 | — | |
KSUJTDNWWVQOFC
|
9.1 | Ki | 3 | — | |
UPNOOQUTVLYBIK
|
9.1 | Ki | 3 | — | |
VHIOBYUNOHKXFT
|
9.1 | IC50 | 2 | — | |
XISLSWZWVQRULG
|
9.1 | IC50 | 3 | — | |
AXLWBOXIQLKYIT
|
9.1 | IC50 | 2 | — | |
GLCSICZREVNVTH
|
9.1 | IC50 | 2 | — | |
LCLHYQYLXQMIBR
|
9.1 | Ki | 3 | — | |
LEGBCPZPNSHFKW
|
9.1 | IC50 | 3 | — | |
OYFIIXZMOKZCBZ
|
9.1 | IC50 | 2 | — | |
PDRMZIBUTGMDNS
|
9.1 | IC50 | 2 | — | |
RLPCQQSZTQVWAR
|
9.1 | Ki | 2 | — | |
SVRMTQIVKSSINT
|
9.1 | IC50 | 2 | — | |
SWHCYMNTFSKTIE
|
9.1 | IC50 | 2 | — | |
YZUVSHPJGNXWDS
|
9.1 | IC50 | 2 | — | |
QSZOWBXCZPNMQY
|
9.0 | Ki | 3 | — | |
KFMIHULBBWHKPZ
|
9.0 | IC50 | 3 | — | |
NRWVKWOODSLDFZ
|
9.0 | Ki | 3 | — | |
KSUJTDNWWVQOFC
|
9.0 | Ki | 3 | — | |
LIKKMSJYXQMOCX
|
9.0 | IC50 | 2 | — | |
NNCWGHBKJIEMSS
|
9.0 | IC50 | 2 | — | |
WJXBLZWJWGLQLR
|
9.0 | Ki | 3 | — | |
AGZJSRNQZKATFR
|
9.0 | IC50 | 3 | — | |
AISMIGRIJQYZHW
|
9.0 | IC50 | 3 | — | |
ATNCLUHEGCYVPT
|
9.0 | IC50 | 3 | — | |
BGFPXHMHXQXNPY
|
9.0 | IC50 | 3 | — | |
BKUXTVCORRDHGA
|
9.0 | IC50 | 3 | — | |
BLBAWGODFTZAEY
|
9.0 | IC50 | 2 | — | |
BOYINUVWSRXXKU
|
9.0 | IC50 | 3 | — | |
BQGUIXOMELYYIP
|
9.0 | IC50 | 3 | — | |
BRURCCZOEKNNPP
|
9.0 | IC50 | 3 | — | |
BTGLPUGPEBTEHU
|
9.0 | IC50 | 3 | — | |
BZURHWWJXUKIOZ
|
9.0 | IC50 | 3 | — | |
CBZNDVANLGVAAJ
|
9.0 | IC50 | 2 | — | |
CGBJYLPDYMUGJF
|
9.0 | IC50 | 3 | — | |
CGBJYLPDYMUGJF
|
9.0 | IC50 | 3 | — | |
COZNGJFVGMJIHO
|
9.0 | IC50 | 2 | — | |
CPHAAKSWOQSYIW
|
9.0 | Ki | 3 | — | |
CSMNPMNSCMKFAN
|
9.0 | IC50 | 3 | — |