Target Details
| UniProt AC | P11309 |
|---|---|
| Gene Symbol | PIM1 |
| Protein Name | Serine/threonine-protein kinase pim-1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) |
Summary
- Multi-target molecules 2,647
- Clinical molecules 25
- Avg pChEMBL 8.21
KEGG Pathways (5)
Active Molecules (2,647)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XGCMEAHEGFLCSF
|
9.2 | IC50 | 2 | — | |
DPNYLXBQKCMOTA
|
9.2 | IC50 | 2 | — | |
KFEFAUXTDOPDKJ
|
9.2 | IC50 | 2 | — | |
KGWJXHXHZOYSEQ
|
9.2 | Ki | 3 | — | |
NZTGSWDBRZMTBV
|
9.2 | IC50 | 2 | — | |
YRYBUDFRAMZDPV
|
9.2 | IC50 | 2 | — | |
GNAXCGUONRASLS
|
9.2 | Ki | 3 | — | |
ZHCCGWZBLZBPDY
|
9.2 | IC50 | 2 | — | |
ABZNMUCRZXRUAU
|
9.2 | IC50 | 2 | — | |
ACVSVHBGMBCOLQ
|
9.2 | IC50 | 2 | — | |
ATMGNNLRUXSWJM
|
9.2 | Ki | 3 | — | |
FARRIJSECFVEQS
|
9.2 | IC50 | 2 | — | |
GACLTRJMGHVCIN
|
9.2 | IC50 | 2 | — | |
HQKQOEMBHUHWCM
|
9.2 | IC50 | 2 | — | |
IANCYKFILINNSQ
|
9.2 | IC50 | 3 | — | |
JAVVLMYHUYZZDN
|
9.2 | IC50 | 3 | — | |
JEKGYBBSKUISTO
|
9.2 | IC50 | 2 | — | |
JRPMCVBHTMZOFM
|
9.2 | IC50 | 2 | — | |
JRPMCVBHTMZOFM
|
9.2 | IC50 | 2 | — | |
MKTNFHCTEKGLHY
|
9.2 | IC50 | 3 | — | |
MPFTYTXJRHGYBP
|
9.2 | IC50 | 2 | — | |
OJYVFIGZGJDMSR
|
9.2 | IC50 | 2 | — | |
QFYWUMPWXIJTRE
|
9.2 | IC50 | 2 | — | |
UPKYTOHUEMELIK
|
9.2 | Ki | 3 | — | |
VLOSGHYSCVRVJH
|
9.2 | IC50 | 2 | — | |
VPLXMHRCNSVLNX
|
9.2 | IC50 | 2 | — | |
XDZHNVNYIFINOV
|
9.2 | Ki | 3 | — | |
YXICKOJWVBGVKW
|
9.2 | Ki | 3 | — | |
HXUHHDBYIBYXPB
|
9.1 | IC50 | 3 | — | |
LHNFUMPDPUCZHQ
|
9.1 | IC50 | 2 | — | |
SDHGIPREFAWIKS
|
9.1 | Ki | 3 | — | |
WIPFTCGFZZZMDW
|
9.1 | IC50 | 2 | — | |
XIIRJPVKFJFUHB
|
9.1 | Ki | 3 | — | |
ZOHXDWMYFQLOMC
|
9.1 | Ki | 3 | — | |
CDPLNEIWXMADGF
|
9.1 | Ki | 3 | — | |
CHFXZLZGCMQMBM
|
9.1 | IC50 | 3 | — | |
GANFQJFXZYPGOX
|
9.1 | IC50 | 2 | — | |
NUMGAHMZNWRORP
|
9.1 | Ki | 3 | — | |
QVRUMXAVDBYHBP
|
9.1 | IC50 | 3 | — | |
HLPARXMUJBJYFM
|
9.1 | IC50 | 3 | — | |
NRDBSOIRIVKMSF
|
9.1 | Ki | 3 | — | |
VZRTVWNQRPJJJV
|
9.1 | IC50 | 2 | — | |
WJXBLZWJWGLQLR
|
9.1 | Ki | 3 | — | |
FRANNCVVJFQWOT
|
9.1 | IC50 | 3 | — | |
KYPWRLVQGWQNEA
|
9.1 | IC50 | 3 | — | |
LLCBENGUWIODIZ
|
9.1 | IC50 | 2 | — | |
OLLSIGPBXQELDV
|
9.1 | Ki | 2 | — | |
PWDDNCBQYVPPFY
|
9.1 | Ki | 3 | — | |
QDMRXIVSBQLTQK
|
9.1 | IC50 | 2 | — | |
RKNBXYNQXGECFV
|
9.1 | IC50 | 2 | — |